武汉永璨生物科技有限公司
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抑制剂/受体激动剂
Angiogenesis
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Amines
Amino Acids
Anilines
Boronic Acids
Bromides
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
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Peg Linkers
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Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
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产品名字索引 E
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产品名字索引 E
ECC-5004
(Catalog# : 26A015, Cas# :
2758659-09-3
)
ECC5004是一款每日一次、低剂量、小分子GLP-1受体激动剂。
Encaleret sulfate
(Catalog# : 26A013, Cas# :
1214922-52-7
)
Encaleret是一种正在研究的钙敏感受体的小分子拮抗剂,用于钙稳态
EDI-048
(Catalog# : 26A005, Cas# :
2767264-57-1
)
EDI048 是一种口服有效的Cryptosporidium PI4K 抑制剂。
Enterololin
(Catalog# : 26A001, Cas# :
1445830-39-6
)
肠毒素是一种对肠杆菌科物种具有靶向活性的抗菌化合物。
Emlenoflast ( 别名: MCC7840 ; IZD174)
(Catalog# : 25168, Cas# :
1995067-59-8
)
Emlenoflast(MCC7840,以前称为IZD174)是一种NLRP3炎症小体的抑制剂,
EP6
(Catalog# : 25161, Cas# :
1353567-32-4
)
EP6 is a 5-lipoxygenase (5-LO) inhibitor. 5-LO is a crucial enzyme of the arachidonic
Elzovantinib
(Catalog# : 25160, Cas# :
2271119-26-5
)
Elzovantinib, also known as TPX-0022 and CSF1R-IN-2, is an orally bioavailable CSF1R
Etavopivat
(Catalog# : 25141, Cas# :
2245053-57-8
)
Etavopivat, also known as FT-4202, is a pyruvate kinase activator. Etavopivat decreas
Etripamil
(Catalog# : 25123, Cas# :
1593673-23-4
)
Etripamil is a calcium channel blocker. Calcium channel blockers (CCB), calcium chann
E-7386
(Catalog# : 25086, Cas# :
1799824-08-0
)
E-7386 is an orally active CBP/beta-catenin modulator.
Emavusertib
(Catalog# : 25069, Cas# :
1801344-14-8
)
Emavusertib, also known as CA-4948 is a potent IRAK4/FLT3 inhibitor with anti-tumor a
Ecopipam ( SCH 39166 )
(Catalog# : 25065, Cas# :
112108-01-7
)
Ecopipam (SCH 39166) 是一种有效的、选择性、具有口服活性的多巴胺
Emraclidine
(Catalog# : 24118, Cas# :
2170722-84-4
)
Emraclidine, also known as CVL-231 and PF-06852231, is a novel, brain-penetrant, high
EG-2184
(Catalog# : 24075, Cas# :
2770297-66-8
)
EPZ-719
(Catalog# : 24032 , Cas# :
2697176-16-0
)
ERAS-801 ( JGK-068S )
(Catalog# : 20635, Cas# :
2490431-16-6
)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。
Edecesertib ( GS-5718 )
(Catalog# : 20636, Cas# :
2408839-73-4
)
GS-5718(Edecesertib)是一种强效、选择性、口服生物可利用的IRAK4抑
Ezurpimtrostat HCl
(Catalog# : 20607, Cas# :
1914148-73-4
)
Ezurpimtrostat is a palmitoyl protein thioesterase 1 (PPT-1) inhibitor.
EN460
(Catalog# : 20603, Cas# :
496807-64-8
)
EN460 is an endoplasmic reticulum oxidoreductase (ERO1) inhibitor. EN460 showed a dos
(E)-4-吗啉酮-2-烯酸盐酸盐
(Catalog# : 20546, Cas# :
1419865-05-6
)
1-乙基-1H-吡唑-4-甲醛
(Catalog# : 20523, Cas# :
304903-10-4
)
ethyl 5-chloro-6-fluoropyrazolo[1,5-a]pyrimidine-3-carboxylate
(Catalog# : 20480, Cas# :
2359650-50-1
)
Ervogastat (PF-06865571)
(Catalog# : 20449, Cas# :
2186700-33-2
)
Ervogastat (PF-06865571) 是一种具有全身作用的二酰基甘油酰基转移酶
ELQ300
(Catalog# : 20447, Cas# :
1354745-52-0
)
ELQ300 is a novel inhibitor of the mitochondrial cytochrome bc1 complex (complex III
Etrumadenant
(Catalog# : 20443, Cas# :
2239273- 34-6
)
Etrumadenant, also known as AB928, is a dual antagonist of the A2aR and A2bR adenosin
E6446
(Catalog# : 20436, Cas# :
1219925-73-1
)
E6446 is a TLR inhibitor. E6446 inhibits Toll-like receptor (TLR)7 and 9 signaling. E
Etrumadenant
(Catalog# : 171455, Cas# :
2239273-34-6
)
Etrumadenant, also known as AB928, is a dual antagonist of the A2aR and A2bR adenosin
EZM0414
(Catalog# : 171652, Cas# :
2411748-50-8
)
EZM0414 是一种有效的、选择性的、具有口服生物利用度的 SETD2 抑制
4,6-二羟基哒嗪-3-甲酸乙酯
(Catalog# : 20390, Cas# :
1352925-63-3
)
5-(Ethoxycarbonyl)-2-formyl-4-methyl-1H-pyrrole-3-propanoic Acid Methyl Ester
(Catalog# : G20384, Cas# :
54278-05-6
)
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AD-8007
(Catalog# : 26A018, Cas# :
1497439-74-3
)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
ZY-444
(Catalog# : 26A020, Cas# :
1802650-31-2
)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
AD-5584
(Catalog# : 26A019, Cas# :
2306525-79-9
)
AD-5584是一种新型脑渗透性ACSS2抑制剂。
IDB-003
(Catalog# : 26A017, Cas# :
3079716-11-0
)
IDB-003在体内抑制MDA-MB-231肿瘤生长。
Vafidemstat
(Catalog# : 18891, Cas# :
1357362-02-7
)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
LLL12
(Catalog# : 25075, Cas# :
1260247-42-4
)
LLL12是一种强效的STAT3抑制剂。LLL12在小鼠异种移植物模型中显示出
ECC-5004
(Catalog# : 26A015, Cas# :
2758659-09-3
)
ECC5004是一款每日一次、低剂量、小分子GLP-1受体激动剂。
SILA-123
(Catalog# : 26A014, Cas# :
2911585-37-8
)
SILA-123是一种II型FLT3抑制剂,对FLT3-WT(IC50=2.1 nM)和FLT3-ITD(IC50=1
Encaleret sulfate
(Catalog# : 26A013, Cas# :
1214922-52-7
)
Encaleret是一种正在研究的钙敏感受体的小分子拮抗剂,用于钙稳态
Iadademstat ( ORY-1001 ) hydrochloride
(Catalog# : 26A011, Cas# :
1431303-72-8
)
Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