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抑制剂/受体激动剂
Angiogenesis
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
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Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
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技术服务
定制合成
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订购信息
联系我们
公司简介
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产品名字索引 U
Umbralisib
(Catalog# : 25085, Cas# :
1532533-67-7
)
Umbralisib, also known as TGR1202 and RP5264 , is a highly specific, orally available
Ulodesine
(Catalog# : 24098, Cas# :
548486-59-5
)
Ulodesine, also known as BCX4208, is a purine nucleoside phosphorylase (PNP) inhibito
UNC5293
(Catalog# : 24094, Cas# :
2226789-82-6
)
UNC5293 is a MERTK -selective and potent inhibitor ( Ki=190 pM).
UJN49930 ( UGT8-IN-1 )
(Catalog# : 20677, Cas# :
2414349-93-0
)
UJN49930 ( UGT8-IN-1 ) 是 UDP-半乳糖神经酰胺半乳糖基转移酶 (UGT8) 的抑
Ulodesine
(Catalog# : 60634, Cas# :
548486- 59-5
)
Usnoflast
(Catalog# : 20629, Cas# :
2455519-86-3
)
Usnoflast is a non-steroidal anti-inflammatory (NSAID).
URAT1 inhibitor 7
(Catalog# : 20573, Cas# :
1632002-28-8
)
URAT1 inhibitor 7 (compound 10f) is a potent URAT1 inhibitor.
UAMC-1110
(Catalog# : 21249, Cas# :
1448440-52-5
)
UAMC-1110, also known as SP-13786, is a novel potent and selective inhibitor of fibro
U-18666A
(Catalog# : 20110401, Cas# :
3039-71-2
)
U-18666A is an inhibitor of cholesterol synthesis. It acts by inhibiting desmosterol
UCB9608
(Catalog# : 2071516, Cas# :
2244989-34-0
)
UCB9608 is a Potent, Orally Bioavailable PI4KIIIβ Inhibitor. UCB9608 showed the impr
UCB9608
(Catalog# : 2071515, Cas# :
1616413-96-7
)
UCB9608 is a Potent, Orally Bioavailable PI4KIIIβ Inhibitor. UCB9608 showed the impr
U-73343
(Catalog# : 112591, Cas# :
142878-12-4
)
U-73343 is a negative control (or inactive analogue) of U73122, which is a putative p
UNC2541
(Catalog# : 6111901, Cas# :
1612782-86-1
)
UNC2541 is a potent and MerTK-specific inhibitor and exhibits sub-micro molar inhibit
UPGL00004
(Catalog# : 193251, Cas# :
1890169-95-5
)
UPGL00004是谷氨酰胺酶C (GAC)的有效抑制剂。
Umibecestat游离
(Catalog# : 193223, Cas# :
1387560-01-1
)
Umibecestat,也被称为CNP-520,是一种β分泌酶抑制剂,是预防阿尔茨
UVI3003
(Catalog# : 19343, Cas# :
847239-17-2
)
UVI3003是一种RXR拮抗剂。显示出较高的RXR结合亲和力。UVI3003并不影
Upacicalcet ( 别名 SK-1403 ; AJT240)
(Catalog# : 192142, Cas# :
1333218-50-0
)
Upacicalcet(别名 SK-1403/AJT240)是一种新型非肽拟钙剂,作为钙敏感
UC-1728
(Catalog# : 1812292, Cas# :
948304-40-3
)
UC-1728,又称t-TUCB,是一种可溶性环氧化物水解酶抑制剂。
URMC-099
(Catalog# : 1810252, Cas# :
1229582-33-5
)
URMC-099是一种口服生物可用的、脑内渗透混合谱系激酶(MLK)抑制剂
UM-164
(Catalog# : 186282, Cas# :
903564-48-7
)
UM-164是一种抗癌抑制剂。CAS号为903564-48-7。
UNC-926游离
(Catalog# : 18584, Cas# :
1184136-10-4
)
UNC-926是一种L3MBTL1域抑制剂. UNC-926联结L3MBTL1蛋白的MBT域。(Kd = 3.9
乌帕替尼
(Catalog# : 184105, Cas# :
1310726-60-3
)
乌帕替尼,也被称为ABT-494,是一种强力和选择性的JAK抑制剂,用
UPF-1069
(Catalog# : 1791520, Cas# :
1048371-03-4
)
UPF-1069是一种选择性的强效PARP2抑制剂。UPF-1069诱导细胞凋亡。UPF-
Ulixertinib HCl
(Catalog# : 179153, Cas# :
1956366-10-1
)
Ulixertinib,也称为BVD-523和VRT752271,是ERK蛋白激酶抑制剂。对ERK蛋白
UK-371804
(Catalog# : 1791114, Cas# :
256477-09-5
)
UK-371804是强有力和有选择性的优良酶效价uPA(Ki 10 nm)抑制剂和选
UNC-669
(Catalog# : 178312, Cas# :
314241-44-5
)
UNC-669是L3MBTL领域抑制剂。UNC669是专门针对 IC50 5μM的致死3恶性脑肿
UK-371804 HCl
(Catalog# : 17031008, Cas# :
256476-36-5
)
UK-371804是一种有效的选择性尿激酶型等离子体激活剂(uPA)抑制剂,
URB602
(Catalog# : 17030711, Cas# :
565460-15-3
)
URB602是monoglycerol脂肪酶的选择性抑制剂(MGL),老鼠大脑的酶展现出I
乌苯美司
(Catalog# : 17030602, Cas# :
58970-76-6
)
Ubenimex, also known as NK 421 and Bestatin, is a CD13 inhibitor. Ubenimex attenuates
UNC3866
(Catalog# : 17011102, Cas# :
1872382-47-2
)
UNC3866是一种强力拮抗剂,对多梳型CBX和CDY家族染色体组的阅读功
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AZD0095
(Catalog# : 237072, Cas# :
2750001-23-9
)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2-MNG
(Catalog# : 24129, Cas# :
2101538-28-5
)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
MAT2A-IN-9
(Catalog# : 25147, Cas# :
2439277-80-0
)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
Acoramidis hydrochloride
(Catalog# : 24068, Cas# :
2242751-53-5
)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
Crelosidenib
(Catalog# : 24101, Cas# :
2230263-60-0
)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
LOXO-435
(Catalog# : 25080, Cas# :
2833703-74-3
)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
Gridegalutamide
(Catalog# : 25138, Cas# :
2446928-30-7
)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
Chiauranib
(Catalog# : 25146, Cas# :
1256349-48-0
)
Chiauranib also known as orally available, small molecule inhibitor of select serine-