武汉永璨生物科技有限公司
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抑制剂/受体激动剂
Angiogenesis
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Bromides
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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产品名字索引 K
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产品名字索引 K
KH-3
(Catalog# : 24143, Cas# :
1215115-03-9
)
KH-3 is a potent RNA-binding protein Hu antigen R (HuR) inhibitor with an IC50 value
KB-0742
(Catalog# : 24040, Cas# :
2416873-83-9
)
KB-0742 是一种有效的,选择性的和具有口服活性的 CDK9 抑制剂。
KUS121
(Catalog# : 20676, Cas# :
1357164-52-3
)
KUS-121 是一种过渡内质网 ATP 酶(含缬氨肽蛋白 [VCP];p97)的小分
KB-0742 dihydrochloride
(Catalog# : 24020, Cas# :
2416874-75-2
)
KB-0742 是一种有效的、选择性的、口服生物可利用的 CDK9 小分子抑
KP-302 ( Synonyms: Lucid-21-302 ; Lucid-MS )
(Catalog# : 20641, Cas# :
2082765-42-0
)
KP-302 ( Synonyms: Lucid-21-302 ; Lucid-MS ) 是一种蛋白质精氨酸脱亚胺酶的
KDM5-C49
(Catalog# : 20493, Cas# :
1596348-16-1
)
KDM5-C49 is a potent and selective inhibitor of KDM5 (also known as JARID1). KDM5-C49
KSQ-4279
(Catalog# : 20472, Cas# :
2446480-97-1
)
KSQ-4279 is a USP1 and PARP inhibitor. KSQ-4279 showed anti-proliferative effects in
KY19382
(Catalog# : L20334, Cas# :
2226664-93-1
)
KY19382 is an orally active dual inhibitor of CXXC5-DVL and GSK3β
KPI-10
(Catalog# : 20277, Cas# :
888032-58-4
)
KPI-10 is a new compound currently being studied for its efficacy in the treatment of
KUN56321
(Catalog# : 21246, Cas# :
1771756-32-1
)
KUN56321 is a luminescent agent. The application of KUN56321 comprises: coating the f
KO-947
(Catalog# : 20122101, Cas# :
1695533-89-1
)
KO-947 is a potent and selective ERK inhibitor with slow dissociation kinetics. KO-94
KY-226
(Catalog# : 2061304)
KY-226 is a protein tyrosine phosphatase 1B (PTP1B) inhibitor that protects neurons f
Kinesore
(Catalog# : 193203, Cas# :
363571-83-9
)
Kinesore是肌动蛋白-1在细胞微管动力学调控中的激活因子。它已被
KH7
(Catalog# : 19362, Cas# :
330676-02-3
)
KH7是一种新型的可溶性腺苷酸环化酶(Sac)抑制剂。
KINK-1
(Catalog# : 192152, Cas# :
600734-06-3
)
IKKßKINK-1是一种抑制剂,阻止NF-kappaB激活。
KHS101盐酸盐
(Catalog# : 191281, Cas# :
1784282-12-7
)
KHS101 HCl是一种转化酸性卷曲蛋白3 (TACC3)的抑制剂。它的作用是通
KU59403
(Catalog# : 19123, Cas# :
845932-30-1
)
KU59403是一种有效的选择性ATM(共济失调毛细血管扩张突变)抑制剂,
KC01
(Catalog# : 1810294, Cas# :
1646795-59-6
)
KC01是ABHD16A的共价抑制剂。ABHD16A是一种磷脂酰丝氨酸(PS)脂肪酶,
KG-501
(Catalog# : 1810226, Cas# :
18228-17-6
)
KG-501是cAMP反应元件结合蛋白(CREB)抑制剂。
KYP-2047
(Catalog# : 187124, Cas# :
796874-99-2
)
KYP-2047是一种非常有效的、选择性的Prolyl寡肽酶(POP)抑制剂,也被
KGP-94
(Catalog# : 3291806, Cas# :
1131456-28-4
)
KGP94 is a reversible, time-dependent and competitive inhibitor of human cathepsin L.
KIN-1148
(Catalog# : 184121, Cas# :
1428729-56-9
)
KIN-1148是一个IRF3激动剂。KIN1148诱导剂量依赖性IRF3核易位和特异性
KKL-10
(Catalog# : 184217, Cas# :
952849-76-2
)
KKL-10是一种抗菌药物。KKL-10在体外和体外感染中均表现出了对弱毒
KI-696
(Catalog# : 1710132, Cas# :
1799974-70-1
)
ki-696代表一个优良的低分子量的工具来研究体内Keap1与Nrf2-Nrf2的相
KAF-156
(Catalog# : 20178211, Cas# :
1261113-96-5
)
KAF-156,也称为GNF-156, 是一种可治疗疟疾的抗疟药。
KM11060
(Catalog# : 17031301, Cas# :
774549-97-2
)
KM11060是一种突变的F508del囊性纤维化跨膜电导调节器(CFTR)。CFTR基因
KRIBB11
(Catalog# : 17031014, Cas# :
342639-96-7
)
KRIBB11废除了热触觉荧光素酶活动的IC50 1.2μM。它是转录因子热休克
Ki8751
(Catalog# : 17022703, Cas# :
228559-41-9
)
Ki8751是一种强力的、选择性的VEGFR- 2酪氨酸激酶(IC50 = 0.9 nM)的抑制
KN-93 phosphate
(Catalog# : 16123029, Cas# :
1188890-41-6
)
KN-93 is a CaMKII inhibitor. KN-93 suppresses ventricular arrhythmia induced by LQT2
K-7174
(Catalog# : 16123028, Cas# :
191089-59-5
)
K-7174 is a novel orally active, potent proteasome inhibitor. K-7174 exerts anti-myel
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AZD0095
(Catalog# : 237072, Cas# :
2750001-23-9
)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2-MNG
(Catalog# : 24129, Cas# :
2101538-28-5
)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
MAT2A-IN-9
(Catalog# : 25147, Cas# :
2439277-80-0
)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
Acoramidis hydrochloride
(Catalog# : 24068, Cas# :
2242751-53-5
)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
Crelosidenib
(Catalog# : 24101, Cas# :
2230263-60-0
)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
LOXO-435
(Catalog# : 25080, Cas# :
2833703-74-3
)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
Gridegalutamide
(Catalog# : 25138, Cas# :
2446928-30-7
)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
Chiauranib
(Catalog# : 25146, Cas# :
1256349-48-0
)
Chiauranib also known as orally available, small molecule inhibitor of select serine-