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Inhibitors & Agonists

编号化学名称Cas号纯度化学结构
51803Semaxanib (SU5416)204005-46-998% 
Semaxanib (SU5416) is a potent and selectiveVEGFR(Flk-1/KDR) inhibitor withIC50of 1.2
102703AZD-88351620576-64-8≧98.0%
AZD8835 is a potent and selective inhibitor ofPI3KαandPI3KδwithIC50s of 6.2 and 5.7
184321Ensartinib ( X396 )1370651-20-9>98%
Ensartinib is an orally available small molecule inhibitor of the receptor tyrosine k
26A016iMQT_0202463893-46-9≧98.0%
iMQT_020是一种特异性小分子抑制剂,靶向线粒体SLC1A5_var(谷氨酰胺
26A009Velzatinib (IDRX-42, M-4205)2590556-80-0≧98.0%
Velzatinib是一种口服生物可利用的小分子抑制剂,可抑制多种突变
26A010DPTX-3186≧98.0%
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
26A011Iadademstat ( ORY-1001 ) hydrochloride1431303-72-8≧98.0%
Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶
26A018AD-80071497439-74-3≧98.0%
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)