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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
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产品名字索引 O
Ofirnoflast
(Catalog# : 26A007, Cas# :
2731294-23-6
)
Ofirnoflast是一种口服生物可利用的NEK7抑制剂。
Oveporexton ( TAK-861 )
(Catalog# : 25194, Cas# :
2460722-04-5
)
Oveporexton是一种口服小分子选择性食欲素2型受体(OX2R)激动剂。
Opakalim
(Catalog# : 25193, Cas# :
2376397-93-0
)
Opakalim(BHV-7000)是Kv7.2/7.3钾通道(KCNQ2/3)的口服小分子激活剂,
Olomorasibum
(Catalog# : 25139, Cas# :
2771246-13-8
)
Olomorasibumis a Kirsten rat sarcoma viral oncogene homolog (KRAS) inhibitor, antineo
Orelabrutinib
(Catalog# : 25116, Cas# :
1655504-04-3
)
Orelabrutinib, also known as ICP-022, is a potent, orally active, and irreversible Br
Orteronel
(Catalog# : 25083, Cas# :
566939-85-3
)
Orterone, also known as TAK-700, is an orally bioavailable non-steroidal androgen syn
OPN expression inhibitor 1
(Catalog# : 25060, Cas# :
2257492-95-6
)
OPN expression inhibitor 1 (Compound 11) is an osteopontin (OPN) expression inhibitor
Opiranserin HCl
(Catalog# : 25040, Cas# :
1440796-75-7 (HCl)
)
Opiranserin HCl is a glycine transporter inhibitor and serotonin receptor antagonist.
Ocedurenone
(Catalog# : 24091, Cas# :
1359969-24-6
)
Ocedurenone is a non-steroidal mineralocorticoid receptor antagonist.
Opevesostat
(Catalog# : 24047, Cas# :
2231294-96-3
)
Opevesostat is cholesterol side-chain cleavage enzyme (CYP11A1) inhibitor.
Olverembatinib (GZD824)
(Catalog# : 24046, Cas# :
1257628-77-5
)
Olverembatinib, also known as GZD824, is a novel orally bioavailable inhibitor agains
OATD-02
(Catalog# : 20642, Cas# :
2146132-73-0
)
OATD-02 是一种口服双精氨酸酶抑制剂(ARG1 和 ARG2),目前在 Molecu
Orismilast ( LEO-32731 )
(Catalog# : 20625, Cas# :
1353546-86-7
)
Orismilast是一种磷酸二酯酶4型(PDE4)抑制剂。
Odevixibat
(Catalog# : 20600, Cas# :
501692-44-0
)
Odevixibat, also known as AZD 8294, is a potent, once-daily, non-systemic ileal bile
O4I4
(Catalog# : 20571, Cas# :
412008-21-0
)
O4I4 (compound 23) is a OCT4-inducing compound with metabolical stability.
orforglipron
(Catalog# : 20537, Cas# :
2212020-52-3
)
Orforglipron, also known as LY3502970, and OWL-833, is a Novel Non-Peptidyl Oral Gluc
omaveloxolone
(Catalog# : 20530, Cas# :
1474034-05-3
)
Omaveloxolone, also known as RTA-408, is a member of the synthetic oleanane triterpen
Osanetant
(Catalog# : 20505, Cas# :
160492-56-8 (free base)
)
Osanetant is a tachykinin NK3 antagonist potentially for the treatment of schizophren
Obicetrapib
(Catalog# : 20314, Cas# :
866399-87-3
)
Obicetrapib (also known as AMG-899, TA-8995, and DEX-001) is a cholesteryl ester tran
ONC201 HCl
(Catalog# : 20305, Cas# :
1638178-82-1
)
ONC-201, also known as TIC10 and imipridone, is a potent, orally active, and stable s
OUN20985v
(Catalog# : 2091912, Cas# :
2244520-98-5
)
OUN20985, also known as Homo-PROTAC cereblon degrader 1, is a cereblon degrader. OUN2
OATD-01 (GLPG-4716)
(Catalog# : 208191, Cas# :
2088453-21-6
)
OATD-01 (GLPG-4716)是一种有效的酸性哺乳动物几丁质酶(AMCase)和壳
Oroxylin A
(Catalog# : 2071536, Cas# :
480-11-5
)
Oroxylin A is a flavonoid that inhibits decreases in cell viability and increases in
O304
(Catalog# : 2071504, Cas# :
1261289-04-6
)
O-304 is a pan-activator of AMP-activated protein kinase (AMPK). It increases levels
olutasidenib
(Catalog# : 20791, Cas# :
1887014-12-1
)
Olutasidenib(FT-2102)是一种有效的突变体选择性IDH1抑制剂。 Olutasi
OUN87710
(Catalog# : 2051503, Cas# :
502887-71-0
)
OUN87710, also known as MMP-9-IN-1 is a specific matrix metalloproteinase-9 (MMP-9) i
2-oxo-5,5-diphenyltetrahydro-4-furancarboxylic acid
(Catalog# : 204123, Cas# :
79371-39-4
)
Oteseconazole
(Catalog# : 111895, Cas# :
1340593-59-0
)
Oteseconazole,也称为 VT-1161,是第一个批准的口服生物利用度和选择
ONC206
(Catalog# : 111891, Cas# :
1638178-87-6
)
ONC206 is a chemical analogue of ONC201. ONC206 is a benzyl-flurobenzyl imipridone th
Ogerin
(Catalog# : 193186, Cas# :
1309198-71-7
)
Ogerin是一种选择性的GPR68 PAM,在野生型小鼠中抑制恐惧条件反射的
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
CT1812 ( Zervimesine )
(Catalog# : 193283, Cas# :
1802632-22-9
)
CT-1812是一种同类首创的、可口服的sigma-2/PGRMC1拮抗剂(αβ寡聚体
BLU-808
(Catalog# : 26A024, Cas# :
3041025-10-6
)
BLU-808是一种针对肥大细胞疾病的野生型c-KIT的强效且具有选择性的
Zedoresertib
(Catalog# : 26A023, Cas# :
2243882-74-6
)
Zedoresertib(Debio 0123)是一种脑渗透剂,高选择性WEE1激酶抑制剂。
BEN-28010
(Catalog# : 26A022, Cas# :
3033961-38-2
)
BEN-28010是一种自由脑渗透剂,强效且具有选择性的CHK1抑制剂。
4-((2-(甲氨基)-6-(2,2,2-三氟乙基)噻吩并[2,3-d]嘧啶-4-基)氨基)哌啶-1-甲酸叔丁酯
(Catalog# : 26B007, Cas# :
3107291-07-3
)
Muvalaplin
(Catalog# : 20528, Cas# :
2565656-70-2
)
Muvalaplin是一种小分子,通过干扰载脂蛋白(a)与载脂蛋白B100的结合
MAT2A-IN-22
(Catalog# : 26A021, Cas# :
2925330-18-1
)
MAT2A-IN-22 (Compound 29-1) 是一种可透过血脑屏障的和口服有效的 MAT2A
AD-8007
(Catalog# : 26A018, Cas# :
1497439-74-3
)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
ZY-444
(Catalog# : 26A020, Cas# :
1802650-31-2
)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
AD-5584
(Catalog# : 26A019, Cas# :
2306525-79-9
)
AD-5584是一种新型脑渗透性ACSS2抑制剂。