武汉永璨生物科技有限公司
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
Nuclear Receptor
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
Nuclear Receptor
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
搜索
首页
网站地图
产品名字索引 P
按首字母搜索
A
B
C
D
E
F
G
H
I
J
K
L
M
N
O
P
Q
R
S
T
U
V
W
X
Y
Z
1
2
3
4
5
6
7
8
9
«
1
2
3
4
5
6
7
8
9
10
»
产品名字索引 P
PTI-428(PTI428)
(Catalog# : 31619, Cas# :
1953130-87-4
)
PTI-428是一种研究性CFTR放大器,开发用于治疗CFTR基因中发生F508del
PF-05085727
(Catalog# : 1932011, Cas# :
1415637-72-7
)
PF-05085727是一种强效、选择性和脑穿透性磷酸二酯酶2A抑制剂。
Petesicatib
(Catalog# : 193206, Cas# :
1252637-35-6
)
Petesicatib是一种组织蛋白酶抑制剂的候选药物。
Pyridone 6
(Catalog# : 193204, Cas# :
457081-03-7
)
吡啶酮6,也被称为CMP 6或JAK抑制剂I,是一种pan-janus-激活的激酶抑
Pretomanid
(Catalog# : 193110, Cas# :
187235-37-6
)
Pretomanid,也被称为PA-824,一种生物还原药物。PA-824具有较强的体
PF-4136309
(Catalog# : 192282, Cas# :
1341224-83-6
)
PF-4136309,又称INCB8761,是一种口服的人趋化因子受体2 (CCR2)拮抗剂
帕利伐米
(Catalog# : 192272, Cas# :
31645-39-3
)
帕利伐米,又名ZIO201,是一种具有潜在抗肿瘤活性的合成芥菜化合
PF-06873600
(Catalog# : 191145, Cas# :
2185857-97-8
)
PF-06873600是一种口服生物利用的细胞周期蛋白依赖性激酶(CDK)抑制
PF04418948
(Catalog# : 191141, Cas# :
1078166-57-0
)
PF-04418948是一种新型高效选择性前列腺素EP2受体拮抗剂。
PF74
(Catalog# : 1812253, Cas# :
1352879-65-2
)
PF-3450074,又称PF74,是一种针对HIV衣壳蛋白的HIV-1抑制剂。PF74与HI
PT2385
(Catalog# : 1812135, Cas# :
1672665-49-4
)
PT2385是一种口服活性小分子缺氧诱导因子(HIF)-2alpha抑制剂,具有潜
PF 1022A
(Catalog# : 1811232, Cas# :
133413-70-4
)
PF1022A是一种新型的驱虫药,与嗜乳激素样跨膜受体结合,对线虫
普拉曲沙
(Catalog# : 1811221, Cas# :
146464-95-1
)
普拉曲沙是二氢叶酸还原酶(DHFR)的一种叶酸模拟抑制剂,对叶酸还
PF-05231023
(Catalog# : 1811162, Cas# :
1037589-69-7
)
PF-05231023是一种长效FGF21仿生产品。PF-05231023可以减轻非人类灵长类
PA-8
(Catalog# : 1810254, Cas# :
878437-15-1
)
PA-8是PAC1受体的小分子拮抗剂。
Pyronaridine Tetraphosphate
(Catalog# : 1810242, Cas# :
76748-86-2
)
Pyronaridine Tetraphosphate是一种抗疟药,能阻断b -血凝素的形成,抑制
PH-002
(Catalog# : 1810234, Cas# :
1311174-68-1
)
PH-002是一种新型的载脂蛋白(apo) E4分子内区域相互作用的神经细胞
Pemigatinib (INCB054828)
(Catalog# : 1810164, Cas# :
1513857-77-6
)
Pemigatinib是一种酪氨酸激酶抑制剂,也是一种抗肿瘤药物候选药物
Pelitrexol
(Catalog# : 189131, Cas# :
446022-33-9
)
Pelitrexol是GARFT抑制剂,也是具有抗增殖活性的水溶性抗叶酸。
PCI-33380
(Catalog# : 18943, Cas# :
1022899-36-0
)
PCI-33380是基于ibrutinib支架设计的,已被用于细胞和体内研究,证实
Perastine
(Catalog# : 187164, Cas# :
4960-10-5
)
Perastine是一种生物化学药。
PCO371
(Catalog# : 187125, Cas# :
1613373-33-3
)
PCO371是一种有效的、选择性的PTHR1激动剂,用于治疗低甲状旁腺功
PQR530
(Catalog# : 18756, Cas# :
1927857-61-1
)
PQR530是一种高效的日常pan-PI3K/mTORC1/2抑制剂。
Pyrotinib
(Catalog# : 18731, Cas# :
1269662-73-8
)
Pyrotinib,又称SHR -1258,是一种口服生物利用的双激酶抑制剂,是表
PX20606反式消旋体
(Catalog# : 186274, Cas# :
1268244-85-4
)
PX20606, 也称为PX-102, 是一种FXR激动剂。
PF-05180999
(Catalog# : 186153, Cas# :
1394033-54-5
)
PF-05180999是一个强有力的和选择性PDE2a抑制剂(PDE2a的IC50 = 0.001μM,
Pritelivir甲磺酸盐
(Catalog# : 186152, Cas# :
1428333-96-3
)
Pritelivir,又名AIC-316和BAY 57-1293,是一种有效的螺旋酶抑制剂。
Pridopidine
(Catalog# : 18673, Cas# :
346688-38-8
)
Pridopidine也被称为ACR16,是一种多巴胺稳定剂,它可以改善运动表
Pamiparib
(Catalog# : 185233, Cas# :
1446261-44-4
)
Pamiparib是高选择性PARP-1/2抑制剂。临床试验中表现出良好的抗肿瘤
PAC 14028
(Catalog# : 185223, Cas# :
1005168-10-4
)
PAC-14028是高效的选择性的瞬时受体电位香草酸亚型1 (TRPV1) 拮抗剂
«
1
2
3
4
5
6
7
8
9
10
»
产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
----
SSTR
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
----
Hemoglobin
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Linafexor (别名: CS-0159)
(Catalog# : 26A089, Cas# :
2765593-43-7
)
Linafexor(同义词:CS-0159)是法尼醇X受体(FXR)的强效非胆汁酸激
Prifetrastat (Synonyms: PF-07248144)
(Catalog# : 26A088, Cas# :
2569008-99-5
)
Prifetrastat (Synonyms: PF-07248144) 是一款首创、选择性、口服活性的
Camonsertib
(Catalog# : 24052, Cas# :
2417489-10-0
)
Camonsertib,也称为RP 3500,是一种新型、强效和选择性的ATR抑制剂,
MRX-2843
(Catalog# : 26A087, Cas# :
1429882-07-4
)
MRX-2843 是一种口服可用的双受体酪氨酸激酶(RTKs)抑制剂,作用
GDC-0134
(Catalog# : 20432, Cas# :
1637394-01-4
)
GDC-0134是一种MAP3K12(DLK)抑制剂。
BI-847325
(Catalog# : 25046, Cas# :
2128698-24-6
)
BI-847325是一种新型的、可口服的、竞争ATP结合位点的Aurora激酶和M
GDD-261
(Catalog# : 26A084, Cas# :
3137699-54-5
)
GDD-261是一种口服活性的磷酸甘油酸脱氢酶变构抑制剂(IC50=61nM)
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
Atebimetinib(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制剂
BH-30643
(Catalog# : 26A047, Cas# :
3062177-59-4
)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制
ERAS-801 ( JGK-068S )
(Catalog# : 20635, Cas# :
2490431-16-6
)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。