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抑制剂/受体激动剂
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Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
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Catalysts
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Deuterated
Fluorides
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Indoles and Oxindoles
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Pyridines
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
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产品名字索引 A
AM281
(Catalog# : 19315, Cas# :
202463-68-1
)
AM281是一种合成大麻素CB1受体拮抗剂。
ASP9521
(Catalog# : 19312, Cas# :
1126084-37-4
)
ASP9521是日常的,选择性,口服生物利用率17β-羟甾类脱氢酶的抑制
AZD0364
(Catalog# : 192275, Cas# :
2097416-76-5
)
AZD0364是一种用于治疗癌症的ERK1和/或ERK2激酶。ERK1和ERK2激酶是广泛
ATF6-活化剂-147
(Catalog# : 192212, Cas# :
393121-74-9
)
ATF6-activator-147是一种ATF6模拟器,它作为一种前体药物,通过一种
AZD1152
(Catalog# : 192156, Cas# :
722543-31-9
)
AZD1152是Barasertib-hQPA的前药,是一种高选择性极光B抑制剂,在无细
AZD3229
(Catalog# : 191287, Cas# :
2248003-60-1
)
AZD3229是治疗胃肠道间质瘤的一种有效的pan-kit突变抑制剂。AZD3229在
AM095钠
(Catalog# : 191251, Cas# :
1345614-59-6
)
AM095是一个强有力的LPA1受体拮抗剂,因为它抑制GTPγS绑定中国仓鼠
AZD4573
(Catalog# : 191212, Cas# :
2057509-72-3
)
AZD-4573是一种选择性的丝氨酸/苏氨酸依赖性激酶9 (CDK9)的短期抑制
AR-9281
(Catalog# : 191146, Cas# :
913548-29-5
)
AR-9281是一种可溶性环氧化物水解酶(s-EH)抑制剂,有望用于高血压
ARRY-797 (ARRY-371797)
(Catalog# : 191112, Cas# :
1036404-17-7
)
ARRY-797(CAS1036404-17-7) is an oral, selective p38 mitogen-activated protein kinase
艾维替尼
(Catalog# : 19141, Cas# :
1557267-42-1
)
艾维替尼,又称AC0010和Avitinib,是酪氨酸激酶抑制剂,抗肿瘤药物
AZD7507
(Catalog# : 1812294, Cas# :
1041852-85-0
)
AZD7507是一种有效的选择性CSF-1R抑制剂(32 nM 细胞活性), AZD7507被认
Auranofin
(Catalog# : 1812281, Cas# :
34031-32-8
)
Auranofin又称Ridaura和SKF-39162,是一种治疗类风湿性关节炎的口服大
AX-024盐酸盐
(Catalog# : 181254, Cas# :
1704801-24-0
)
AX-024是一种口服的TCR-Nck相互作用抑制剂,选择性地抑制TCR-触发的
AG 879
(Catalog# : 1811303, Cas# :
148741-30-4
)
AG-879是一种酪氨酸磷酸化抑制剂复合物,可抑制PC-12细胞中依赖神
Avagacestat
(Catalog# : 1811283, Cas# :
1146699-66-2
)
Avagacestat,也称为BMS- 708163是一种口服GSI用于选择性抑制Aβ合成,目
AS1842856
(Catalog# : 1811265, Cas# :
836620-48-5
)
AS1842856是一种细胞可渗透的Foxo1抑制剂,IC50为33 nM,阻断Foxo1的转
Anlotinib HCl ( AL-3818 )
(Catalog# : 1811211, Cas# :
1360460-82-7
)
Anlotinib也被称为AL3818,是一种受体酪氨酸激酶(RTK)抑制剂,具有潜
Avatrombopag maleate
(Catalog# : 5141902, Cas# :
677007-74-8
)
Avatrombopag maleate 是一种口服生物可用的小分子血栓生成素受体激动
AZD-3514
(Catalog# : 1810251, Cas# :
1240299-33-5
)
AZD-3514是一种具有潜在抗癌活性的雄激素受体下调因子。
AZ32
(Catalog# : 1810223, Cas# :
no
)
AZ32 是一种口服可利用的,可穿透血脑屏障的 ATM 抑制剂,IC50<6
ARS-1620
(Catalog# : 1810222, Cas# :
1698055-85-4
)
ARS-1620是一种具有理想药代动力学的阿托品选择性KRAS-G12C抑制剂。
AGL-2263
(Catalog# : 1810175, Cas# :
638213-98-6
)
AGL-2263是一种新型的胰岛素受体抑制剂。
AM211
(Catalog# : 1810173, Cas# :
1175526-27-8
)
AM-211是前列腺素D2受体2型的一种新型强效拮抗剂。
Arimoclomol maleate
(Catalog# : 188281, Cas# :
289893-26-1
)
Arimoclomol,也被称为BRX-220,能够潜在有用的治疗Niemann-Pick疾病C型
ASP7663
(Catalog# : 187123, Cas# :
1190217-35-6
)
ASP7663是口服生物可利用选择性TRPA1激活剂。
Aldoxorubicin盐酸盐
(Catalog# : 187111, Cas# :
480998-12-7
)
Aldoxorubicin,也称为INNO-206和Doxo-EMCH,是蒽醌类抗生素类霉素的6-马来
ABT 702盐酸盐
(Catalog# : 18791, Cas# :
1188890-28-9
)
ABT 702二盐酸盐是一种强效的非核苷腺苷激酶抑制剂,对腺甘酸相
Avacopan
(Catalog# : 18761, Cas# :
1346623-17-3
)
Avacopan也被称为CCX168,是一种口服活性、选择性和有效的C5aR抑制剂
AEW-541
(Catalog# : 18753, Cas# :
475489-16-8
)
AEW541, 也称为NVP-AEW541,是一种有日常有效的IGF-IR激酶抑制剂。
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Dencatistat (STP938)
(Catalog# : 25177, Cas# :
2377000-84-3
)
Dencatistat 是一种口服生物可利用的小分子胞苷三磷酸合酶 1 (CTPS1)
DS-1001b
(Catalog# : 25178, Cas# :
1898207-64-1
)
DS-1001 是一种口服的脑渗透性突变 IDH1 选择性抑制剂。
Z57346765
(Catalog# : 25191, Cas# :
1016340-64-9
)
Z57346765 是一种 PGK1 特异性抑制剂,可降低 PGK1 糖酵解中代谢酶的
CBR-470-1
(Catalog# : 25192, Cas# :
2416095-06-0
)
CBR-470-1 是诱导 Nrf2 活性的糖酵解酶 PGK1 的抑制剂。
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
HC-7366
(Catalog# : 25076, Cas# :
2803470-63-3
)
HC-7366 is a potent and selective activator of the general control nonderepressible 2
Flavopiridol ( 夫拉平度 )
(Catalog# : 237071, Cas# :
146426-40-6
)
Alvocidib is a synthetic dihydroxyflavone that is 5,7-dihydroxyflavone which is subst
AG-270
(Catalog# : 25176, Cas# :
2201056-66-6
)
MAT2A 抑制剂 AG-270 是一种口服的蛋氨酸腺苷转移酶 II α (MAT2A) 小分
AZD-5904
(Catalog# : 181121, Cas# :
618913-30-7
)
AZD5904是一个有效的口服生物利用率MPO抑制剂。在临床前研究中,AZ
ALT-007
(Catalog# : 25157, Cas# :
2035010-37-6
)
ALT-007 是一种口服生物可利用的 SPT 抑制剂,比多球菌素更有效,