武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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Amines
Amino Acids
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Boronic Acids
Bromides
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Deuterated
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Indoles and Oxindoles
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Peg Linkers
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
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On Sale
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产品名字索引 A
Alobresib
(Catalog# : 185222, Cas# :
1637771-14-2
)
Alobresib是抗肿瘤药物的候选药物。
Adavivint
(Catalog# : 185221, Cas# :
1467013-03-3
)
Adavivint是一种Wnt通道抑制剂和免疫调制剂药物候选者。
ALX 1393
(Catalog# : 185213, Cas# :
949164-09-4
)
ALX 1393是一种甘氨酸转运体-2抑制剂。
A-485
(Catalog# : 185211, Cas# :
1889279-16-6
)
A-485是一种有效且具有选择性的p300/CBP在体外的HAT抑制剂。
AS-1517499
(Catalog# : 185187, Cas# :
919486-40-1
)
AS-1517499是一种有效且具有选择性的STAT6抑制剂。
AMG-176
(Catalog# : 185185, Cas# :
1883727-34-1
)
AMG-176是诱导髓系白血病细胞分化蛋白MCL-1(骨髓细胞白血病-1)的抑
A-350619盐酸盐
(Catalog# : 185183, Cas# :
1217201-17-6
)
A-350619盐酸盐是可溶性的胍基环酶(sGC)的激活剂。
ARQ-531
(Catalog# : 185176, Cas# :
2095393-15-8
)
ARQ-531是一种具有潜在抗肿瘤活性的有效的口服BTK抑制剂。
ADX-47273
(Catalog# : 185173, Cas# :
851881-60-2
)
ADX-47273是一种强有力的和选择性mGluR5受体PAM(积极的变构调制器),E
AMG-511
(Catalog# : 18542, Cas# :
1253573-53-3
)
AMG-511是一种有效的选择性的泛型I PI3K抑制剂。
AZD1390
(Catalog# : 18541, Cas# :
2089288-03-7
)
AZD1390是一种强效和选择性的ATM抑制剂,适合治疗颅内恶性肿瘤,
ALW-II-41-27
(Catalog# : 1842813, Cas# :
1186206-79-0
)
ALW-II-41-27是一种Eph受体酪氨酸激酶抑制剂。
AZD4635
(Catalog# : 184289, Cas# :
1321514-06-0
)
AZD-4635,也叫HTL-1071,是一种口服的小分子腺苷A2A受体拮抗剂。
Acrizanib
(Catalog# : 184181, Cas# :
1229453-99-9
)
Acrizanib,又名LHA510,是一种有效的选择性血管生成抑制剂和VEGFR -
2-amino-3-methoxy-4-(3-morpholin-4-ylpropoxy)benzonitrile
(Catalog# : 184163, Cas# :
1032570-98-1
)
2-amino-3-methoxy-4-(3-morpholin-4-ylpropoxy)benzonitrile是一种药物中间体。
安罗替尼
(Catalog# : 184132, Cas# :
1058156-90-3
)
安罗替尼,又名AL3818,是一种受体酪氨酸激酶(RTK)抑制剂,具有潜
A-804598
(Catalog# : 184125, Cas# :
1125758-85-1
)
A-804598是一种P2X7选择性、竞争性的拮抗剂。
AMD3465 HCl salt
(Catalog# : 184310, Cas# :
185991-07-5
)
AMD3465是一种新型CXCR4受体拮抗剂,具有潜在的抗癌和抗艾滋病活性
阿必鲁肽
(Catalog# : 18438, Cas# :
782500-75-8
)
阿必鲁肽是一种胰高血糖素-样 肽-1受体激动剂(GLP-1 受体激动剂)。
AVN-492
(Catalog# : 18425, Cas# :
1220646-23-0
)
AVN-492是一种有效且具有选择性的5-HT6R拮抗剂。AVN-492具有良好的体
ALB-127158A
(Catalog# : 18424, Cas# :
1173154-32-9
)
ALB-127158A, also known as ALB-127158(a), is a MCH1 antagonist for the treatment of o
AZD-5904
(Catalog# : 181121, Cas# :
618913-30-7
)
AZD5904是一个有效的口服生物利用率MPO抑制剂。在临床前研究中,AZ
2-氨基嘧啶-5-羧酸
(Catalog# : 171281, Cas# :
3167-50-8
)
2-氨基嘧啶-5-羧酸
Asciminib ( ABL001 )
(Catalog# : 1711222, Cas# :
1492952-76-7
)
Asciminib, 也叫ABL001,是一种有效的BCR-ABL的变构抑制剂。ABL001在与尼
Autophinib
(Catalog# : 17101617, Cas# :
1644443-47-9
)
Autophinib是一种新颖有效的自噬抑制剂,抑制通过靶向脂质激酶VPS
Adarigiline
(Catalog# : 1710167, Cas# :
1124197-79-0
)
adarigiline是单胺氧化酶B抑制剂的候选药物。
Adafosbuvir
(Catalog# : 1710166, Cas# :
1613589-09-5
)
Adafosbuvir是一种抗病毒药物。
AZD-5153 HNT salt
(Catalog# : 1710161, Cas# :
1869912-40-2
)
AZD-5153 HNT盐,是AZD-5153的6-hydroxy-2-naphthoic酸盐。AZD-5153对抗血液系
ABT-100
(Catalog# : 1710131, Cas# :
450839-40-4
)
abt-100是一种口服的法尼基转移酶抑制剂.
阿西鲁司特
(Catalog# : 179159, Cas# :
943764-99-6
)
阿西鲁司特,也称为ZK322,是强有力的和有选择性的白三烯A4水解酶
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AZD0095
(Catalog# : 237072, Cas# :
2750001-23-9
)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2-MNG
(Catalog# : 24129, Cas# :
2101538-28-5
)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
MAT2A-IN-9
(Catalog# : 25147, Cas# :
2439277-80-0
)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
Acoramidis hydrochloride
(Catalog# : 24068, Cas# :
2242751-53-5
)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
Crelosidenib
(Catalog# : 24101, Cas# :
2230263-60-0
)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
LOXO-435
(Catalog# : 25080, Cas# :
2833703-74-3
)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
Gridegalutamide
(Catalog# : 25138, Cas# :
2446928-30-7
)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
Chiauranib
(Catalog# : 25146, Cas# :
1256349-48-0
)
Chiauranib also known as orally available, small molecule inhibitor of select serine-