武汉永璨生物科技有限公司
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抑制剂/受体激动剂
Angiogenesis
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
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技术服务
定制合成
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订购信息
联系我们
公司简介
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产品名字索引 G
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产品名字索引 G
GSK2193874
(Catalog# : 178914, Cas# :
1336960-13-4
)
GSK2193874被认定为一种选择性的、口服的TRPV4阻断剂。
GW4869
(Catalog# : 178912, Cas# :
6823-69-4
)
GW4869(二氯化物水合物)是一种可渗透的、选择性的N- Smase(中性鞘磷
GSK2982772
(Catalog# : 178911, Cas# :
1622848-92-3
)
GSK2982772是一种ATP竞争性的受体- 1(激酶)抑制剂,IC50值为1 nM。它有
GSK180736A (GSK180736)
(Catalog# : 178901, Cas# :
817194-38-0
)
GSK180736A是一种有效的、具有选择性的IC50 0.77 M25的GRK2抑制剂,比其
GSK2269557
(Catalog# : 2017883, Cas# :
1254036-77-5
)
GSK2269557,也称为GSK-2269557, 是一种有效且选择性的PI3K抑制剂.。
GDC-0326
(Catalog# : 2017881, Cas# :
1282514-88-8
)
GDC-0326是一种有效且选择性的磷酸肌醇的α-同种型3-激酶抑制剂(PI
GSK-1521498
(Catalog# : 20178215, Cas# :
1007573-18-3
)
GSK-1521498是一种新型阿片受体拮抗剂。它已经被证明可以减弱奖励
GSK321
(Catalog# : 2017821, Cas# :
1816331-63-1
)
GSK321是一种有效的、选择性的IDH1突变抑制剂。GSK321对HT- 1080细胞内
GNE-272
(Catalog# : 20178121, Cas# :
1936428-93-1
)
GNE-272对CBP / EP300的溴域具有很强的选择性(CBP IC50 = 0.02 μM, EP300 IC5
胍氯酚
(Catalog# : 17030702, Cas# :
5001-32-1
)
胍氯酚是一种抗高血压的药物。
GRA Ex-25
(Catalog# : 17030701, Cas# :
307983-31-9
)
GRA Ex-25是胰高血糖素受体的抑制剂。
GTS-21
(Catalog# : 16123016, Cas# :
156223-05-1
)
GTS-21, also known as DMBX-A, is a derivative of the natural product anabaseine that
GSK6853 (GSK-6853)
(Catalog# : 16123015, Cas# :
1910124-24-1
)
GSK6853 is a potent (300 pM), soluble, cell active (20 nM), and highly selective inhi
GSK583
(Catalog# : 16123014, Cas# :
1346547-00-9
)
GSK583 is a Highly Potent and Selective Inhibitor of RIP2 Kinase (RIP2K bing IC50=5 n
GSK369796 Dihydrochloride
(Catalog# : 16123013, Cas# :
1010411-21-8
)
GSK369796, also known as N-tert-butylisoquine, is an anti-malaria drug candidate. GSK
GSK2801
(Catalog# : 16123012, Cas# :
1619994-68-1
)
GSK2801 is a A Selective Chemical Probe for BAZ2B/A bromodomains. BAZ2A/B belong to a
GSK-2256098
(Catalog# : 16123011, Cas# :
1224887-10-8
)
GSK2256098, also known as GTPL7939, is a focal adhesion kinase-1 (FAK) inhibitor with
GSK137647A
(Catalog# : 16123010, Cas# :
349085-82-1
)
GSK137647A is an agonist of the free fatty acid receptor 4 (FFA4/GPR120) with pEC50s
GSK0660
(Catalog# : 16123009, Cas# :
1014691-61-2
)
GSK0660 is a selective PPAR antagonist. GSK0660 differentially regulated 273 transcri
Go6983
(Catalog# : 16123008, Cas# :
