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抑制剂/受体激动剂
Angiogenesis
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Apoptosis
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Cytoskeleton
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MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
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分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
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Pyrimidines
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
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定制合成
工艺研发
订购信息
联系我们
公司简介
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Cas号索引 9
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Cas号索引 9
97207-47-1 | Meisoindigo
(Catalog# : 52542)
Meisoindigo(Natura-; N-Methylisoindigotin; Dian III), a derivative of Indigo naturali
936092-53-4 | N-tert-butyl-3-[(2-chloro-5-methylpyrimidin-4-yl)amino]benzenesulfonamide
(Catalog# : 2062304)
959551-10-1 | NIH-12848
(Catalog# : 1781103)
NIH-12848是一种普遍认为的磷脂酰肌醇5 -磷酸四激酶(PI5P4K)抑制剂。
912-60-7 | 那可汀盐酸盐
(Catalog# : 17022711)
那可汀, 也被称为麻醉药物,阿片烷,是一种来自罂粟科植物的be
923564-51-6 | Navitoclax (ABT-263)
(Catalog# : 16070102)
Navitoclax, also known as ABT-263, is an orally bioavailable, synthetic small-molecul
923288-90-8 | Nilotinib HCl hydrate
(Catalog# : 122901)
Nilotinib is an orally bioavailable aminopyrimidine-derivative Bcr-Abl tyrosine kinas
913830-15-6 | NS 9283
(Catalog# : 122828)
Coming soon!
95734-82-0 | Nedaplatin
(Catalog# : 122513)
Nedaplatin is a derivative of cisplatin and DNA damage agent.
940310-85-0 | NVP-BHG712
(Catalog# : 122213)
NVP-BHG712 is a specific EphB4 inhibitor with ED50 of 25 nM that discriminates betwee
956014-19-0 | Ns11021
(Catalog# : 120425)
Coming soon!
91419-53-3 | N-Boc-3-Cyanopiperidine
(Catalog# : 81713)
Coming soon!
951650-22-9 | NS11394
(Catalog# : 52567)
NS11394 is a potent and subtype-selective GABA(A) receptor-positive modulator; posses
923287-50-7 | Opicapone
(Catalog# : 6111514)
Opicapone(BIA 9-1067) is a long-acting, peripherally selective inhibitor of catechol-
936890-98-1 | OSI-027 HCl salt
(Catalog# : 161009007)
mTOR kinase inhibitor OSI-027 binds to and inhibits both the raptor-mTOR (TOR complex
951127-25-6 | Omarigliptin intermediate I
(Catalog# : 82718)
Coming soon!
919973-83-4 | OF-1
(Catalog# : 82407)
Selective BRPF1B and BRPF2 bromodomain inhibitor (Kd values are 100 and 500 nM respec
94790-37-1 | O-(Benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium Hexafluorophosphate
(Catalog# : 81023)
Coming soon!
935888-69-0 | Oprozomib
(Catalog# : 52630)
Oprozomib (ONX 0912; PR047) is an orally bioavailable inhibitor for CT-L activity of
960374-59-8 | ONX-0914 ( PR-957 )
(Catalog# : 52013)
ONX-0914 是免疫蛋白酶体 LMP7 和 LMP2 亚基的抑制剂,在多种自身免疫
98570-83-3 | Phylloflavan
(Catalog# : 24155)
Phylloflavan is an antileishmanial agent with an intracellular EC50 of 3.2 nM in RAW
903576-44-3 | Pitolisant HCl
(Catalog# : 20624)
Pitolisant, also known as Tiprolisant, BF2649 and Ciproxidine, is a histamine recepto
952021-60-2 | PF-477736
(Catalog# : 2071540)
PF-477736, also known as PF-00477736, is a potent CHK1 inhibitor with potential chemo
942425-68-5 | PHA-767491盐酸盐
(Catalog# : 184286)
PHA-767491,又名CAY10572,是一种有效的、具有ATP-竞争力的双cdc7/cdk9
939791-41-0 | PF-562271 HCl
(Catalog# : 179302)
PF-562271,也称为PF-562,271 and PF-271,是口服小分子与ATP竞争性粘着斑
95153-31-4 | 培哚普利
(Catalog# : 2017829)
培哚普利是一种有效且长效的血管紧张素转换酶抑制剂,可引起周
908115-27-5 | PF 04929113
(Catalog# : 2017826)
PF-04929113, 也称为SNX-5422,是一种针对人体热休克蛋白90(Hsp90)的合成
950762-95-5 | PCI-34051
(Catalog# : 17022402)
PCI-34051是一种有效的组蛋白去乙酰化酶8(HDAC8)特异性抑制剂,在其
944118-01-8 | Peficitinib (ASP015K, JNJ-54781532)
(Catalog# : 16122707)
Peficitinib (ASP015K, JNJ-54781532) is an orally bioavailable JAK inhibitor. Phase 3.
900185-02-6 | PIK-294
(Catalog# : 160926013)
PIK-294 is a highly selective inihibitor of the phosphoinositide 3-kinase (PI3K) p110
905579-51-3 | Pevonedistat
(Catalog# : 16071408)
Pevonedistat, also known as MLN-4924 and TAK-924, is a small molecule inhibitor of Ne
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2750001-23-9 | AZD0095
(Catalog# : 237072)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2101538-28-5 | 2-MNG
(Catalog# : 24129)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
2439277-80-0 | MAT2A-IN-9
(Catalog# : 25147)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
1898206-17-1 | Safusidenib
(Catalog# : 25149)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
2669009-92-9 | Atebimetinib
(Catalog# : 25148)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
2242751-53-5 | Acoramidis hydrochloride
(Catalog# : 24068)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
2230263-60-0 | Crelosidenib
(Catalog# : 24101)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
2833703-74-3 | LOXO-435
(Catalog# : 25080)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
2446928-30-7 | Gridegalutamide
(Catalog# : 25138)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
1256349-48-0 | Chiauranib
(Catalog# : 25146)
Chiauranib also known as orally available, small molecule inhibitor of select serine-