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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
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分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
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Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
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Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
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产品名字索引 P
PD 168 077
(Catalog# : 185156, Cas# :
190383-31-4
)
PD168077是一种多巴胺D4受体激动剂,对记忆巩固有促进作用。
PF-06462894
(Catalog# : 185155, Cas# :
1622291-66-0
)
PF-06462894是一种形态学上的mGlu5 (mGlu5 Ki = 6nm)。
PF-06291874
(Catalog# : 185154, Cas# :
1393124-08-7
)
PF-06291874是一种胰高血糖素受体拮抗剂,对2型糖尿病患者有效。
Poseltinib
(Catalog# : 185153, Cas# :
1353552-97-2
)
Poseltinib, 也称为HM-71224和LY3337641,一种酪氨酸激酶抑制剂。
Pibrentasvir
(Catalog# : 185148, Cas# :
1353900-92-1
)
Pibrentasvir,也被称为ABT-530,是一种蛋白酶抑制剂,可用于治疗丙
PP2 Analog
(Catalog# : 185147, Cas# :
309739-67-1
)
PP2 Analog是一种PP2类似物,它发挥蛋白质交易调制器的作用。
PP2
(Catalog# : 185146, Cas# :
172889-27-9
)
PP2,也被称为AG 1879,是一种经常被用于癌症研究的物质,作为src
PP1
(Catalog# : 185145, Cas# :
172889-26-8
)
PP1是一种有效的选择性Src家族蛋白酪氨酸激酶抑制剂。
Pocapavir
(Catalog# : 185144, Cas# :
146949-21-5
)
Pocapavir,也被称为SCH -48973和V-073,是一种强效、选择性的抗肠道病
PSMA617 TFA
(Catalog# : 185143, Cas# :
1702967-37-0
)
PSMA-617是一种配体,用于制造177Lu -PSMA-617,这是一种用于对抗癌症
Pyridostatin TFA盐
(Catalog# : 185142, Cas# :
1472611-44-1
)
Pyridostatin在细胞中稳定G-四链体(G4s),并通过DNA双链断裂(DSB)的形成
PF-06260933
(Catalog# : 18544, Cas# :
1811510-56-1
)
PF-06260933是一种有效且高选择性MAP4K4抑制剂。
PHA-767491盐酸盐
(Catalog# : 184286, Cas# :
942425-68-5
)
PHA-767491,又名CAY10572,是一种有效的、具有ATP-竞争力的双cdc7/cdk9
PLX51107
(Catalog# : 184285, Cas# :
1627929-55-8
)
PLX51107是一种高效、选择性的BRD4抑制剂或BET抑制剂,其体外和体内
PD 158780
(Catalog# : 184284, Cas# :
171179-06-9
)
PD 158780是表皮生长因子受体(EGFR) (IC50为0.08 nM)的酪氨酸激酶活性的
PZM21
(Catalog# : 184162, Cas# :
1997387-43-5
)
PZM21是强有力Gi活化剂,对μOR和最小β-arrestin-2具有特殊选择性的补
PF-9366
(Catalog# : 184107, Cas# :
72882-78-1
)
PF-9366是一种新型的人蛋氨酸腺苷转移酶2A (Mat2A),肝外同种型。
PFI-2盐酸盐
(Catalog# : 184106, Cas# :
1627607-87-7
)
在其他甲基转移酶和其他非表观遗传靶点上,PFI-2是一种具有IC50为
PCI-29732
(Catalog# : 184101, Cas# :
330786-25-9
)
PCI-29732是BTK抑制剂。它通过阻断B细胞抗原受体(BCR)介导的CD20+ B细
PF-0684000
(Catalog# : 184318, Cas# :
198474-05-4
)
PF-0684000,也称为EOS200271,是强有力的IDO-1抑制剂(IC50 0.15μM)。PF-06
PF-06409577
(Catalog# : 18434, Cas# :
1467057-23-3
)
PF-06409577是一种有效和具有选择的5腺苷酸活化蛋白激酶(AMPK)激活剂
PRN-1371
(Catalog# : 17101614, Cas# :
1802929-43-6
)
PRN-1371是一种共价键,不可逆的,高选择性的纤维母细胞生长因子
PF-5006739
(Catalog# : 17101612, Cas# :
1293395-67-1
)
PF-5006739是一种有效的CK1δ/ε抑制剂。PF-5006739对阿片类药物具有药
PF-04628935
(Catalog# : 17101611, Cas# :
1383719-97-8
)
PF-04628935是一种有效的关于胃肽感受器的拮抗激动剂,生长激素促
PIM447
(Catalog# : 1710134, Cas# :
1210608-43-7
)
PIM447,也称为lgh447,是一种有效的Moloney小鼠白血病(PIM)1, 2,和
PF-562271 HCl
(Catalog# : 179302, Cas# :
939791-41-0
)
PF-562271,也称为PF-562,271 and PF-271,是口服小分子与ATP竞争性粘着斑
Pemafibrate
(Catalog# : 179221, Cas# :
848259-27-8
)
Pemafibrate, also known as K-877 and (R)-K 13675, is a PPAR alpha agonist. (R)-K-1367
Pyridostatin TFA盐
(Catalog# : 1791517, Cas# :
179474-81-8
)
Pyridostatin稳定G-四链体(G4S)在细胞和诱导引起的DNA双链断裂形成
琥珀酸普卡比利
(Catalog# : 1791516, Cas# :
179474-85-2
)
琥珀酸普卡比利,也称为r-108512,是一种选择性、高亲和力的5-羟
PRT4165
(Catalog# : 1791515, Cas# :
31083-55-3
)
PRT4165是一个核心蛋白复合体1的小分子抑制剂,从而抑制泛素蛋白
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive-Oxygen-Species-ROS
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Mitoquinol mesylate (MitoQ)
(Catalog# : 26A042, Cas# :
845959-55-9
)
Mitoquinol mesylate (MitoQ) 是一种线粒体靶向抗氧化剂,具体而言,它
SPG-601 ( VSN-16R )
(Catalog# : 24042, Cas# :
1246960-09-7
)
SPG-601(原名VSN-16R)是一种口服给药、同类首创的小分子药物,是
LY3039478 ( Crenigacestat )
(Catalog# : 17021601, Cas# :
1421438-81-4
)
LY3039478 ( Crenigacestat ) 是一种选择性 NOTCH1 抑制剂,通过阻断 VEGFA/
PF-9366
(Catalog# : 184107, Cas# :
72882-78-1
)
PF-9366是一种新型的人蛋氨酸腺苷转移酶2A (Mat2A),肝外同种型。
MAT2A-IN-22
(Catalog# : 26A021, Cas# :
2925330-18-1
)
MAT2A-IN-22 (Compound 29-1) 是一种可透过血脑屏障的和口服有效的 MAT2A
Pantothenate kinase-IN-3
(Catalog# : 26A041)
泛酸激酶-IN-3(亦称化合物21,https://doi.org/10.1021/acs.jmedchem.5c03452)
Claziprotamidum ( Claziprotamide ; BBP-671 )
(Catalog# : 26A040, Cas# :
2361124-03-8
)
Claziprotamidum(Claziprotamide;BBP-671)是一种强效、口服有效且能透过
PZ-3022
(Catalog# : 26A039, Cas# :
2170608-85-0
)
PZ-3022是一种别构型的PanK激活剂,能够抵消C3-CoA的抑制作用。
PZ-2891
(Catalog# : 193282, Cas# :
2170608-82-7
)
PZ-2891是一种强效的、选择性的、口服活性泛酸激酶(PANK)调制剂,
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,