编号 | 化学名称 | Cas号 | 纯度 |
---|---|---|---|
24017 | AMG-193 AMG-193是安进公司开发的一种口服小分子甲硫腺苷协同PRMT5酶抑制剂 |
2790567-82-5 | 98.62%; EE 98.28% |
41788 | CB-6644 CB-6644 acts as a noncompetitive ATPase inhibitor. Additionally, it can inhibit RUVBL |
2316817-88-4 | 96.33% |
24068 | Acoramidis hydrochloride Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR |
2242751-53-5 | ≧98.0% |
24064 | Cirtuvivint ( SM08502 ) Cirtuvivint是一种CDC样激酶(CLK)和双特异性酪氨酸磷酸化调节激酶 |
2143917-62-6 | ≧98.0% |
181121 | AZD-5904 AZD5904是一个有效的口服生物利用率MPO抑制剂。在临床前研究中,AZ |
618913-30-7 | ≧98.0% |
237071 | Flavopiridol ( 夫拉平度 ) Alvocidib is a synthetic dihydroxyflavone that is 5,7-dihydroxyflavone which is subst |
146426-40-6 | ≧98.0% |
24107 | LXH-3-71 LXH-3-71是一种新型“分子胶”,可诱导PHGDH和DDB1-CUL4泛素连接酶之 |
2251753-65-6 | ≧97.0% |
20509 | GLPG3667 GLPG3667 是一种口服强效选择性小分子 TYK2 抑制剂,正在开发用于治 |
2308520-97-8 | ≧98.0% |
121431 | KW-2478 KW-2478 是一种针对人类热休克蛋白 90 (Hsp90) 的药物,具有潜在的抗 |
819812-04-9 | 98% |
18576 | VU0467154 VU0467154 is a positive allosteric modulator of theM4 muscarinic acetylcholine recept |
1451993-15-9 | ≧98.0% |
171452 | BGB 15025 ; BGB-15025 ; BGB15025 BGB-15025 是一种有效的选择性 HPK1 抑制剂,在多种肿瘤模型中作为 |
2766481-17-6 | ≧98.0% |
17021601 | LY3039478 ( Crenigacestat ) LY3039478 ( Crenigacestat ) 是一种选择性 NOTCH1 抑制剂,通过阻断 VEGFA/ |
1421438-81-4 | ≧98.0% |
711401 | Eganelisib ( IPI-549 ) Eganelisib (IPI-549) 是一种首创、口服、高选择性 PI3Kγ 抑制剂,单独 |
1693758-51-8 | ≧98.0% |
24067 | PBT434 氢溴酸盐 PBT434, also known as ATH434 , is a novel, brain-penetrant, inhibitor of α-synuclein |
1232841-78-9 | ≧98.0% |
233141 | NXP-800 ( CCT361814 ) NXP800 是一种口服小分子热休克因子 1 (HSF1) 通路抑制剂。 NXP800 可 |
1693734-80-3 | ≧98.0% |