武汉永璨生物科技有限公司
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
搜索
首页
网站地图
产品名字索引 P
按首字母搜索
A
B
C
D
E
F
G
H
I
J
K
L
M
N
O
P
Q
R
S
T
U
V
W
X
Y
Z
1
2
3
4
5
6
7
8
9
«
1
2
3
4
5
6
7
8
9
10
»
产品名字索引 P
盐酸普拉克索
(Catalog# : 1791510, Cas# :
104632-25-9
)
普拉克索是一个GαI-联多巴胺受体D2、D3和D4受体激动剂。它是相对
PF-06281355
(Catalog# : 1791312, Cas# :
1435467-38-1
)
PF-06281355,也称为PF-1355,是一种口服有效的、选择性的,有效的机
Puromycin Aminonucleoside
(Catalog# : 1791310, Cas# :
58-60-6
)
嘌呤霉素,也被称为PAN,NSC3056,在人类肾小球疾病的研究和肾小
P7C3-OMe
(Catalog# : 179116, Cas# :
1235481-43-2
)
P7C3-OMe,也称为(R)- P7C3-OMe,是P3C3-A20和P7C3的模拟。减轻C57BL/6J小
PF-CBP1 游离
(Catalog# : 179113, Cas# :
1962928-21-7
)
PF-CBP1,也称为 PF06670910,是强效、高选择性的CREB结合蛋白布罗莫
PF-CBP1盐酸
(Catalog# : 179112, Cas# :
2070014-93-4
)
PF-CBP1,也称为 PF06670910,是强效、高选择性的CREB结合蛋白布罗莫
PF-06650833
(Catalog# : 17988, Cas# :
1817626-54-2
)
PF-06650833是一种白细胞介素-1受体相关激酶4 (IRAK4)抑制剂。IRAK4位于
Prexasertib 甲磺酸
(Catalog# : 17986, Cas# :
1234015-55-4
)
Prexasertib也称为LY2606368,是一种有效,具有选择性的Chk1/Chk2抑制剂
PF-01247324
(Catalog# : 1781102, Cas# :
875051-72-2
)
PF-01247324一种新的选择性和口服生物利用率的Nav 1.8通道阻滞剂,能
PD166866
(Catalog# : 178814, Cas# :
192705-79-6
)
PD166866有明显的抗增殖作用。
培哚普利
(Catalog# : 2017829, Cas# :
95153-31-4
)
培哚普利是一种有效且长效的血管紧张素转换酶抑制剂,可引起周
PF 04929113
(Catalog# : 2017826, Cas# :
908115-27-5
)
PF-04929113, 也称为SNX-5422,是一种针对人体热休克蛋白90(Hsp90)的合成
帕洛诺司琼
(Catalog# : 2017080119, Cas# :
135729-61-2
)
帕洛诺司琼是一种5-HT3拮抗剂,用于预防和治疗化疗引起的恶心和
霜霉威盐酸盐
(Catalog# : 2017080115, Cas# :
25606-41-1
)
霜霉威盐酸盐是一种高效、广谱、氨基甲酸酯类杀菌剂。
PF-06747775
(Catalog# : 175161, Cas# :
1776112-90-3
)
PF-06747775(PF06747775;CAS 1776112-90- 3)是表皮生长因子受体(EGFR)突变体T7
PF-04995274
(Catalog# : 17031017, Cas# :
1331782-27-4
)
PF-04995274是一个5 - HT4受体部分激动剂。它被认为是作为一种治疗阿
吡西卡尼盐酸盐
(Catalog# : 17031016, Cas# :
88069-49-2
)
吡西卡尼,也叫SUN 1165,是日本临床上用来治疗心律失常的一种药
PNU-74654
(Catalog# : 17031011, Cas# :
113906-27-7
)
PNU-75654扰乱通过抑制Wnt信号通路β-catenin与Tcf4之间的交互(KD50 = 450
垂体腺苷酸环酶激活多肽
(Catalog# : 17031005, Cas# :
127317-03-7
)
垂体腺苷酸环酶激活多肽(PACAP 1- 27)是一种有效的PACAP受体拮抗剂。
Ponesimod
(Catalog# : 17030918, Cas# :
854107-55-4
)
Ponesimod,也被称为ACT - 128800,是一个强有力的,而且是积极的选择
