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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
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Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
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Chiral Compounds
Deuterated
Fluorides
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Pyrimidines
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Cas号索引 4
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Cas号索引 4
435327-40-5 | Avasopasem manganese
(Catalog# : 25108)
Avasopasem manganese, also known as GC-4419; M 40419 and SC-72325A, is a superoxide d
441022-64-6 | AMXT-1501 ( AMX-513 )
(Catalog# : 24026)
AMXT-1501 ( AMX-513 )是一种新型多胺转运系统抑制剂。 AMXT1501 可以阻
41294-56-8 | Alfacalcidol
(Catalog# : 20501)
Alfacalcidol is an active metabolite of Vitamin D, which performs important functions
422518-10-3 | 1-acetyl-5-amino-2-indolinone
(Catalog# : 2061313)
496791-37-8 | AR-C155858
(Catalog# : 193291)
AR-C155858是一种强效的单羧酸转运蛋白MCT1和MCT2的抑制剂,它与细胞
475479-34-6 | 阿格列扎
(Catalog# : 193125)
阿格列扎, 也称为RG-1439或RO-0728804,是一个过氧物酶体增生激活受
480998-12-7 | Aldoxorubicin盐酸盐
(Catalog# : 187111)
Aldoxorubicin,也称为INNO-206和Doxo-EMCH,是蒽醌类抗生素类霉素的6-马来
475489-16-8 | AEW-541
(Catalog# : 18753)
AEW541, 也称为NVP-AEW541,是一种有日常有效的IGF-IR激酶抑制剂。
450839-40-4 | ABT-100
(Catalog# : 1710131)
abt-100是一种口服的法尼基转移酶抑制剂.
451493-31-5 | AV-412甲苯磺酸盐
(Catalog# : 17030105)
AV-412,也称为MP-412,是第二代生物可利用的双激酶抑制剂,具有潜在
410074-74-7 | Amitifadine hydrochloride
(Catalog# : 6111104)
Amitifadine hydrochloride is a triple reuptake inhibitor (TRI) or serotonin-norepinep
473719-41-4 | AMG 487
(Catalog# : 122942)
AMG 487 is a small molecule antagonist of the chemokine receptor CXCR3.
486424-20-8 | AZD2858
(Catalog# : 122838)
AZD2858 is a selective GSK-3 inhibitor with an IC50 of 68 nM, inhibits tau phosphoryl
451492-95-8 | AV-412
(Catalog# : 112101)
AV-412 is an EGFR/HER2 inhibitor that binds to and inhibits the epidermal growth fact
497839-62-0 | AEE788
(Catalog# : 52750)
AEE788(NVP-AEE 788) is a potent inhibitor of EGFR and HER2/ErbB2 with IC50 of 2 nM an
487021-52-3 | AR-A014418
(Catalog# : 52523)
AR-A014418 is a selective and effective GSK3 inhibitor with an IC 50 value of 104 +/-
445000-45-3 | BBT
(Catalog# : 20570)
BBT is an enhancer of impaired glucose-stimulated insulin secretion (GSIS).
497223-19-5 | 497223-19-5
(Catalog# : 20403)
497223-19-5 | 497223-19-5
(Catalog# : 20386)
439575-02-7 | BMS-509744
(Catalog# : 1811291)
BMS-509744是一种有效的白介素-2诱导T细胞激酶(ITK)抑制剂(IC50 = 19 nM
406205-74-1 | BAY-59-3074
(Catalog# : 16122805)
BAY-59-3074 is a novel cannabinoid CB1/CB2 receptor partial agonist with analgesic pr
408502-43-2 | 3-Bromo-2-iodopyridine
(Catalog# : 032507)
Coming soon!
468740-43-4 | BMS-536924
(Catalog# : 010818)
BMS-536924 is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM.
444643-16-7 | Benzenemethanamine, 3,5-difluoro-α-methyl-, (alphaS)- (9CI)
(Catalog# : 91121)
Coming soon!
42287-90-1 | 3-(3-Bromophenyl)propionic acid
(Catalog# : 90707)
Coming soon!
461432-23-5 | 5-bromo-2-chloro-4'-ethoxydiphenylmethane
(Catalog# : 82713)
Coming soon!
405057-75-2 | benzyl 4-(methylamino)piperidine-1-carboxylate
(Catalog# : 81808)
Coming soon!
414864-00-9 | Belinostat
(Catalog# : 52521)
Belinostat (PXD101) is a novel pan-HDAC inhibitor with IC50 of 27 nM, with activity d
475301-73-6 | 2-(4-chlorophenyl)-2,2-difluoroacetic acid
(Catalog# : 20393)
456-04-2 | 2-氯代-4'-氟苯乙酮
(Catalog# : 20387)
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
1802632-22-9 | CT1812 ( Zervimesine )
(Catalog# : 193283)
CT-1812是一种同类首创的、可口服的sigma-2/PGRMC1拮抗剂(αβ寡聚体
3041025-10-6 | BLU-808
(Catalog# : 26A024)
BLU-808是一种针对肥大细胞疾病的野生型c-KIT的强效且具有选择性的
2243882-74-6 | Zedoresertib
(Catalog# : 26A023)
Zedoresertib(Debio 0123)是一种脑渗透剂,高选择性WEE1激酶抑制剂。
3033961-38-2 | BEN-28010
(Catalog# : 26A022)
BEN-28010是一种自由脑渗透剂,强效且具有选择性的CHK1抑制剂。
3107291-07-3 | 4-((2-(甲氨基)-6-(2,2,2-三氟乙基)噻吩并[2,3-d]嘧啶-4-基)氨基)哌啶-1-甲酸叔丁酯
(Catalog# : 26B007)
2565656-70-2 | Muvalaplin
(Catalog# : 20528)
Muvalaplin是一种小分子,通过干扰载脂蛋白(a)与载脂蛋白B100的结合
2925330-18-1 | MAT2A-IN-22
(Catalog# : 26A021)
MAT2A-IN-22 (Compound 29-1) 是一种可透过血脑屏障的和口服有效的 MAT2A
1497439-74-3 | AD-8007
(Catalog# : 26A018)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
1802650-31-2 | ZY-444
(Catalog# : 26A020)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
2306525-79-9 | AD-5584
(Catalog# : 26A019)
AD-5584是一种新型脑渗透性ACSS2抑制剂。