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抑制剂/受体激动剂
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
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Pyrimidines
Quinolines
Sulfonamides
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Trifluoroborates
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产品名字索引 A
AMG-9810
(Catalog# : 179117, Cas# :
545395-94-6
)
AMG 9810是对香草类受体1的辣椒素激活竞争性拮抗剂(TRPV1)。此外
AS-2444697 HCl
(Catalog# : 179832, Cas# :
1287665-60-4
)
AS-2444697是一种 RAK-4抑制剂。六周重复给药AS2444697(0.3-3mg/kg,一天
乙酰卡尼盐酸盐
(Catalog# : 179829, Cas# :
34118-92-8
)
乙酰卡尼,又名N-乙酰普鲁卡因胺和ASL 601,普鲁卡因胺是N-乙酰化
ASC-J9
(Catalog# : 179816, Cas# :
52328-98-0
)
ASC-J9,也称为GO-Y025和去甲氧基姜黄素,是一个AR降解剂,ASC-J9通过
AMG-009
(Catalog# : 17987, Cas# :
1027847-67-1
)
AMG 009是一种口服活性小分子CRTH2受体(趋化受体的同源分子表达在
5-氨基-2-氟-4-甲基苯腈
(Catalog# : 1781603, Cas# :
1426136-04-0
)
5-氨基-2-氟-4-甲基苯腈,5-amino-2-fluoro-4-methylbenzonitrile
2-azaspiro[3.5]nonan-7-ol hydrochloride
(Catalog# : 1781602, Cas# :
1434141-67-9
)
2-azaspiro[3.5]nonan-7-ol hydrochloride
Abemaciclib ( LY2835219)
(Catalog# : 178141, Cas# :
1231929-97-7
)
Abemaciclib,也被称为LY2835219,可口服细胞周期依赖性激酶(CDK)抑制
AZD3264
(Catalog# : 178910, Cas# :
1609281-86-8
)
AZD3264是一种新型的小分子IKK2抑制剂。IKK2作为IB激酶的蛋白质亚基
A-971432
(Catalog# : 178816, Cas# :
1240308-45-5
)
A - 971432对S1P5具有高度选择性,在临床前口服剂量后,显露出良好
A-1165442
(Catalog# : 20178812, Cas# :
1221443-94-2
)
A-1165442是一种中性温度具有止痛功效的瞬时受体电位香草酸亚型1
AZD4205
(Catalog# : 20178710, Cas# :
2091134-35-7
)
AZD4205是一种高效JAK1-选择性激酶抑制剂,拥有优秀的临床前药代动
ACY-775
(Catalog# : 77821, Cas# :
1375466-18-4
)
ACY-775是一种组蛋白去乙酰化酶6(HDAC6)选择性抑制剂。
AAI-101
(Catalog# : 1773101, Cas# :
1001404-83-6
)
AAI101(AAI101)是一种新型的增谱-乳酸酶抑制剂。AAI101(AAI101)与头孢吡
AV-412甲苯磺酸盐
(Catalog# : 17030105, Cas# :
451493-31-5
)
AV-412,也称为MP-412,是第二代生物可利用的双激酶抑制剂,具有潜在
AZD-7594
(Catalog# : 17022812, Cas# :
1196509-60-0
)
AZD-7594,也叫AZ13189620,是一种吸入选择性糖皮质激素受体(GCCR)调制
ABT888
(Catalog# : 17022801, Cas# :
912445-05-7
)
Veliparib (ABT-888)是PARP1和PARP2的有效抑制剂,Ki分别为5.2 nM和2.9 nM。
AZD3839
(Catalog# : 17022710, Cas# :
1227163-56-5
)
AZD3839是一种有效的选择性BACE1抑制剂。AZD3839是治疗阿尔茨海默病
A-1210477
(Catalog# : 17022404, Cas# :
1668553-26-1
)
A-1210477是一种有效、选择性的MCL-1抑制剂。
阿帕替尼
(Catalog# : 17022301, Cas# :
811803-05-1
)
阿帕替尼是一种具有生物口服、选择性的IC50为1 nM的VEGFR2 抑制剂。
