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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
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Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
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Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
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Oxazoles
Peg Linkers
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Pyridines
Pyrimidines
Quinolines
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Cas号索引 9
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Cas号索引 9
925701-49-1 | KU-60019
(Catalog# : 52576)
KU-60019 is an improved analogue of KU-55933, with IC50 of 6.3 nM for ATM
924835-67-6 | LP-184
(Catalog# : 24121)
LP-184 is an acylfulvene-derived prodrug activated by the oxidoreductase PTGR1 that a
935283-04-8 | Linzagolix
(Catalog# : 20266)
Linzagolix 是一种新型的口服 GnRH 受体拮抗剂,可有效治疗子宫内膜
915412-67-8 | LP-261
(Catalog# : 210507)
LP-261 is a novel tubulin targeting anticancer agent that binds at the colchicine sit
917111-49-0 | Lexibulin
(Catalog# : 19122)
Lexibulin,又称CYT997,是一种n型口服生物利用小分子,具有管蛋白
927961-18-0 | Lanifibranor
(Catalog# : 184177)
Lanifibranor,也叫IVA-337,是一种过氧化物酶体激活受体(PPAR)激动剂
934593-90-5 | LW6
(Catalog# : 17101618)
LW6减少HIF-1alpha蛋白表达不影响hif-1beta表达。
928134-65-0 | LCI699
(Catalog# : 17021314)
LCI699(Osilodrostat)是一种强有力的抑制剂11β-羟化酶,酶催化合成皮质
950455-15-9 | Liproxstatin-1
(Catalog# : 6111018)
Liproxstatin-1
910634-41-2 | Litronesib
(Catalog# : 611944)
Litronesib is a selective, allosteric inhibitor of Eg5, which may result in mitotic d
917111-44-5 | Lexibulin
(Catalog# : 122803)
Lexibulin is an orally bioavailable small-molecule with tubulin-inhibiting, vascular-
946518-60-1 | LY2409881 trihydrochloride
(Catalog# : 101914)
LY2409881 trihydrochloride is a novel selective inhibitor of IKK2 with IC50 of 30 nM;
942594-93-6 | Mavodelpar
(Catalog# : 20615)
Mavodelpar is a peroxisome proliferator activated receptor (PPAR) delta agonist.
928821-41-4 | MBX-8025 lysine anhydrous
(Catalog# : 20542)
MBX-8025 lysine anhydrous is a selective PPAR-delta agonist.
915412-80-5 | Methanone, (3,5-dibromophenyl)(2-methoxy-4-pyridinyl)-
(Catalog# : 20414)
944547-46-0 | Mycro3
(Catalog# : L20346)
Mycro3 is an inhibitor of Myc-Max dimerization.
94164-88-2 | MDK4882
(Catalog# : 1810301)
MDK4882也称为PKM2抑制剂或化学物3k,是一种 PKM2抑制剂。
957118-49-9 | MK-3207
(Catalog# : 185284)
MK-3207是一种有效的口服降钙素基因相关肽受体拮抗剂。
947914-18-3 | ML365
(Catalog# : 184215)
ML365 is a potent and selective K2P3.1 TASK-1 channel blocker.
92831-11-3 | MN-64
(Catalog# : 17030717)
MN-64 是一种有效的、选择性的Tankyrase 1和2抑制剂(IC50值分别为6和
926927-61-9 | Motolimod
(Catalog# : 6111017)
Motolimod
935273-79-3 | MK-4101
(Catalog# : 6111008)
MK-4101 is a potent SMO Inhibitor of the Hedgehog PathwayMK-4101 is a potent SMO Inhi
916489-36-6 | MS417
(Catalog# : 16070106)
MS417, also known as GTPL7512, is a potent and selective BRD4 inhibitor. MS417 inhibi
955365-80-7 | MK-1775
(Catalog# : 011110)
MK-1775 is a potent and selective Wee1 inhibitor with IC50 of 5.2 nM; hinders G2 DNA
917879-39-1 | MK-2461
(Catalog# : 010806)
MK-2461 is a novel ATP-competitive multitargeted inhibitor of activated c-Met.
924909-16-0 | 1-(4-methoxybenzyl)-1H-pyrazolo[3,4-b]pyridin-4-ol
(Catalog# : 5112803)
1-(4-methoxybenzyl)-1H-pyrazolo[3,4-b]pyridin-4-ol
921927-88-0 | methyl 2-formyl-1,3-thiazole-4-carboxylate
(Catalog# : 92215)
Coming soon!
916177-00-9 | 5-(methoxycarbonyl)-1-tosyl-1Hpyrrol-3-yl-3-boronic acid
(Catalog# : 92213)
Coming soon!
94413-64-6 | Methyl 2-cyanoisonicotinate
(Catalog# : 91702)
Coming soon!
913742-54-8 | Methyl (2S,4R)-4-Boc-aminopyrrolidine-2-carboxylate hydrochloride
(Catalog# : 90601)
Coming soon!
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2750001-23-9 | AZD0095
(Catalog# : 237072)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2101538-28-5 | 2-MNG
(Catalog# : 24129)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
2439277-80-0 | MAT2A-IN-9
(Catalog# : 25147)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
1898206-17-1 | Safusidenib
(Catalog# : 25149)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
2669009-92-9 | Atebimetinib
(Catalog# : 25148)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
2242751-53-5 | Acoramidis hydrochloride
(Catalog# : 24068)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
2230263-60-0 | Crelosidenib
(Catalog# : 24101)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
2833703-74-3 | LOXO-435
(Catalog# : 25080)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
2446928-30-7 | Gridegalutamide
(Catalog# : 25138)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
1256349-48-0 | Chiauranib
(Catalog# : 25146)
Chiauranib also known as orally available, small molecule inhibitor of select serine-