武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
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订购信息
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产品名字索引 A
Asciminib ( ABL001 )
(Catalog# : 1711222, Cas# :
1492952-76-7
)
Asciminib, 也叫ABL001,是一种有效的BCR-ABL的变构抑制剂。ABL001在与尼
Autophinib
(Catalog# : 17101617, Cas# :
1644443-47-9
)
Autophinib是一种新颖有效的自噬抑制剂,抑制通过靶向脂质激酶VPS
Adarigiline
(Catalog# : 1710167, Cas# :
1124197-79-0
)
adarigiline是单胺氧化酶B抑制剂的候选药物。
Adafosbuvir
(Catalog# : 1710166, Cas# :
1613589-09-5
)
Adafosbuvir是一种抗病毒药物。
AZD-5153 HNT salt
(Catalog# : 1710161, Cas# :
1869912-40-2
)
AZD-5153 HNT盐,是AZD-5153的6-hydroxy-2-naphthoic酸盐。AZD-5153对抗血液系
ABT-100
(Catalog# : 1710131, Cas# :
450839-40-4
)
abt-100是一种口服的法尼基转移酶抑制剂.
阿西鲁司特
(Catalog# : 179159, Cas# :
943764-99-6
)
阿西鲁司特,也称为ZK322,是强有力的和有选择性的白三烯A4水解酶
AR-7
(Catalog# : 179158, Cas# :
80306-38-3
)
AR-7,亦称非典型维甲酸7,是一种有效的和选择性的自噬(CMA)增
阿地米屈
(Catalog# : 179151, Cas# :
1675-66-7
)
阿地米屈是壬二酸的合成酰胺衍生物,具有对称的化学结构。它被
AZD7545
(Catalog# : 179136, Cas# :
252017-04-2
)
AZD7545是丙酮酸脱氢酶激酶2抑制剂(pdhk2)(对6.4nm IC50值)用于治
AMG-9810
(Catalog# : 179117, Cas# :
545395-94-6
)
AMG 9810是对香草类受体1的辣椒素激活竞争性拮抗剂(TRPV1)。此外
AS-2444697 HCl
(Catalog# : 179832, Cas# :
1287665-60-4
)
AS-2444697是一种 RAK-4抑制剂。六周重复给药AS2444697(0.3-3mg/kg,一天
乙酰卡尼盐酸盐
(Catalog# : 179829, Cas# :
34118-92-8
)
乙酰卡尼,又名N-乙酰普鲁卡因胺和ASL 601,普鲁卡因胺是N-乙酰化
ASC-J9
(Catalog# : 179816, Cas# :
52328-98-0
)
ASC-J9,也称为GO-Y025和去甲氧基姜黄素,是一个AR降解剂,ASC-J9通过
AMG-009
(Catalog# : 17987, Cas# :
1027847-67-1
)
AMG 009是一种口服活性小分子CRTH2受体(趋化受体的同源分子表达在
5-氨基-2-氟-4-甲基苯腈
(Catalog# : 1781603, Cas# :
1426136-04-0
)
5-氨基-2-氟-4-甲基苯腈,5-amino-2-fluoro-4-methylbenzonitrile
2-azaspiro[3.5]nonan-7-ol hydrochloride
(Catalog# : 1781602, Cas# :
1434141-67-9
)
2-azaspiro[3.5]nonan-7-ol hydrochloride
AZD3264
(Catalog# : 178910, Cas# :
1609281-86-8
)
AZD3264是一种新型的小分子IKK2抑制剂。IKK2作为IB激酶的蛋白质亚基
A-971432
(Catalog# : 178816, Cas# :
1240308-45-5
)
A - 971432对S1P5具有高度选择性,在临床前口服剂量后,显露出良好
A-1165442
(Catalog# : 20178812, Cas# :
