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24101 | Crelosidenib

241012230263-60-0

Crelosidenib

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25079 | Sevabertinib ( 别名:BAY-2927088 )

250792521285-05-0

Sevabertinib ( 别名:BAY-2927088 )

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20633 | Tersolisib ( STX-478 )

206332883540-92-7

Tersolisib ( STX-478 )

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24084 | Iclepertin (BI-425809)

240841421936-85-7

Iclepertin (BI-425809)

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193264 | PF-06835919 ( MDK-1846 )

1932642102501-84-6

PF-06835919 ( MDK-1846 )

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20657 | Zilurgisertib

206572173389-57-4

Zilurgisertib

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20636 | Edecesertib ( GS-5718 )

206362408839-73-4

Edecesertib ( GS-5718 )

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174191 | SU5402

174191215543-92-3

SU5402

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编号化学名称Cas号纯度
25076 HC-7366
HC-7366 is a potent and selective activator of the general control nonderepressible 2
2803470-63-3 ≧98.0%
41788 CB-6644
CB-6644 acts as a noncompetitive ATPase inhibitor. Additionally, it can inhibit RUVBL
2316817-88-4 96.33%
25148 Atebimetinib
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
2669009-92-9 ≧98.0%
25075 LLL12
LLL12是一种强效的STAT3抑制剂。LLL12在小鼠异种移植物模型中显示出
1260247-42-4 ≧97.0%
181121 AZD-5904
AZD5904是一个有效的口服生物利用率MPO抑制剂。在临床前研究中,AZ
618913-30-7 ≧98.0%
237071 Flavopiridol ( 夫拉平度 )
Alvocidib is a synthetic dihydroxyflavone that is 5,7-dihydroxyflavone which is subst
146426-40-6 ≧98.0%
24107 LXH-3-71
LXH-3-71是一种新型“分子胶”,可诱导PHGDH和DDB1-CUL4泛素连接酶之
2251753-65-6 ≧97.0%
20509 GLPG3667
GLPG3667 是一种口服强效选择性小分子 TYK2 抑制剂,正在开发用于治
2308520-97-8 ≧98.0%
121431 KW-2478
KW-2478 是一种针对人类热休克蛋白 90 (Hsp90) 的药物,具有潜在的抗
819812-04-9 98% 
18576 VU0467154
VU0467154 is a positive allosteric modulator of theM4 muscarinic acetylcholine recept
1451993-15-9 ≧98.0%
171452 BGB 15025 ; BGB-15025 ; BGB15025
BGB-15025 是一种有效的选择性 HPK1 抑制剂,在多种肿瘤模型中作为
2766481-17-6 ≧98.0%
17021601 LY3039478 ( Crenigacestat )
LY3039478 ( Crenigacestat ) 是一种选择性 NOTCH1 抑制剂,通过阻断 VEGFA/
1421438-81-4 ≧98.0%
711401 Eganelisib ( IPI-549 )
Eganelisib (IPI-549) 是一种首创、口服、高选择性 PI3Kγ 抑制剂,单独
1693758-51-8 ≧98.0%
24067 PBT434 氢溴酸盐
PBT434, also known as ATH434 , is a novel, brain-penetrant, inhibitor of α-synuclein
1232841-78-9 ≧98.0%
233141 NXP-800 ( CCT361814 )
NXP800 是一种口服小分子热休克因子 1 (HSF1) 通路抑制剂。 NXP800 可
1693734-80-3 ≧98.0%