武汉永璨生物科技有限公司
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抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
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定制合成
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联系我们
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联系我们
+86-27-65522453
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
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产品名字索引 L
Linzagolix
(Catalog# : 20266, Cas# :
935283-04-8
)
Linzagolix 是一种新型的口服 GnRH 受体拮抗剂,可有效治疗子宫内膜
LY-3475070
(Catalog# : 21244, Cas# :
2375815-63-5
)
LY-3475070 is a potent and selective CD73 Inhibitor with IC50 of 28 nM. LY3475070 Alo
LP-261
(Catalog# : 210507, Cas# :
915412-67-8
)
LP-261 is a novel tubulin targeting anticancer agent that binds at the colchicine sit
LM11A-31 HCl
(Catalog# : 21225, Cas# :
1243259-19-9
)
LVN84663
(Catalog# : 20113001, Cas# :
103784-66-3
)
LVN84663 is a useful reagent for determination of blood coagulating protease. It was
LUN42518
(Catalog# : 2091908, Cas# :
47142-51-8
)
LUN42518, also known as Phentolamine Analogue 1, is an analogue of phentolamine. Phen
Lerociclib HCl (G1T38 HCl)
(Catalog# : 2073106, Cas# :
2097938-59-3
)
Lerociclib HCl (G1T38 dihydrochloride)是一种分化型口服CDK4 / 6抑制剂,对
Lobaplatin
(Catalog# : 2071555, Cas# :
135558-11-1
)
Lobaplatin (D-19466) is a diastereometric mixture of platinum(II) complexes containin
Lixivaptan
(Catalog# : 2071524, Cas# :
168079-32-1
)
Lixivaptan, laso known as CRTX-080; VPA-985; WAY-VPA-985, is a potent, orally active,
LAU159
(Catalog# : 2071505, Cas# :
2055050-87-6
)
LAU159 is a potent modulator of α6β3γ2 GABAA receptor.
Lificiguat
(Catalog# : 2071502, Cas# :
170632-47-0
)
Lificiguat, also known as YC-1, is a inhibitor of Hypoxia-inducible factor-1alpha (HI
Lanraplenib
(Catalog# : 20732, Cas# :
1800046-95-0
)
GS-9876(lanraplenib)是一种高度选择性的口服SYK抑制剂,主要用于狼
Linperlisib free base
(Catalog# : 2061309, Cas# :
1702816-75-8
)
Linperlisib, also known as YY-20394 and PI3Kδ-IN-2, is a potent and selective PI3Kδ
L006235
(Catalog# : 2061307, Cas# :
294623-49-7
)
L006235 is a potent, reversible cathepsin K inhibitor (IC50 = 0.25 nM) that displays
LML-134
(Catalog# : 2051510, Cas# :
1542135-76-1
)
LML134 是一种具有口服活性,高选择性 H3R (组胺 3 受体) 反向激动剂
LUT-014
(Catalog# : 2042701, Cas# :
2274819-46-2
)
LUT-014 is a B-Raf Inhibitor. Leveraging the paradoxical effect of B-Raf Inhibitors,
LSZ102
(Catalog# : 2041502, Cas# :
2135600-76-7
)
LSZ102 is a potent ERα antagonist and degrader. LSZ102 showed ERα degradation IC50
LUN42589
(Catalog# : 204502, Cas# :
1848242-58-9
)
LUN42589,也称为PI3K / mTOR抑制剂2,是一种有效的双重pan-PI3K / mTOR抑
Lerociclib
(Catalog# : 204302, Cas# :
1628256-23-4 (free base)
)
Lerociclib,也称为G1T38,是一种口服,有效和选择性的CDK4 / 6抑制剂
Lemborexant (E-2006)
(Catalog# : 6111904, Cas# :
1369764-02-2
)
Lemborexant( E-2006, CAS 1369764-02-2)是食欲素OX 1和OX 2受体的双重拮抗
LY2794193
(Catalog# : 193262, Cas# :
2173037-97-1
)
LY2794193是一种高效选择性的mGlu3受体激动剂。
LY-3381916
(Catalog# : 193123, Cas# :
2166616-75-5
)
LY-3381916是一种强效的、选择性的、脑透性的IDO1活性抑制剂,与缺
LR-90
(Catalog# : 19364, Cas# :
245075-84-7
)
LR-90是一种晚期糖基化终产物(AGE)抑制剂,可抑制人单核细胞的炎
LCL521
(Catalog# : 19357, Cas# :
1226851-11-1
)
LCL521是一种酸性神经酰胺酶(ACDase)抑制剂。LCL521还抑制溶酶体酸鞘
Larotaxel
(Catalog# : 1922710, Cas# :
156294-36-9
)
Larotaxel是紫杉烷10-脱乙酰巴卡丁III的半合成衍生物,具有潜在的抗
Leniolisib
(Catalog# : 192271, Cas# :
1354690-24-6
)
Leniolisib,又名CDZ173,是一种有效的磷脂酰肌醇3激酶抑制剂(PI3K抑
Leuprolide Acetate
(Catalog# : 192261, Cas# :
74381-53-6
)
Leuprolide Acetate是一种合成的类似促性腺激素释放激素的非肽类似物
LOXO-292
(Catalog# : 192195, Cas# :
2222755-14-6
)
LOXO-292 (ARRY-192)是一种口服和临床开发的选择性研究药物,用于治
Lexibulin
(Catalog# : 19122, Cas# :
917111-49-0
)
Lexibulin,又称CYT997,是一种n型口服生物利用小分子,具有管蛋白
LP-211
(Catalog# : 1811302, Cas# :
1052147-86-0
)
LP-211是血清素5-HT7受体的选择性激动剂。
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
JPH203 HCl ( Nanvuranlat )
(Catalog# : 18381, Cas# :
1597402-27-1
)
JPH203,也称为KYT- 0353,是一个强有力的和选择性(l型氨基酸转运蛋白
(S)-2-甲基-5-氧代哌嗪-1-甲酸叔丁酯
(Catalog# : G20374, Cas# :
1627749-02-3
)
AZD-5904
(Catalog# : 181121, Cas# :
618913-30-7
)
AZD5904是一个有效的口服生物利用率MPO抑制剂。在临床前研究中,AZ
Fosgonimeton
(Catalog# : 1711225, Cas# :
2093305-05-4
)
SRI-37330 free base
(Catalog# : 1711224, Cas# :
2322245-42-9 (free base)
)
SRI-37330 is a novel inhibitor of TXNIP expression, decreasing glucagon secretion and
Asciminib HCl
(Catalog# : 1711223, Cas# :
2119669-71-3 (HCl)
)
Asciminib, also known as ABL001, is a potent allosteric inhibitor of BCR-ABL. ABL001
1,7,9-Triazaspiro[4.5]dec-1-ene-6,10-dione, 2,4-bis(4-chlorophenyl)-8-thioxo-
(Catalog# : G20373, Cas# :
2377858-38-1
)
SRI-37330 HCl
(Catalog# : 20306, Cas# :
2322245-49-6
)
SRI-37330 hydrochloride 是一种新型 TXNIP 表达抑制剂,呈剂量依赖性抑
SHMT-IN-2 抑制剂
(Catalog# : 20368, Cas# :
2102681-49-0
)
SHMT-IN-2 是一种丝氨酸羟甲基转移酶 (SHMT) 抑制剂,可有效抑制人
Anlotinib HCl ( AL-3818 )
(Catalog# : 1811211, Cas# :
1360460-82-7
)
Anlotinib也被称为AL3818,是一种受体酪氨酸激酶(RTK)抑制剂,具有潜