1221443-94-2
)
A-1165442是一种中性温度具有止痛功效的瞬时受体电位香草酸亚型1
AZD4205
(Catalog# : 20178710, Cas# :
2091134-35-7
)
AZD4205是一种高效JAK1-选择性激酶抑制剂,拥有优秀的临床前药代动
ACY-775
(Catalog# : 77821, Cas# :
1375466-18-4
)
ACY-775是一种组蛋白去乙酰化酶6(HDAC6)选择性抑制剂。
AAI-101
(Catalog# : 1773101, Cas# :
1001404-83-6
)
AAI101(AAI101)是一种新型的增谱-乳酸酶抑制剂。AAI101(AAI101)与头孢吡
AV-412甲苯磺酸盐
(Catalog# : 17030105, Cas# :
451493-31-5
)
AV-412,也称为MP-412,是第二代生物可利用的双激酶抑制剂,具有潜在
AZD-7594
(Catalog# : 17022812, Cas# :
1196509-60-0
)
AZD-7594,也叫AZ13189620,是一种吸入选择性糖皮质激素受体(GCCR)调制
AZD3839
(Catalog# : 17022710, Cas# :
1227163-56-5
)
AZD3839是一种有效的选择性BACE1抑制剂。AZD3839是治疗阿尔茨海默病
A-1210477
(Catalog# : 17022404, Cas# :
1668553-26-1
)
A-1210477是一种有效、选择性的MCL-1抑制剂。
阿帕替尼
(Catalog# : 17022301, Cas# :
811803-05-1
)
阿帕替尼是一种具有生物口服、选择性的IC50为1 nM的VEGFR2 抑制剂。
硫酸阿米卡星
(Catalog# : 17021407, Cas# :
39831-55-5
)
硫酸阿米卡星(BAY416651 硫酸)是一种由卡那霉素a衍生的半合成氨基
AFN-1252
(Catalog# : 17021406, Cas# :
620175-39-5
)
AFN-1252(Debio 1452) 是enoyl -酰基载体蛋白还原酶(FabI)的有效抑制剂。
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
QBS10072S
(Catalog# : 25190, Cas# :
1802735-28-9
)
QBS10072S 是一种血脑屏障 (BBB) 渗透剂,由细胞毒性化疗结构域 N-双
TAK-071
(Catalog# : 186269, Cas# :
1820812-16-5
)
TAK-071 是一种毒蕈碱 M1 受体正变构调节剂。
MTX115325
(Catalog# : 186264, Cas# :
2750895-97-5
)
MTX115325是一种强效、选择性、脑渗透性USP30抑制剂,具有良好的类
LY-3381916
(Catalog# : 193123, Cas# :
2166616-75-5
)
LY-3381916是一种强效的、选择性的、脑透性的IDO1活性抑制剂,与缺
Opakalim
(Catalog# : 25193, Cas# :
2376397-93-0
)
Opakalim(BHV-7000)是Kv7.2/7.3钾通道(KCNQ2/3)的口服小分子激活剂,
DS68591889
(Catalog# : 25158, Cas# :
2488609-21-6
)
DS68591889 (PTDSS1i) 特异性抑制 PTDSS1,而 PTDSS1 可催化丝氨酸掺入 PC。
CAY 10566
(Catalog# : 10403, Cas# :
944808-88-2
)
CAY 10566是一种强效的选择性SCD-1抑制剂。
Cadefrecitinib (GLPG-3667)
(Catalog# : 20509, Cas# :
2308520-97-8
)
Cadefrecitinib(GLPG-3667)是一种口服小分子TYK2激酶抑制剂,目前正处
Dencatistat (STP938)
(Catalog# : 25177, Cas# :
2377000-84-3
)
Dencatistat 是一种口服生物可利用的小分子胞苷三磷酸合酶 1 (CTPS1)
DS-1001b
(Catalog# : 25178, Cas# :
1898207-64-1
)
DS-1001 是一种口服的脑渗透性突变 IDH1 选择性抑制剂。