武汉永璨生物科技有限公司
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
搜索
首页
网站地图
产品名字索引 O
按首字母搜索
A
B
C
D
E
F
G
H
I
J
K
L
M
N
O
P
Q
R
S
T
U
V
W
X
Y
Z
1
2
3
4
5
6
7
8
9
«
1
2
3
4
»
产品名字索引 O
Ofirnoflast
(Catalog# : 26A007, Cas# :
2731294-23-6
)
Ofirnoflast是一种口服生物可利用的NEK7抑制剂。
Oveporexton ( TAK-861 )
(Catalog# : 25194, Cas# :
2460722-04-5
)
Oveporexton是一种口服小分子选择性食欲素2型受体(OX2R)激动剂。
Opakalim
(Catalog# : 25193, Cas# :
2376397-93-0
)
Opakalim(BHV-7000)是Kv7.2/7.3钾通道(KCNQ2/3)的口服小分子激活剂,
Olomorasibum
(Catalog# : 25139, Cas# :
2771246-13-8
)
Olomorasibumis a Kirsten rat sarcoma viral oncogene homolog (KRAS) inhibitor, antineo
Orelabrutinib
(Catalog# : 25116, Cas# :
1655504-04-3
)
Orelabrutinib, also known as ICP-022, is a potent, orally active, and irreversible Br
Orteronel
(Catalog# : 25083, Cas# :
566939-85-3
)
Orterone, also known as TAK-700, is an orally bioavailable non-steroidal androgen syn
OPN expression inhibitor 1
(Catalog# : 25060, Cas# :
2257492-95-6
)
OPN expression inhibitor 1 (Compound 11) is an osteopontin (OPN) expression inhibitor
Opiranserin HCl
(Catalog# : 25040, Cas# :
1440796-75-7 (HCl)
)
Opiranserin HCl is a glycine transporter inhibitor and serotonin receptor antagonist.
Ocedurenone
(Catalog# : 24091, Cas# :
1359969-24-6
)
Ocedurenone is a non-steroidal mineralocorticoid receptor antagonist.
Opevesostat
(Catalog# : 24047, Cas# :
2231294-96-3
)
Opevesostat is cholesterol side-chain cleavage enzyme (CYP11A1) inhibitor.
Olverembatinib (GZD824)
(Catalog# : 24046, Cas# :
1257628-77-5
)
Olverembatinib, also known as GZD824, is a novel orally bioavailable inhibitor agains
OATD-02
(Catalog# : 20642, Cas# :
2146132-73-0
)
OATD-02 是一种口服双精氨酸酶抑制剂(ARG1 和 ARG2),目前在 Molecu
Orismilast ( LEO-32731 )
(Catalog# : 20625, Cas# :
1353546-86-7
)
Orismilast是一种磷酸二酯酶4型(PDE4)抑制剂。
Odevixibat
(Catalog# : 20600, Cas# :
501692-44-0
)
Odevixibat, also known as AZD 8294, is a potent, once-daily, non-systemic ileal bile
O4I4
(Catalog# : 20571, Cas# :
412008-21-0
)
O4I4 (compound 23) is a OCT4-inducing compound with metabolical stability.
orforglipron
(Catalog# : 20537, Cas# :
2212020-52-3
)
Orforglipron, also known as LY3502970, and OWL-833, is a Novel Non-Peptidyl Oral Gluc
omaveloxolone
(Catalog# : 20530, Cas# :
1474034-05-3
)
Omaveloxolone, also known as RTA-408, is a member of the synthetic oleanane triterpen
Osanetant
(Catalog# : 20505, Cas# :
160492-56-8 (free base)
)
Osanetant is a tachykinin NK3 antagonist potentially for the treatment of schizophren
Obicetrapib
(Catalog# : 20314, Cas# :
866399-87-3
)
Obicetrapib (also known as AMG-899, TA-8995, and DEX-001) is a cholesteryl ester tran
ONC201 HCl
(Catalog# : 20305, Cas# :
1638178-82-1
)
ONC-201, also known as TIC10 and imipridone, is a potent, orally active, and stable s
OUN20985v
(Catalog# : 2091912, Cas# :
2244520-98-5
)
OUN20985, also known as Homo-PROTAC cereblon degrader 1, is a cereblon degrader. OUN2
OATD-01 (GLPG-4716)
(Catalog# : 208191, Cas# :
2088453-21-6
)
OATD-01 (GLPG-4716)是一种有效的酸性哺乳动物几丁质酶(AMCase)和壳
Oroxylin A
(Catalog# : 2071536, Cas# :
480-11-5
)
Oroxylin A is a flavonoid that inhibits decreases in cell viability and increases in
O304
(Catalog# : 2071504, Cas# :
1261289-04-6
)
O-304 is a pan-activator of AMP-activated protein kinase (AMPK). It increases levels
olutasidenib
(Catalog# : 20791, Cas# :
1887014-12-1
)
Olutasidenib(FT-2102)是一种有效的突变体选择性IDH1抑制剂。 Olutasi
OUN87710
(Catalog# : 2051503, Cas# :
502887-71-0
)
OUN87710, also known as MMP-9-IN-1 is a specific matrix metalloproteinase-9 (MMP-9) i
2-oxo-5,5-diphenyltetrahydro-4-furancarboxylic acid
(Catalog# : 204123, Cas# :
79371-39-4
)
Oteseconazole
(Catalog# : 111895, Cas# :
1340593-59-0
)
Oteseconazole,也称为 VT-1161,是第一个批准的口服生物利用度和选择
ONC206
(Catalog# : 111891, Cas# :
1638178-87-6
)
ONC206 is a chemical analogue of ONC201. ONC206 is a benzyl-flurobenzyl imipridone th
Ogerin
(Catalog# : 193186, Cas# :
1309198-71-7
)
Ogerin是一种选择性的GPR68 PAM,在野生型小鼠中抑制恐惧条件反射的
«
1
2
3
4
»
产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AD-8007
(Catalog# : 26A018, Cas# :
1497439-74-3
)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
ZY-444
(Catalog# : 26A020, Cas# :
1802650-31-2
)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
AD-5584
(Catalog# : 26A019, Cas# :
2306525-79-9
)
AD-5584是一种新型脑渗透性ACSS2抑制剂。
IDB-003
(Catalog# : 26A017, Cas# :
3079716-11-0
)
IDB-003在体内抑制MDA-MB-231肿瘤生长。
Vafidemstat
(Catalog# : 18891, Cas# :
1357362-02-7
)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
LLL12
(Catalog# : 25075, Cas# :
1260247-42-4
)
LLL12是一种强效的STAT3抑制剂。LLL12在小鼠异种移植物模型中显示出
ECC-5004
(Catalog# : 26A015, Cas# :
2758659-09-3
)
ECC5004是一款每日一次、低剂量、小分子GLP-1受体激动剂。
SILA-123
(Catalog# : 26A014, Cas# :
2911585-37-8
)
SILA-123是一种II型FLT3抑制剂,对FLT3-WT(IC50=2.1 nM)和FLT3-ITD(IC50=1
Encaleret sulfate
(Catalog# : 26A013, Cas# :
1214922-52-7
)
Encaleret是一种正在研究的钙敏感受体的小分子拮抗剂,用于钙稳态
Iadademstat ( ORY-1001 ) hydrochloride
(Catalog# : 26A011, Cas# :
1431303-72-8
)
Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