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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
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Anilines
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Pyrimidines
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Cas号索引 9
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Cas号索引 9
955979-06-3 | (R)-tert-Butyl 2-isopropylpiperazine-1-carboxylate hydrochloride
(Catalog# : 81903)
Coming soon!
911222-45-2 | Rabusertib(LY2603618)
(Catalog# : 52807)
LY2603618(IC-83) is a potent and selective small molecule inhibitor of Chk1 protein k
956697-53-3 | Sonidegib (LDE-225)
(Catalog# : 21232)
Sonidegib, also known as, erismodegib, LDE225, NVP-LDE225, is an orally bioavailable
910562-15-1 | Simenepag
(Catalog# : 1810172)
Simenepag,又名AGN-210676,是一种用于治疗青光眼和高眼压的小分子
923359-38-0 | SAR407899游离
(Catalog# : 185115)
SAR407899是一种有效且具有选择性的、前景的抗高血压活性Rho激酶抑
927871-76-9 | S107 HCl
(Catalog# : 1791111)
S107是类型1 利阿诺定受体(RYR1)稳定剂;结合 RyR1提高calstabin-1亲
908112-43-6 | SNX-2112
(Catalog# : 179815)
SNX-2112,又称为PF 04928473,是一种HSP90抑制剂,目前正在进行1期临
940929-33-9 | SB-743921盐酸盐
(Catalog# : 17011609)
SB-743921是一种具有潜在抗肿瘤性质的合成小分子。
923262-96-8 | SAR407899 HCl
(Catalog# : 17011606)
SAR407899是一种具有良好的抗高血压活性的强效和选择性的激酶抑制
910462-43-0 | 4SC-202
(Catalog# : 161227110)
4SC-202 is an orally bioavailable benzamide and inhibitor of human class I histone de
909089-13-0 | SKL2001
(Catalog# : 16122784)
SKL2001 is a novel agonist of the Wnt/-catenin pathway that disrupts the Axin/-cateni
913822-46-5 | SC75741
(Catalog# : 16122748)
SC75741 is a potent NF-B inhibitor with EC50 of 200 nM.SC75741 shows immunosuppressiv
906805-42-3 | SCH 546738
(Catalog# : 161113)
SCH 546738 is a novel, potent and non-competitive small molecule CXCR3 antagonist wit
923604-59-5 | Simeprevir
(Catalog# : 16062201)
Simeprevir (formerly TMC435; trade name Olysio) is a drug for the treatment and cure
929901-49-5 | SGI-110
(Catalog# : 011806)
SGI-110 is a small molecule, DNMT inhibitor with demonstrated activity in restoring s
942183-80-4 | SCH772984
(Catalog# : 11106)
SCH772984 is a novel, specific inhibitor of ERK1/2 with IC50 of 4 nM and 1 nM, respec
936487-67-1 | SF1126
(Catalog# : 010804)
SF1126 is a water soluble, small-molecule prodrug containing the pan-PI3K/mTOR inhibi
957135-43-2 | SM-164
(Catalog# : 122802)
SM-164 is a potent cell-permeable and bivalent Smac mimetic which bind to a XIAP prot
912545-86-9 | SAG
(Catalog# : 92802)
SAG is a potent Smoothened (Smo) receptor agonist (Kd = 59 nM); antagonizes Cyclopami
946053-90-3 | (S)-4-Fluoro-2,3-dihydro-1H-inden-1-amine
(Catalog# : 91115)
Coming soon!
911417-87-3 | SLx-2119
(Catalog# : 91002)
SLx-2119(KD-025) is a small molecule and selective inhibitor of ROCK2 with IC50 of 10
916214-30-7 | (S)-1-Boc-3-Aminomethylpyrrolidine hydrochloride
(Catalog# : 83120)
Coming soon!
943760-74-5 | (1S)-1-(4-chloro-3-methylphenyl)ethanamine
(Catalog# : 81017)
Coming soon!
942271-61-6 | 4-(4-甲基哌嗪-1-基)-2-硝基苯甲酸叔丁酯
(Catalog# : 24062)
95727-86-9 | 2-氰基-5-三氟甲基吡啶
(Catalog# : 24061)
928659-17-0 | Triazavirin ( Riamilovir )
(Catalog# : 2071631)
Triazavirin是一种广谱抗病毒药物,由乌拉尔联邦大学,俄罗斯科学
925436-46-0 | tert-butyl 4-[[6-[2-(quinoxaline-2-carbonylamino)phenyl]imidazo[2,1-b][1,3]thiazol-3-yl]methyl]piperazine-1-carboxylate
(Catalog# : 2062035)
951395-08-7 | Tafamidis meglumine
(Catalog# : 193183)
Tafamidis meglumine,也被称为Fx-1006或PF-06291826,是一种改善经胸腺素
94497-51-5 | 他米巴罗汀
(Catalog# : 191254)
他米巴罗汀,也称为SY-1425,是一种具有口服活性的合成类维生素
903565-83-3 | 托格列净
(Catalog# : 184311)
托格列净,也称为CSG452,是一种高效、高选择性的SGLT2抑制剂,在
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
3054692-62-2 | ECI830
(Catalog# : 26A031)
ECI830是一种实验性的CDK2抑制剂。
1394076-92-6 | GNE-317
(Catalog# : 52282)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
3118994-80-9 | DPTX-3186
(Catalog# : 26A010)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
435327-40-5 | Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
1421936-85-7 | Iclepertin (BI-425809)
(Catalog# : 24084)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
4727-31-5 | Kartogenin ( KGN )
(Catalog# : 52215)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
218791-21-0 | Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
2311863-36-0 | Apecotrep (BI 764198)
(Catalog# : 26A048)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
902614-04-4 | Pantothenate kinase-IN-2
(Catalog# : 26A038)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
3062177-59-4 | BH-30643
(Catalog# : 26A047)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制