武汉永璨生物科技有限公司
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
搜索
首页
网站地图
产品名字索引 A
按首字母搜索
A
B
C
D
E
F
G
H
I
J
K
L
M
N
O
P
Q
R
S
T
U
V
W
X
Y
Z
1
2
3
4
5
6
7
8
9
«
1
2
3
4
5
6
7
8
9
10
»
产品名字索引 A
AMG-510 racemate
(Catalog# : 112194, Cas# :
2252403-56-6
)
AMG-510 is a potent KRAS G12C covalent inhibitor. AMG-510 selectively targets the KRA
Aprocitentan
(Catalog# : 112191, Cas# :
1103522-45-7
)
Aprocitentan is an orally active, dual endothelin (ET) receptor antagonist developed
Aramchol
(Catalog# : 6111903, Cas# :
246529-22-6
)
From:https://galmedpharma.com/about-aramchol/Aramchol(arachidyl amido cholanoic aci
阿拉酸式苯
(Catalog# : 513191, Cas# :
35272-27-6
)
benzo[d][1,2,3]thiadiazole-7-carboxylic acid,Acibenzolar acid,CGA 210 007
AR-C155858
(Catalog# : 193291, Cas# :
496791-37-8
)
AR-C155858是一种强效的单羧酸转运蛋白MCT1和MCT2的抑制剂,它与细胞
ACT-709478
(Catalog# : 193288, Cas# :
1838651-58-3
)
ACT-709478是一种强效、选择性的T型钙通道阻滞剂,是治疗全身性癫
A1874
(Catalog# : 193287, Cas# :
2064292-12-0
)
A1874是一种以核桃仁为基础的,BRD4降解的丙交酯,诱导BRD4在细胞
AZD9567
(Catalog# : 193254, Cas# :
1893415-00-3
)
AZD9567是一种口服分化非甾体选择性糖皮质激素受体调节剂(SGRM)。
AZ1495
(Catalog# : 193222, Cas# :
2196204-23-4
)
AZ1495是一种有效且具有选择性的IRAK4抑制剂。
ATR-101盐酸盐
(Catalog# : 193208, Cas# :
133825-81-7
)
ATR-101,也被称为PD-132301 (游离)或PD-132301-2 (盐酸盐),正在临床开发
ARN-3236
(Catalog# : 193192, Cas# :
1613710-01-2
)
ARN-3236是一种强效、口服活性和选择性的SIK2抑制剂。在攻击- 3236抑
ARN 077
(Catalog# : 193134, Cas# :
1373625-34-3
)
ARN 077是一种强效选择性N -乙酰乙醇胺酸酰胺酶(NAAA)抑制剂,IC50为
阿格列扎
(Catalog# : 193125, Cas# :
475479-34-6
)
阿格列扎, 也称为RG-1439或RO-0728804,是一个过氧物酶体增生激活受
Alvimopan
(Catalog# : 19382, Cas# :
156053-89-3
)
Alvimopan,也称为HSDB-7704和LY246736, 是一种作为一个次要地行动的μ-
Abrocitinib
(Catalog# : 19381, Cas# :
1622902-68-4
)
Abrocitinib(PF-04965842)是Pifzer研发的是一种Janus激酶抑制剂药物,目
AA26-9
(Catalog# : 19372, Cas# :
1312782-34-5
)
AA26-9是一种高效广谱丝氨酸水解酶抑制剂。AA26 -9抑制酶来源于丝
AZD-0284
(Catalog# : 19365, Cas# :
2101291-07-8
)
AZD-0284是一种强有力的、有选择性的反兴奋剂,可以潜在治疗核受
AZ304
(Catalog# : 19363, Cas# :
942507-42-8
)
AZ304是一种ATP-竞争性双BRAF激酶抑制剂,对野生型BRAF、V600E突变型
AZ876
(Catalog# : 19356, Cas# :
898800-26-5
)
AZ876,又称AZ-876,是一种肝脏X受体激动剂。AZ876可预防病理性心肌
AGN-190299
(Catalog# : 19316, Cas# :
118292-41-4
)
