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抑制剂/受体激动剂
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订购信息
联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
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Aldehydes
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Amino Acids
Anilines
Boronic Acids
Bromides
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Chiral Compounds
Deuterated
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Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
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订购信息
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联系我们
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产品名字索引 P
盐酸普拉克索
(Catalog# : 1791510, Cas# :
104632-25-9
)
普拉克索是一个GαI-联多巴胺受体D2、D3和D4受体激动剂。它是相对
PF-06281355
(Catalog# : 1791312, Cas# :
1435467-38-1
)
PF-06281355,也称为PF-1355,是一种口服有效的、选择性的,有效的机
Puromycin Aminonucleoside
(Catalog# : 1791310, Cas# :
58-60-6
)
嘌呤霉素,也被称为PAN,NSC3056,在人类肾小球疾病的研究和肾小
P7C3-OMe
(Catalog# : 179116, Cas# :
1235481-43-2
)
P7C3-OMe,也称为(R)- P7C3-OMe,是P3C3-A20和P7C3的模拟。减轻C57BL/6J小
PF-CBP1 游离
(Catalog# : 179113, Cas# :
1962928-21-7
)
PF-CBP1,也称为 PF06670910,是强效、高选择性的CREB结合蛋白布罗莫
PF-CBP1盐酸
(Catalog# : 179112, Cas# :
2070014-93-4
)
PF-CBP1,也称为 PF06670910,是强效、高选择性的CREB结合蛋白布罗莫
PF-06650833
(Catalog# : 17988, Cas# :
1817626-54-2
)
PF-06650833是一种白细胞介素-1受体相关激酶4 (IRAK4)抑制剂。IRAK4位于
Prexasertib 甲磺酸
(Catalog# : 17986, Cas# :
1234015-55-4
)
Prexasertib也称为LY2606368,是一种有效,具有选择性的Chk1/Chk2抑制剂
PF-01247324
(Catalog# : 1781102, Cas# :
875051-72-2
)
PF-01247324一种新的选择性和口服生物利用率的Nav 1.8通道阻滞剂,能
PD166866
(Catalog# : 178814, Cas# :
192705-79-6
)
PD166866有明显的抗增殖作用。
培哚普利
(Catalog# : 2017829, Cas# :
95153-31-4
)
培哚普利是一种有效且长效的血管紧张素转换酶抑制剂,可引起周
PF 04929113
(Catalog# : 2017826, Cas# :
908115-27-5
)
PF-04929113, 也称为SNX-5422,是一种针对人体热休克蛋白90(Hsp90)的合成
帕洛诺司琼
(Catalog# : 2017080119, Cas# :
135729-61-2
)
帕洛诺司琼是一种5-HT3拮抗剂,用于预防和治疗化疗引起的恶心和
霜霉威盐酸盐
(Catalog# : 2017080115, Cas# :
25606-41-1
)
霜霉威盐酸盐是一种高效、广谱、氨基甲酸酯类杀菌剂。
PF-06747775
(Catalog# : 175161, Cas# :
1776112-90-3
)
PF-06747775(PF06747775;CAS 1776112-90- 3)是表皮生长因子受体(EGFR)突变体T7
PF-04995274
(Catalog# : 17031017, Cas# :
1331782-27-4
)
PF-04995274是一个5 - HT4受体部分激动剂。它被认为是作为一种治疗阿
吡西卡尼盐酸盐
(Catalog# : 17031016, Cas# :
88069-49-2
)
吡西卡尼,也叫SUN 1165,是日本临床上用来治疗心律失常的一种药
PNU-74654
(Catalog# : 17031011, Cas# :
113906-27-7
)
PNU-75654扰乱通过抑制Wnt信号通路β-catenin与Tcf4之间的交互(KD50 = 450
垂体腺苷酸环酶激活多肽
(Catalog# : 17031005, Cas# :
127317-03-7
)
垂体腺苷酸环酶激活多肽(PACAP 1- 27)是一种有效的PACAP受体拮抗剂。
Ponesimod
(Catalog# : 17030918, Cas# :
854107-55-4
)
Ponesimod,也被称为ACT - 128800,是一个强有力的,而且是积极的选择
匹莫苯丹
(Catalog# : 17030916, Cas# :
74150-27-9
)
匹莫苯丹是一种兽医药物。Pimobendan是一种钙敏化剂,是一种磷酸
PFK-158
(Catalog# : 17030915, Cas# :
1462249-75-7
)
PFK-158, 也称为ACT-PFK-158,是一种6 -磷酸果糖- 2激酶/果糖- 2,6 -双磷酸
PH-797804
(Catalog# : 17030914, Cas# :
586379-66-0
)
PH-797804是一种有效的p38 mit原活化蛋白(MAP)激酶的选择性抑制剂。P
PIK-75
(Catalog# : 17030913, Cas# :
372196-67-3
)
PIK-75是作为一个3 -激酶药物发现计划的一部分而发展的。PIK75在10
PF-05089771
(Catalog# : 17030912, Cas# :
1235403-62-9
)
PF-05089771是一种选择性的Nav1.7抑制剂(IC50 = 1nm),它与域四的电压传
PF-CBP1
(Catalog# : 17030716)
PF-CBP1也被称为PF- 06670910,是一种强力的、高度选择性的抑制CREB结
Piperoxan HCl
(Catalog# : 17030708, Cas# :
135-87-5
)
Piperoxan,也叫benodaine,是一种药物,它是最先被发现的抗组胺剂。
PFI-1
(Catalog# : 17030704, Cas# :
1403764-72-6
)
PFI-1是一种有效、选择性高的蛋白质相互作用抑制剂,它的目标为
吡美诺
(Catalog# : 17030702, Cas# :
68252-19-7
)
吡美诺是一种抗心律失常的药物。在豚鼠心脏中,吡美诺抑制了毒
帕纳替尼盐酸盐
(Catalog# : 17030607, Cas# :
1114544-31-8
)
帕纳替尼,又名AP24534,是一种口服药物,用于治疗慢性粒细胞白
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
ECI830
(Catalog# : 26A031, Cas# :
3054692-62-2
)
ECI830是一种实验性的CDK2抑制剂。
GNE-317
(Catalog# : 52282, Cas# :
1394076-92-6
)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
DPTX-3186
(Catalog# : 26A010, Cas# :
3118994-80-9
)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108, Cas# :
435327-40-5
)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
Iclepertin (BI-425809)
(Catalog# : 24084, Cas# :
1421936-85-7
)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
Kartogenin ( KGN )
(Catalog# : 52215, Cas# :
4727-31-5
)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602, Cas# :
218791-21-0
)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
Apecotrep (BI 764198)
(Catalog# : 26A048, Cas# :
2311863-36-0
)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
BH-30643
(Catalog# : 26A047, Cas# :
3062177-59-4
)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制