133053-19-7
)
GO6983 is a potent protein kinase C (PKC) inhibitor. GO6893 displays cardioprotective
GNE-617
(Catalog# : 16123007, Cas# :
1362154-70-8
)
GNE-617 is a potent nicotinamide phosphoribosyltransferase (NAMPT) inhibitor with IC5
GlyH-101
(Catalog# : 16123006, Cas# :
328541-79-3
)
GlyH-101 is a CFTR inhibitor (cystic fibrosis transmembrane conductance regulator). G
GLPG-1690(ziritaxestat)
(Catalog# : 16123005, Cas# :
1628260-79-6
)
GLPG1690 is a selective autotaxin inhibitor discovered by Galapagos, with potential a
GDC-0853
(Catalog# : 16123004, Cas# :
1434048-34-6
)
GDC-0853 is orally available inhibitor of Bruton's tyrosine kinase (BTK) with potenti
GABOB (beta-hydroxy-GABA)
(Catalog# : 16122815, Cas# :
7013-05-0
)
GABOB, also known as -Amino--hydroxybutyric acid, -hydroxy--aminobutyric acid, -hydro
Gabexate mesylate
(Catalog# : 16122814, Cas# :
56974-61-9
)
Gabexate is a serine protease inhibitor which is used therapeutically (as gabexate me
Glasdegib (PF-04449913)
(Catalog# : 16122787, Cas# :
1095173-27-5
)
Glasdegib (PF-04449913) is a potent, and orally bioavailable Smoothened (Smo) inhibit
Go6976
(Catalog# : 16122723, Cas# :
136194-77-9
)
Go6976 is a potent PKC inhibitor with IC50 of 7.9 nM, 2.3 nM, and 6.2 nM for PKC (Rat
GSK2292767
(Catalog# : 16122702, Cas# :
1254036-66-2
)
GSK2292767 is a potent and selective PI3K inhibitor.GSK2292767 is highly selective fo
GSK2981278
(Catalog# : 6111521, Cas# :
1474110-21-8
)
ROR modulator 1 is a retinoid-related orphan receptor gamma (RORy) modulator, extract
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
NSD1 抑制剂 BT5
(Catalog# : 25207, Cas# :
2351225-46-0
)
BT5可有效抑制NSD1,与细胞中的SET结构域结合,并降低H3K36me2水平。
MA242 TFA
(Catalog# : 25206, Cas# :
1049704-18-8
)
MA242是一种MDM2和NFAT1双重抑制剂,可诱导MDM2自泛素化及降解,并抑
Dabogratinib ( TYRA-300 )
(Catalog# : 24073, Cas# :
2800223-30-5
)
Dabogratinib ( TYRA-300 )是一种口服选择性成纤维细胞生长因子受体3(
AF710B
(Catalog# : 25205, Cas# :
N/A
)
AF710B 是一种高效、选择性变构 M1 毒蕈碱和 σ1 受体激动剂。 AF710
MAT2A inhibitor 5
(Catalog# : 25204, Cas# :
2957874-18-7
)
MAT2A抑制剂5具有抑制MAT2A的高效力和对MTAP缺失的癌症细胞系的显著
(Rac)-AF710B
(Catalog# : 24083, Cas# :
1235733-73-9
)
AF-710B 是 σ 和 M1 毒蕈碱受体的激动剂;AF710B 是 AF710 的对映体。
Flurpiridaz-nonradiolabeled
(Catalog# : 25203, Cas# :
863888-33-9
)
Flurpiridaz是一种有前景的新型心脏PET成像示踪剂,是通过用氟-18放
Flurpiridaz-Precursor
(Catalog# : 25202, Cas# :
863888-32-8
)
现货
KL1333
(Catalog# : 25201, Cas# :
1800405-30-4
)
KL1333是一种口服的小有机分子,与NAD(P)H:醌氧化还原酶1(NQO1)
Palupiprant ( E7046 )
(Catalog# : 24055, Cas# :
1369489-71-3
)
E7046 is a potent and selective antagonist of the type 4 prostaglandin E2 (PGE2) rece