Tazarotene是一种视黄醇类前体药物,通过在动物和人体内的快速脱
AM281
(Catalog# : 19315, Cas# :
202463-68-1
)
AM281是一种合成大麻素CB1受体拮抗剂。
ASP9521
(Catalog# : 19312, Cas# :
1126084-37-4
)
ASP9521是日常的,选择性,口服生物利用率17β-羟甾类脱氢酶的抑制
AZD0364
(Catalog# : 192275, Cas# :
2097416-76-5
)
AZD0364是一种用于治疗癌症的ERK1和/或ERK2激酶。ERK1和ERK2激酶是广泛
ATF6-活化剂-147
(Catalog# : 192212, Cas# :
393121-74-9
)
ATF6-activator-147是一种ATF6模拟器,它作为一种前体药物,通过一种
AZD1152
(Catalog# : 192156, Cas# :
722543-31-9
)
AZD1152是Barasertib-hQPA的前药,是一种高选择性极光B抑制剂,在无细
AZD3229
(Catalog# : 191287, Cas# :
2248003-60-1
)
AZD3229是治疗胃肠道间质瘤的一种有效的pan-kit突变抑制剂。AZD3229在
AM095钠
(Catalog# : 191251, Cas# :
1345614-59-6
)
AM095是一个强有力的LPA1受体拮抗剂,因为它抑制GTPγS绑定中国仓鼠
AZD4573
(Catalog# : 191212, Cas# :
2057509-72-3
)
AZD-4573是一种选择性的丝氨酸/苏氨酸依赖性激酶9 (CDK9)的短期抑制
AR-9281
(Catalog# : 191146, Cas# :
913548-29-5
)
AR-9281是一种可溶性环氧化物水解酶(s-EH)抑制剂,有望用于高血压
ARRY-797 (ARRY-371797)
(Catalog# : 191112, Cas# :
1036404-17-7
)
ARRY-797(CAS1036404-17-7) is an oral, selective p38 mitogen-activated protein kinase
«
1
2
3
4
5
6
7
8
9
10
»
产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
PLX8394
(Catalog# : 20613, Cas# :
1393466-87-9
)
PLX8394 is an orally bioavailable inhibitor of serine/threonine-protein kinase B-raf
Zelasudil
(Catalog# : 24014, Cas# :
2365193-22-0
)
Zelasudil 是一种有效的、高选择性的口服活性抑制剂,针对 Rho 相关
Ziftomenib ( KO-539 )
(Catalog# : 24013, Cas# :
2134675-36-6
)
Ziftomenib 是一种口服、有效、选择性的小分子抑制剂,针对 menin 和
Zunsemetinib
(Catalog# : 24012, Cas# :
1640282-42-3
)
Zunsemetinib是一种在研口服丝裂原活化蛋白激酶活化蛋白激酶2(MK2
Zongertinib ( BI 1810631 )
(Catalog# : 24011, Cas# :
2728667-27-2
)
Zongertinib [BI 1810631] 是一种人表皮生长因子受体 2 (HER2) 抑制剂。
Zasocitinib
(Catalog# : 24010, Cas# :
2272904-53-5
)
Zasocitinib是一种作用于非受体酪氨酸蛋白激酶 (TYK2)靶点的抑制
RNK-05047
(Catalog# : 24008, Cas# :
2503036-46-0
)
RNK-05047 为BRD4降解剂,其在小鼠荷瘤异种移植模型中展现出显著抑
Asengeprast (FT011)
(Catalog# : 24009, Cas# :
1001288-58-9
)
Asengeprast (FT011) 是一种抗纤维化剂,降低胶原蛋白 I 和 III 的 mRNA
ERAS-801 ( JGK-068S )
(Catalog# : 20635, Cas# :
2490431-16-6
)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。
T-1095
(Catalog# : 24004, Cas# :
209746-59-8
)
T-1095 is a potent and selective inhibitor of Na+-glucose cotransporters (SGLTs).