武汉永璨生物科技有限公司
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抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
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Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
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Other Heterocycles
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技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
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产品名字索引 Y
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产品名字索引 Y
YTX-465
(Catalog# : 24139, Cas# :
2225824-53-1
)
YTX-465 is a SCD inhibitor. YTX-465 strongly reduced fatty desaturation in a concentr
YCT529
(Catalog# : 24120, Cas# :
2863670-67-9
)
YCT529, an RAR-α inhibitor, is used as a contraceptive, with a 99% effectiveness. YC
YK-029A
(Catalog# : 20670, Cas# :
2064269-82-3
)
YW2065
(Catalog# : 20494, Cas# :
2131223-85-1
)
YW2065 has excellent anti-colorectal cancer effects in vitro and in vivo. YW2065 achi
YKL-05-099
(Catalog# : 21241, Cas# :
1936529-65-5
)
YKL-05-099 is a selective inhibitor of Salt-Inducible Kinase (SIK).
YCN47284
(Catalog# : 2073105, Cas# :
181147-28-4
)
YCN47284 is an aromatic guanylhydrazone compounds with antimalarial activity.
YUN27078
(Catalog# : 2071610, Cas# :
879127-07-8
)
YUN27078, also known as EGFR inhibitor, is an EGFR inhibitor. It directly depolymeriz
Y06137
(Catalog# : 193193, Cas# :
2226534-49-0
)
Y06137是一种有效的选择性BET抑制剂,它与Kd为81 nM的BRD4(1)溴域结合
YF-2盐酸盐
(Catalog# : 193151, Cas# :
1312005-62-1
)
YF-2盐酸盐是一个具有高度选择性,血脑屏障渗透组蛋白乙酰转移酶
YH239-EE
(Catalog# : 192213, Cas# :
1364488-67-4
)
YH239-EE是一种高效的p53-MDM2拮抗剂。
Y-39983游离
(Catalog# : 185172, Cas# :
199433-58-4
)
Y-39983 (游离),也被称为Y-33075,是一种有效的、选择性的ROCK家族抑
YL-0919
(Catalog# : 18578, Cas# :
1339058-04-6
)
YL-0919是一种日常5-HT1A受体拮抗剂,具有选择性的 5 -羟色胺再摄取
YU-238259
(Catalog# : 1710139, Cas# :
1943733-16-1
)
YU238259表现出有效的合成致死性设置中的DNA损伤反应和DNA修复缺陷
Y-29794 甲苯磺酸酯
(Catalog# : 1791521, Cas# :
143984-17-2
)
Y-29794甲苯磺酸酯是一种口服有效的,强有力的和特定的非肽脯氨
Y15盐酸
(Catalog# : 17030112, Cas# :
4506-66-5
)
Y15盐酸,也称为FAK抑制剂14,是一种直接FAK自身磷酸化抑制剂,阻塞
Y-39983盐酸盐
(Catalog# : 17021305, Cas# :
173897-44-4
)
Y-39983是一种选择性的与之相关的蛋白激酶(ROCK)抑制剂,其IC50为3.
740 Y-P (PDGFR 740Y-P)
(Catalog# : 17021302, Cas# :
1236188-16-1
)
740 Y-P是PI3K的细胞渗透磷肽激活剂。
YM-58483 (BTP2)
(Catalog# : 17109009, Cas# :
223499-30-7
)
YM-58483/BTP2是一种能调节非兴奋细胞(如淋巴细胞)活化的贮藏操作C
YM-90709
(Catalog# : 16122849, Cas# :
163769-88-8
)
YM-90709 is an interleukin-5 receptor antagonist. YM-90709 inhibits the binding of IL
Y-29794 Tosylate
(Catalog# : 16122848, Cas# :
129184-48-1
)
Y-29794 Tosylate is an orally active, potent and specific non-peptide prolyl endopept
YHO-13351
(Catalog# : 6111512, Cas# :
1346753-00-1
)
YHO-13351 is the water-soluble prodrug of YHO-13177, which is a potent and specific i
YHO-13177
(Catalog# : 6111511, Cas# :
912287-56-0
)
YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of
YM-155 hydrochloride
(Catalog# : 6111414, Cas# :
355406-09-6
)
YM155 is a potent survivin suppressant by inhibiting Survivin promoter activity with
YLF-466D
(Catalog# : 611813, Cas# :
1273323-67-3
)
YLF-466D is an allosteric AMPK activator.YLF466D activated recombinant human 111, 211
Y27632(free base)
(Catalog# : 16070918, Cas# :
146986-50-7
)
Y27632 is a selective ROCK inhibitor, which inhibits ET-1-induced increases in natriu
YK11
(Catalog# : 030910, Cas# :
1370003-76-1
)
Coming soon!
Y-27632 dihydrochloride
(Catalog# : 010421, Cas# :
129830-38-2
)
Y-27632 2Hcl is a selective ROCK1 (p160ROCK) inhibitor with Ki of 140 nM, exhibits &g
YM-201636
(Catalog# : 121426, Cas# :
371942-69-7
)
YM201636 is a selective PIKfyve inhibitor with IC50 of 33 nM, less potent to p110.
YL-109
(Catalog# : 110219, Cas# :
36341-25-0
)
YL-109 has ability to inhibit breast cancer cell growth and invasiveness in vitro and
Y-320
(Catalog# : 52516, Cas# :
288250-47-5
)
Y-320 is a new phenylpyrazoleanilide immunomodulator; inhibits IL-17 production by CD
产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AZD0095
(Catalog# : 237072, Cas# :
2750001-23-9
)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2-MNG
(Catalog# : 24129, Cas# :
2101538-28-5
)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
MAT2A-IN-9
(Catalog# : 25147, Cas# :
2439277-80-0
)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
Acoramidis hydrochloride
(Catalog# : 24068, Cas# :
2242751-53-5
)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
Crelosidenib
(Catalog# : 24101, Cas# :
2230263-60-0
)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
LOXO-435
(Catalog# : 25080, Cas# :
2833703-74-3
)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
Gridegalutamide
(Catalog# : 25138, Cas# :
2446928-30-7
)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
Chiauranib
(Catalog# : 25146, Cas# :
1256349-48-0
)
Chiauranib also known as orally available, small molecule inhibitor of select serine-