匹莫苯丹
(Catalog# : 17030916, Cas# :
74150-27-9
)
匹莫苯丹是一种兽医药物。Pimobendan是一种钙敏化剂,是一种磷酸
PFK-158
(Catalog# : 17030915, Cas# :
1462249-75-7
)
PFK-158, 也称为ACT-PFK-158,是一种6 -磷酸果糖- 2激酶/果糖- 2,6 -双磷酸
PH-797804
(Catalog# : 17030914, Cas# :
586379-66-0
)
PH-797804是一种有效的p38 mit原活化蛋白(MAP)激酶的选择性抑制剂。P
PIK-75
(Catalog# : 17030913, Cas# :
372196-67-3
)
PIK-75是作为一个3 -激酶药物发现计划的一部分而发展的。PIK75在10
PF-05089771
(Catalog# : 17030912, Cas# :
1235403-62-9
)
PF-05089771是一种选择性的Nav1.7抑制剂(IC50 = 1nm),它与域四的电压传
PF-CBP1
(Catalog# : 17030716)
PF-CBP1也被称为PF- 06670910,是一种强力的、高度选择性的抑制CREB结
Piperoxan HCl
(Catalog# : 17030708, Cas# :
135-87-5
)
Piperoxan,也叫benodaine,是一种药物,它是最先被发现的抗组胺剂。
PFI-1
(Catalog# : 17030704, Cas# :
1403764-72-6
)
PFI-1是一种有效、选择性高的蛋白质相互作用抑制剂,它的目标为
吡美诺
(Catalog# : 17030702, Cas# :
68252-19-7
)
吡美诺是一种抗心律失常的药物。在豚鼠心脏中,吡美诺抑制了毒
帕纳替尼盐酸盐
(Catalog# : 17030607, Cas# :
1114544-31-8
)
帕纳替尼,又名AP24534,是一种口服药物,用于治疗慢性粒细胞白
«
1
2
3
4
5
6
7
8
9
10
»
产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive-Oxygen-Species-ROS
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Mitoquinol mesylate (MitoQ)
(Catalog# : 26A042, Cas# :
845959-55-9
)
Mitoquinol mesylate (MitoQ) 是一种线粒体靶向抗氧化剂,具体而言,它
SPG-601 ( VSN-16R )
(Catalog# : 24042, Cas# :
1246960-09-7
)
SPG-601(原名VSN-16R)是一种口服给药、同类首创的小分子药物,是
LY3039478 ( Crenigacestat )
(Catalog# : 17021601, Cas# :
1421438-81-4
)
LY3039478 ( Crenigacestat ) 是一种选择性 NOTCH1 抑制剂,通过阻断 VEGFA/
PF-9366
(Catalog# : 184107, Cas# :
72882-78-1
)
PF-9366是一种新型的人蛋氨酸腺苷转移酶2A (Mat2A),肝外同种型。
MAT2A-IN-22
(Catalog# : 26A021, Cas# :
2925330-18-1
)
MAT2A-IN-22 (Compound 29-1) 是一种可透过血脑屏障的和口服有效的 MAT2A
Pantothenate kinase-IN-3
(Catalog# : 26A041)
泛酸激酶-IN-3(亦称化合物21,https://doi.org/10.1021/acs.jmedchem.5c03452)
Claziprotamidum ( Claziprotamide ; BBP-671 )
(Catalog# : 26A040, Cas# :
2361124-03-8
)
Claziprotamidum(Claziprotamide;BBP-671)是一种强效、口服有效且能透过
PZ-3022
(Catalog# : 26A039, Cas# :
2170608-85-0
)
PZ-3022是一种别构型的PanK激活剂,能够抵消C3-CoA的抑制作用。
PZ-2891
(Catalog# : 193282, Cas# :
2170608-82-7
)
PZ-2891是一种强效的、选择性的、口服活性泛酸激酶(PANK)调制剂,
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,