| 编号 | 化学名称 | Cas号 | 纯度 | 化学结构 |
|---|---|---|---|---|
| 51803 | Semaxanib (SU5416) | 204005-46-9 | 98% | ![]() |
| Semaxanib (SU5416) is a potent and selectiveVEGFR(Flk-1/KDR) inhibitor withIC50of 1.2 | ||||
| 102703 | AZD-8835 | 1620576-64-8 | ≧98.0% | ![]() |
| AZD8835 is a potent and selective inhibitor ofPI3KαandPI3KδwithIC50s of 6.2 and 5.7 | ||||
| 184321 | Ensartinib ( X396 ) | 1370651-20-9 | >98% | ![]() |
| Ensartinib is an orally available small molecule inhibitor of the receptor tyrosine k | ||||
| 26A016 | iMQT_020 | 2463893-46-9 | ≧98.0% | ![]() |
| iMQT_020是一种特异性小分子抑制剂,靶向线粒体SLC1A5_var(谷氨酰胺 | ||||
| 26A009 | Velzatinib (IDRX-42, M-4205) | 2590556-80-0 | ≧98.0% | ![]() |
| Velzatinib是一种口服生物可利用的小分子抑制剂,可抑制多种突变 | ||||
| 26A010 | DPTX-3186 | ≧98.0% | ![]() | |
| DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin | ||||
| 26A011 | Iadademstat ( ORY-1001 ) hydrochloride | 1431303-72-8 | ≧98.0% | ![]() |
| Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶 | ||||
| 26A018 | AD-8007 | 1497439-74-3 | ≧98.0% | ![]() |
| AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2) | ||||
