武汉永璨生物科技有限公司
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
搜索
首页
网站地图
产品名字索引 A
按首字母搜索
A
B
C
D
E
F
G
H
I
J
K
L
M
N
O
P
Q
R
S
T
U
V
W
X
Y
Z
1
2
3
4
5
6
7
8
9
«
2
3
4
5
6
7
8
9
10
11
»
产品名字索引 A
AR-7
(Catalog# : 179158, Cas# :
80306-38-3
)
AR-7,亦称非典型维甲酸7,是一种有效的和选择性的自噬(CMA)增
阿地米屈
(Catalog# : 179151, Cas# :
1675-66-7
)
阿地米屈是壬二酸的合成酰胺衍生物,具有对称的化学结构。它被
AZD7545
(Catalog# : 179136, Cas# :
252017-04-2
)
AZD7545是丙酮酸脱氢酶激酶2抑制剂(pdhk2)(对6.4nm IC50值)用于治
AMG-9810
(Catalog# : 179117, Cas# :
545395-94-6
)
AMG 9810是对香草类受体1的辣椒素激活竞争性拮抗剂(TRPV1)。此外
AS-2444697 HCl
(Catalog# : 179832, Cas# :
1287665-60-4
)
AS-2444697是一种 RAK-4抑制剂。六周重复给药AS2444697(0.3-3mg/kg,一天
乙酰卡尼盐酸盐
(Catalog# : 179829, Cas# :
34118-92-8
)
乙酰卡尼,又名N-乙酰普鲁卡因胺和ASL 601,普鲁卡因胺是N-乙酰化
ASC-J9
(Catalog# : 179816, Cas# :
52328-98-0
)
ASC-J9,也称为GO-Y025和去甲氧基姜黄素,是一个AR降解剂,ASC-J9通过
AMG-009
(Catalog# : 17987, Cas# :
1027847-67-1
)
AMG 009是一种口服活性小分子CRTH2受体(趋化受体的同源分子表达在
5-氨基-2-氟-4-甲基苯腈
(Catalog# : 1781603, Cas# :
1426136-04-0
)
5-氨基-2-氟-4-甲基苯腈,5-amino-2-fluoro-4-methylbenzonitrile
2-azaspiro[3.5]nonan-7-ol hydrochloride
(Catalog# : 1781602, Cas# :
1434141-67-9
)
2-azaspiro[3.5]nonan-7-ol hydrochloride
AZD3264
(Catalog# : 178910, Cas# :
1609281-86-8
)
AZD3264是一种新型的小分子IKK2抑制剂。IKK2作为IB激酶的蛋白质亚基
A-971432
(Catalog# : 178816, Cas# :
1240308-45-5
)
A - 971432对S1P5具有高度选择性,在临床前口服剂量后,显露出良好
A-1165442
(Catalog# : 20178812, Cas# :
1221443-94-2
)
A-1165442是一种中性温度具有止痛功效的瞬时受体电位香草酸亚型1
AZD4205
(Catalog# : 20178710, Cas# :
2091134-35-7
)
AZD4205是一种高效JAK1-选择性激酶抑制剂,拥有优秀的临床前药代动
ACY-775
(Catalog# : 77821, Cas# :
1375466-18-4
)
ACY-775是一种组蛋白去乙酰化酶6(HDAC6)选择性抑制剂。
AAI-101
(Catalog# : 1773101, Cas# :
1001404-83-6
)
AAI101(AAI101)是一种新型的增谱-乳酸酶抑制剂。AAI101(AAI101)与头孢吡
AV-412甲苯磺酸盐
(Catalog# : 17030105, Cas# :
451493-31-5
)
AV-412,也称为MP-412,是第二代生物可利用的双激酶抑制剂,具有潜在
AZD-7594
(Catalog# : 17022812, Cas# :
1196509-60-0
)
AZD-7594,也叫AZ13189620,是一种吸入选择性糖皮质激素受体(GCCR)调制
AZD3839
(Catalog# : 17022710, Cas# :
1227163-56-5
)
AZD3839是一种有效的选择性BACE1抑制剂。AZD3839是治疗阿尔茨海默病
A-1210477
(Catalog# : 17022404, Cas# :
1668553-26-1
)
A-1210477是一种有效、选择性的MCL-1抑制剂。
阿帕替尼
(Catalog# : 17022301, Cas# :
811803-05-1
)
阿帕替尼是一种具有生物口服、选择性的IC50为1 nM的VEGFR2 抑制剂。
硫酸阿米卡星
(Catalog# : 17021407, Cas# :
39831-55-5
)
硫酸阿米卡星(BAY416651 硫酸)是一种由卡那霉素a衍生的半合成氨基
AFN-1252
(Catalog# : 17021406, Cas# :
620175-39-5
)
AFN-1252(Debio 1452) 是enoyl -酰基载体蛋白还原酶(FabI)的有效抑制剂。
AZD3293 (LY3314814)
(Catalog# : 17021318, Cas# :
1383982-64-6
)
AZD3293,也称为LY3314814是一种口服β-分泌酶1裂解酶(BACE)抑制剂。
APR-246 (PRIMA-1MET)
(Catalog# : 17021316, Cas# :
5291-32-7
)
APR-246, 也称为PRIMA-1MET, 是一种小型的有机分子,已被证明可以恢复
AZD-8835
(Catalog# : 102703, Cas# :
1620576-64-8
)
AZD8835 is a potent and selective inhibitor ofPI3KαandPI3KδwithIC50s of 6.2 and 5.7
AZD6482 (S-isomer)
(Catalog# : 17011901, Cas# :
1173900-37-2
)
AZD6482是强有力的,选择性和ATP竞争PI3K抑制剂(IC50为0.01μm)。
7ACC2
(Catalog# : 17011302, Cas# :
1472624-85-3
)
7ACC2是一种有效的MCT抑制剂。
AZD-5597
(Catalog# : 16122865, Cas# :
924641-59-8
)
AZD-5597 is potent CDK inhibitor with in vitro anti-proliferative effects against a r
AZD-5069
(Catalog# : 16122864, Cas# :
878385-84-3
)
AZD-5069 is a potent and selective CXCR2 antagonist with the potential to inhibit neu
«
2
3
4
5
6
7
8
9
10
11
»
产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AZD0095
(Catalog# : 237072, Cas# :
2750001-23-9
)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2-MNG
(Catalog# : 24129, Cas# :
2101538-28-5
)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
MAT2A-IN-9
(Catalog# : 25147, Cas# :
2439277-80-0
)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
Acoramidis hydrochloride
(Catalog# : 24068, Cas# :
2242751-53-5
)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
Crelosidenib
(Catalog# : 24101, Cas# :
2230263-60-0
)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
LOXO-435
(Catalog# : 25080, Cas# :
2833703-74-3
)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
Gridegalutamide
(Catalog# : 25138, Cas# :
2446928-30-7
)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
Chiauranib
(Catalog# : 25146, Cas# :
1256349-48-0
)
Chiauranib also known as orally available, small molecule inhibitor of select serine-