硫酸阿米卡星
(Catalog# : 17021407, Cas# :
39831-55-5
)
硫酸阿米卡星(BAY416651 硫酸)是一种由卡那霉素a衍生的半合成氨基
AFN-1252
(Catalog# : 17021406, Cas# :
620175-39-5
)
AFN-1252(Debio 1452) 是enoyl -酰基载体蛋白还原酶(FabI)的有效抑制剂。
AZD3293 (LY3314814)
(Catalog# : 17021318, Cas# :
1383982-64-6
)
AZD3293,也称为LY3314814是一种口服β-分泌酶1裂解酶(BACE)抑制剂。
APR-246 (PRIMA-1MET)
(Catalog# : 17021316, Cas# :
5291-32-7
)
APR-246, 也称为PRIMA-1MET, 是一种小型的有机分子,已被证明可以恢复
AZD-8835
(Catalog# : 102703, Cas# :
1620576-64-8
)
AZD8835 is a potent and selective inhibitor ofPI3KαandPI3KδwithIC50s of 6.2 and 5.7
AZD6482 (S-isomer)
(Catalog# : 17011901, Cas# :
1173900-37-2
)
AZD6482是强有力的,选择性和ATP竞争PI3K抑制剂(IC50为0.01μm)。
7ACC2
(Catalog# : 17011302, Cas# :
1472624-85-3
)
7ACC2是一种有效的MCT抑制剂。
AZD-5597
(Catalog# : 16122865, Cas# :
924641-59-8
)
AZD-5597 is potent CDK inhibitor with in vitro anti-proliferative effects against a r
AZD-5069
(Catalog# : 16122864, Cas# :
878385-84-3
)
AZD-5069 is a potent and selective CXCR2 antagonist with the potential to inhibit neu
AZD-2461
(Catalog# : 16122863, Cas# :
1174043-16-3
)
AZD2461 is a novel and potent PARP inhibitor with lower affinity to P-glycoprotein. A
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Zelasudil
(Catalog# : 24014, Cas# :
2365193-22-0
)
Zelasudil 是一种有效的、高选择性的口服活性抑制剂,针对 Rho 相关
Ziftomenib ( KO-539 )
(Catalog# : 24013, Cas# :
2134675-36-6
)
Ziftomenib 是一种口服、有效、选择性的小分子抑制剂,针对 menin 和
Zunsemetinib
(Catalog# : 24012, Cas# :
1640282-42-3
)
Zunsemetinib是一种在研口服丝裂原活化蛋白激酶活化蛋白激酶2(MK2
Zongertinib ( BI 1810631 )
(Catalog# : 24011, Cas# :
2728667-27-2
)
Zongertinib [BI 1810631] 是一种人表皮生长因子受体 2 (HER2) 抑制剂。
Zasocitinib
(Catalog# : 24010, Cas# :
2272904-53-5
)
Zasocitinib是一种作用于非受体酪氨酸蛋白激酶 (TYK2)靶点的抑制
RNK-05047
(Catalog# : 24008, Cas# :
2503036-46-0
)
RNK-05047 为BRD4降解剂,其在小鼠荷瘤异种移植模型中展现出显著抑
Asengeprast (FT011)
(Catalog# : 24009, Cas# :
1001288-58-9
)
Asengeprast (FT011) 是一种抗纤维化剂,降低胶原蛋白 I 和 III 的 mRNA
ERAS-801 ( JGK-068S )
(Catalog# : 20635, Cas# :
2490431-16-6
)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。
T-1095
(Catalog# : 24004, Cas# :
209746-59-8
)
T-1095 is a potent and selective inhibitor of Na+-glucose cotransporters (SGLTs).
NVL-655 ( ALK-IN-27 )
(Catalog# : 24003, Cas# :
2739866-40-9
)
NVL-655是一种新型脑渗透性ALK选择性抑制剂,旨在解决目前可用的