武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
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Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
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产品名字索引 K
KL1333
(Catalog# : 25201, Cas# :
1800405-30-4
)
KL1333是一种口服的小有机分子,与NAD(P)H:醌氧化还原酶1(NQO1)
KT-474 ( 别名: SAR-444656 )
(Catalog# : 25165, Cas# :
2432994-31-3
)
KT-474 (SAR-444656) 是一种口服的 IRAK4 降解诱导剂。
KH-3
(Catalog# : 24143, Cas# :
1215115-03-9
)
KH-3 is a potent RNA-binding protein Hu antigen R (HuR) inhibitor with an IC50 value
KB-0742
(Catalog# : 24040, Cas# :
2416873-83-9
)
KB-0742 是一种有效的,选择性的和具有口服活性的 CDK9 抑制剂。
KUS121
(Catalog# : 20676, Cas# :
1357164-52-3
)
KUS-121 是一种过渡内质网 ATP 酶(含缬氨肽蛋白 [VCP];p97)的小分
KB-0742 dihydrochloride
(Catalog# : 24020, Cas# :
2416874-75-2
)
KB-0742 是一种有效的、选择性的、口服生物可利用的 CDK9 小分子抑
KP-302 ( Synonyms: Lucid-21-302 ; Lucid-MS )
(Catalog# : 20641, Cas# :
2082765-42-0
)
KP-302 ( Synonyms: Lucid-21-302 ; Lucid-MS ) 是一种蛋白质精氨酸脱亚胺酶的
KDM5-C49
(Catalog# : 20493, Cas# :
1596348-16-1
)
KDM5-C49 is a potent and selective inhibitor of KDM5 (also known as JARID1). KDM5-C49
KSQ-4279
(Catalog# : 20472, Cas# :
2446480-97-1
)
KSQ-4279 is a USP1 and PARP inhibitor. KSQ-4279 showed anti-proliferative effects in
KY19382
(Catalog# : L20334, Cas# :
2226664-93-1
)
KY19382 is an orally active dual inhibitor of CXXC5-DVL and GSK3β
KPI-10
(Catalog# : 20277, Cas# :
888032-58-4
)
KPI-10 is a new compound currently being studied for its efficacy in the treatment of
KUN56321
(Catalog# : 21246, Cas# :
1771756-32-1
)
KUN56321 is a luminescent agent. The application of KUN56321 comprises: coating the f
KO-947
(Catalog# : 20122101, Cas# :
1695533-89-1
)
KO-947 is a potent and selective ERK inhibitor with slow dissociation kinetics. KO-94
KY-226
(Catalog# : 2061304)
KY-226 is a protein tyrosine phosphatase 1B (PTP1B) inhibitor that protects neurons f
Kinesore
(Catalog# : 193203, Cas# :
363571-83-9
)
Kinesore是肌动蛋白-1在细胞微管动力学调控中的激活因子。它已被
KH7
(Catalog# : 19362, Cas# :
330676-02-3
)
KH7是一种新型的可溶性腺苷酸环化酶(Sac)抑制剂。
KINK-1
(Catalog# : 192152, Cas# :
600734-06-3
)
IKKßKINK-1是一种抑制剂,阻止NF-kappaB激活。
KHS101盐酸盐
(Catalog# : 191281, Cas# :
1784282-12-7
)
KHS101 HCl是一种转化酸性卷曲蛋白3 (TACC3)的抑制剂。它的作用是通
KU59403
(Catalog# : 19123, Cas# :
845932-30-1
)
KU59403是一种有效的选择性ATM(共济失调毛细血管扩张突变)抑制剂,
KC01
(Catalog# : 1810294, Cas# :
1646795-59-6
)
KC01是ABHD16A的共价抑制剂。ABHD16A是一种磷脂酰丝氨酸(PS)脂肪酶,
KG-501
(Catalog# : 1810226, Cas# :
18228-17-6
)
KG-501是cAMP反应元件结合蛋白(CREB)抑制剂。
KYP-2047
(Catalog# : 187124, Cas# :
796874-99-2
)
KYP-2047是一种非常有效的、选择性的Prolyl寡肽酶(POP)抑制剂,也被
KGP-94
(Catalog# : 3291806, Cas# :
1131456-28-4
)
KGP94 is a reversible, time-dependent and competitive inhibitor of human cathepsin L.
KIN-1148
(Catalog# : 184121, Cas# :
1428729-56-9
)
KIN-1148是一个IRF3激动剂。KIN1148诱导剂量依赖性IRF3核易位和特异性
KKL-10
(Catalog# : 184217, Cas# :
952849-76-2
)
KKL-10是一种抗菌药物。KKL-10在体外和体外感染中均表现出了对弱毒
KI-696
(Catalog# : 1710132, Cas# :
1799974-70-1
)
ki-696代表一个优良的低分子量的工具来研究体内Keap1与Nrf2-Nrf2的相
KAF-156
(Catalog# : 20178211, Cas# :
1261113-96-5
)
KAF-156,也称为GNF-156, 是一种可治疗疟疾的抗疟药。
KM11060
(Catalog# : 17031301, Cas# :
774549-97-2
)
KM11060是一种突变的F508del囊性纤维化跨膜电导调节器(CFTR)。CFTR基因
KRIBB11
(Catalog# : 17031014, Cas# :
342639-96-7
)
KRIBB11废除了热触觉荧光素酶活动的IC50 1.2μM。它是转录因子热休克
Ki8751
(Catalog# : 17022703, Cas# :
228559-41-9
)
Ki8751是一种强力的、选择性的VEGFR- 2酪氨酸激酶(IC50 = 0.9 nM)的抑制
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AD-8007
(Catalog# : 26A018, Cas# :
1497439-74-3
)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
ZY-444
(Catalog# : 26A020, Cas# :
1802650-31-2
)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
AD-5584
(Catalog# : 26A019, Cas# :
2306525-79-9
)
AD-5584是一种新型脑渗透性ACSS2抑制剂。
IDB-003
(Catalog# : 26A017, Cas# :
3079716-11-0
)
IDB-003在体内抑制MDA-MB-231肿瘤生长。
Vafidemstat
(Catalog# : 18891, Cas# :
1357362-02-7
)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
LLL12
(Catalog# : 25075, Cas# :
1260247-42-4
)
LLL12是一种强效的STAT3抑制剂。LLL12在小鼠异种移植物模型中显示出
ECC-5004
(Catalog# : 26A015, Cas# :
2758659-09-3
)
ECC5004是一款每日一次、低剂量、小分子GLP-1受体激动剂。
SILA-123
(Catalog# : 26A014, Cas# :
2911585-37-8
)
SILA-123是一种II型FLT3抑制剂,对FLT3-WT(IC50=2.1 nM)和FLT3-ITD(IC50=1
Encaleret sulfate
(Catalog# : 26A013, Cas# :
1214922-52-7
)
Encaleret是一种正在研究的钙敏感受体的小分子拮抗剂,用于钙稳态
Iadademstat ( ORY-1001 ) hydrochloride
(Catalog# : 26A011, Cas# :
1431303-72-8
)
Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