武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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Aldehydes
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Bromides
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
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产品名字索引 O
Olomorasibum
(Catalog# : 25139, Cas# :
2771246-13-8
)
Olomorasibumis a Kirsten rat sarcoma viral oncogene homolog (KRAS) inhibitor, antineo
Orelabrutinib
(Catalog# : 25116, Cas# :
1655504-04-3
)
Orelabrutinib, also known as ICP-022, is a potent, orally active, and irreversible Br
Orteronel
(Catalog# : 25083, Cas# :
566939-85-3
)
Orterone, also known as TAK-700, is an orally bioavailable non-steroidal androgen syn
OPN expression inhibitor 1
(Catalog# : 25060, Cas# :
2257492-95-6
)
OPN expression inhibitor 1 (Compound 11) is an osteopontin (OPN) expression inhibitor
Opiranserin HCl
(Catalog# : 25040, Cas# :
1440796-75-7 (HCl)
)
Opiranserin HCl is a glycine transporter inhibitor and serotonin receptor antagonist.
Ocedurenone
(Catalog# : 24091, Cas# :
1359969-24-6
)
Ocedurenone is a non-steroidal mineralocorticoid receptor antagonist.
Opevesostat
(Catalog# : 24047, Cas# :
2231294-96-3
)
Opevesostat is cholesterol side-chain cleavage enzyme (CYP11A1) inhibitor.
Olverembatinib (GZD824)
(Catalog# : 24046, Cas# :
1257628-77-5
)
Olverembatinib, also known as GZD824, is a novel orally bioavailable inhibitor agains
OATD-02
(Catalog# : 20642, Cas# :
2146132-73-0
)
OATD-02 是一种口服双精氨酸酶抑制剂(ARG1 和 ARG2),目前在 Molecu
Orismilast ( LEO-32731 )
(Catalog# : 20625, Cas# :
1353546-86-7
)
Orismilast是一种磷酸二酯酶4型(PDE4)抑制剂。
Odevixibat
(Catalog# : 20600, Cas# :
501692-44-0
)
Odevixibat, also known as AZD 8294, is a potent, once-daily, non-systemic ileal bile
O4I4
(Catalog# : 20571, Cas# :
412008-21-0
)
O4I4 (compound 23) is a OCT4-inducing compound with metabolical stability.
orforglipron
(Catalog# : 20537, Cas# :
2212020-52-3
)
Orforglipron, also known as LY3502970, and OWL-833, is a Novel Non-Peptidyl Oral Gluc
omaveloxolone
(Catalog# : 20530, Cas# :
1474034-05-3
)
Omaveloxolone, also known as RTA-408, is a member of the synthetic oleanane triterpen
Osanetant
(Catalog# : 20505, Cas# :
160492-56-8 (free base)
)
Osanetant is a tachykinin NK3 antagonist potentially for the treatment of schizophren
Obicetrapib
(Catalog# : 20314, Cas# :
866399-87-3
)
Obicetrapib (also known as AMG-899, TA-8995, and DEX-001) is a cholesteryl ester tran
ONC201 HCl
(Catalog# : 20305, Cas# :
1638178-82-1
)
ONC-201, also known as TIC10 and imipridone, is a potent, orally active, and stable s
OUN20985v
(Catalog# : 2091912, Cas# :
2244520-98-5
)
OUN20985, also known as Homo-PROTAC cereblon degrader 1, is a cereblon degrader. OUN2
OATD-01 (GLPG-4716)
(Catalog# : 208191, Cas# :
2088453-21-6
)
OATD-01 (GLPG-4716)是一种有效的酸性哺乳动物几丁质酶(AMCase)和壳
Oroxylin A
(Catalog# : 2071536, Cas# :
480-11-5
)
Oroxylin A is a flavonoid that inhibits decreases in cell viability and increases in
O304
(Catalog# : 2071504, Cas# :
1261289-04-6
)
O-304 is a pan-activator of AMP-activated protein kinase (AMPK). It increases levels
olutasidenib
(Catalog# : 20791, Cas# :
1887014-12-1
)
Olutasidenib(FT-2102)是一种有效的突变体选择性IDH1抑制剂。 Olutasi
OUN87710
(Catalog# : 2051503, Cas# :
502887-71-0
)
OUN87710, also known as MMP-9-IN-1 is a specific matrix metalloproteinase-9 (MMP-9) i
2-oxo-5,5-diphenyltetrahydro-4-furancarboxylic acid
(Catalog# : 204123, Cas# :
79371-39-4
)
Oteseconazole
(Catalog# : 111895, Cas# :
1340593-59-0
)
Oteseconazole,也称为 VT-1161,是第一个批准的口服生物利用度和选择
ONC206
(Catalog# : 111891, Cas# :
1638178-87-6
)
ONC206 is a chemical analogue of ONC201. ONC206 is a benzyl-flurobenzyl imipridone th
Ogerin
(Catalog# : 193186, Cas# :
1309198-71-7
)
Ogerin是一种选择性的GPR68 PAM,在野生型小鼠中抑制恐惧条件反射的
ONO-8590580
(Catalog# : 1810162, Cas# :
1802661-73-9
)
ONO-8590580是一个GABAA α5的消极变构调制器。
奥瑞布林盐酸盐
(Catalog# : 186291, Cas# :
253426-24-3
)
奥瑞布林是一种合成的水溶性类似物,与combrestyatin A4类似,源自
寡霉素A
(Catalog# : 186154, Cas# :
579-13-5
)
寡霉素A,又称 MCH 32,是一种ATP合酶抑制剂。
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AZD0095
(Catalog# : 237072, Cas# :
2750001-23-9
)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2-MNG
(Catalog# : 24129, Cas# :
2101538-28-5
)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
MAT2A-IN-9
(Catalog# : 25147, Cas# :
2439277-80-0
)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
Acoramidis hydrochloride
(Catalog# : 24068, Cas# :
2242751-53-5
)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
Crelosidenib
(Catalog# : 24101, Cas# :
2230263-60-0
)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
LOXO-435
(Catalog# : 25080, Cas# :
2833703-74-3
)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
Gridegalutamide
(Catalog# : 25138, Cas# :
2446928-30-7
)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
Chiauranib
(Catalog# : 25146, Cas# :
1256349-48-0
)
Chiauranib also known as orally available, small molecule inhibitor of select serine-