武汉永璨生物科技有限公司
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抑制剂/受体激动剂
Angiogenesis
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分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
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Indoles and Oxindoles
Iodos
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Peg Linkers
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Pyridines
Pyrimidines
Quinolines
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
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Deuterated
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Iodos
Nitro Compounds
Oxazoles
Peg Linkers
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Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
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产品名字索引 A
AMD-070盐酸盐
(Catalog# : 18741, Cas# :
880549-30-4
)
AMD11070,也称为 AMD070, X4P-001和mavorixafor, 是一种有效的口服生物活
AG-494
(Catalog# : 186273, Cas# :
133550-35-3
)
AG-494,也被称为Tyrphostin AG- 494,是表皮生长因子受体激酶的抑制剂
AZD5153
(Catalog# : 186254, Cas# :
1869912-39-9
)
AZD5153是一种有效的双价三唑吡啶溴化和外治(BET)抑制剂。
阿莫奈韦
(Catalog# : 186252, Cas# :
841301-32-4
)
阿莫奈韦是一种 helicase-primase 抑制剂,对 HSVs 具有强效的抗病毒活
A22盐酸盐
(Catalog# : 186211, Cas# :
22816-60-0
)
A22是一种MreB的抑制剂,是一种类似actin样的细菌蛋白,已经被证明
AST487
(Catalog# : 186158, Cas# :
630124-46-8
)
AST487, 也称为NVP- AST487, 是一种RET激酶抑制剂/FLT3抑制剂。
ARV-825
(Catalog# : 185253, Cas# :
1818885-28-7
)
ARV-825是一种保护蛋白(蛋白酶-靶向嵌合体)。ARV-825与溴域抑制剂(B
Alobresib
(Catalog# : 185222, Cas# :
1637771-14-2
)
Alobresib是抗肿瘤药物的候选药物。
Adavivint
(Catalog# : 185221, Cas# :
1467013-03-3
)
Adavivint是一种Wnt通道抑制剂和免疫调制剂药物候选者。
ALX 1393
(Catalog# : 185213, Cas# :
949164-09-4
)
ALX 1393是一种甘氨酸转运体-2抑制剂。
A-485
(Catalog# : 185211, Cas# :
1889279-16-6
)
A-485是一种有效且具有选择性的p300/CBP在体外的HAT抑制剂。
AS-1517499
(Catalog# : 185187, Cas# :
919486-40-1
)
AS-1517499是一种有效且具有选择性的STAT6抑制剂。
AMG-176
(Catalog# : 185185, Cas# :
1883727-34-1
)
AMG-176是诱导髓系白血病细胞分化蛋白MCL-1(骨髓细胞白血病-1)的抑
A-350619盐酸盐
(Catalog# : 185183, Cas# :
1217201-17-6
)
A-350619盐酸盐是可溶性的胍基环酶(sGC)的激活剂。
ARQ-531
(Catalog# : 185176, Cas# :
2095393-15-8
)
ARQ-531是一种具有潜在抗肿瘤活性的有效的口服BTK抑制剂。
ADX-47273
(Catalog# : 185173, Cas# :
851881-60-2
)
ADX-47273是一种强有力的和选择性mGluR5受体PAM(积极的变构调制器),E
AMG-511
(Catalog# : 18542, Cas# :
1253573-53-3
)
AMG-511是一种有效的选择性的泛型I PI3K抑制剂。
AZD1390
(Catalog# : 18541, Cas# :
2089288-03-7
)
AZD1390是一种强效和选择性的ATM抑制剂,适合治疗颅内恶性肿瘤,
ALW-II-41-27
(Catalog# : 1842813, Cas# :
1186206-79-0
)
ALW-II-41-27是一种Eph受体酪氨酸激酶抑制剂。
AZD4635
(Catalog# : 184289, Cas# :
1321514-06-0
)
AZD-4635,也叫HTL-1071,是一种口服的小分子腺苷A2A受体拮抗剂。
Acrizanib
(Catalog# : 184181, Cas# :
1229453-99-9
)
Acrizanib,又名LHA510,是一种有效的选择性血管生成抑制剂和VEGFR -
2-amino-3-methoxy-4-(3-morpholin-4-ylpropoxy)benzonitrile
(Catalog# : 184163, Cas# :
1032570-98-1
)
2-amino-3-methoxy-4-(3-morpholin-4-ylpropoxy)benzonitrile是一种药物中间体。
安罗替尼
(Catalog# : 184132, Cas# :
1058156-90-3
)
安罗替尼,又名AL3818,是一种受体酪氨酸激酶(RTK)抑制剂,具有潜
A-804598
(Catalog# : 184125, Cas# :
1125758-85-1
)
A-804598是一种P2X7选择性、竞争性的拮抗剂。
AMD3465 HCl salt
(Catalog# : 184310, Cas# :
185991-07-5
)
AMD3465是一种新型CXCR4受体拮抗剂,具有潜在的抗癌和抗艾滋病活性
阿必鲁肽
(Catalog# : 18438, Cas# :
782500-75-8
)
阿必鲁肽是一种胰高血糖素-样 肽-1受体激动剂(GLP-1 受体激动剂)。
AVN-492
(Catalog# : 18425, Cas# :
1220646-23-0
)
AVN-492是一种有效且具有选择性的5-HT6R拮抗剂。AVN-492具有良好的体
ALB-127158A
(Catalog# : 18424, Cas# :
1173154-32-9
)
ALB-127158A, also known as ALB-127158(a), is a MCH1 antagonist for the treatment of o
AZD-5904
(Catalog# : 181121, Cas# :
618913-30-7
)
AZD5904是一个有效的口服生物利用率MPO抑制剂。在临床前研究中,AZ
2-氨基嘧啶-5-羧酸
(Catalog# : 171281, Cas# :
3167-50-8
)
2-氨基嘧啶-5-羧酸
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Dencatistat (STP938)
(Catalog# : 25177, Cas# :
2377000-84-3
)
Dencatistat 是一种口服生物可利用的小分子胞苷三磷酸合酶 1 (CTPS1)
DS-1001b
(Catalog# : 25178, Cas# :
1898207-64-1
)
DS-1001 是一种口服的脑渗透性突变 IDH1 选择性抑制剂。
Z57346765
(Catalog# : 25191, Cas# :
1016340-64-9
)
Z57346765 是一种 PGK1 特异性抑制剂,可降低 PGK1 糖酵解中代谢酶的
CBR-470-1
(Catalog# : 25192, Cas# :
2416095-06-0
)
CBR-470-1 是诱导 Nrf2 活性的糖酵解酶 PGK1 的抑制剂。
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
HC-7366
(Catalog# : 25076, Cas# :
2803470-63-3
)
HC-7366 is a potent and selective activator of the general control nonderepressible 2
Flavopiridol ( 夫拉平度 )
(Catalog# : 237071, Cas# :
146426-40-6
)
Alvocidib is a synthetic dihydroxyflavone that is 5,7-dihydroxyflavone which is subst
AG-270
(Catalog# : 25176, Cas# :
2201056-66-6
)
MAT2A 抑制剂 AG-270 是一种口服的蛋氨酸腺苷转移酶 II α (MAT2A) 小分
AZD-5904
(Catalog# : 181121, Cas# :
618913-30-7
)
AZD5904是一个有效的口服生物利用率MPO抑制剂。在临床前研究中,AZ
ALT-007
(Catalog# : 25157, Cas# :
2035010-37-6
)
ALT-007 是一种口服生物可利用的 SPT 抑制剂,比多球菌素更有效,