武汉永璨生物科技有限公司
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抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
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Cytoskeleton
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MAPK
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Metabolism
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分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
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Deuterated
Fluorides
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Indoles and Oxindoles
Iodos
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Peg Linkers
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Pyrimidines
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
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产品名字索引 G
GCN2iB
(Catalog# : 2071802, Cas# :
2183470-12-2
)
GCN2iB is an ATP-competitive GCN2 inhibitory compound with a better pharmacokinetic p
GRL0617
(Catalog# : 2071625, Cas# :
1093070-16-6
)
GRL0617 is a potent, selective and competitive noncovalent inhibitor of SARS PLPro. G
GS-441524
(Catalog# : 2071546, Cas# :
1191237-69-0
)
GS-441524 is a potent inhibitor of feline infectious peritonitis (FIP) virus with an
GSK3145095
(Catalog# : 2071533, Cas# :
1622849-43-7
)
GSK3145095 is a potent and orally active RIPK1 inhibitor (IC50 = 5 nM) with potential
GSK2894631A
(Catalog# : 2071528, Cas# :
2101626-26-8
)
GSK2894631A is a hematopoietic PGD synthase (HPGDS) inhibitor.
GSK8612
(Catalog# : 2071527, Cas# :
2361659-62-1
)
GSK8612 is a potent and highly selective TBK1 inhibitor. GSK8612 inhibited recombinan
GSK547
(Catalog# : 2071522)
GSK547 is a highly selective and potent inhibitor of RIP1 kinase that targets RIP1 in
GSK1016790A
(Catalog# : 2071511, Cas# :
942206-85-1
)
GSK1016790A, also known as GSK101, is a TRPV4 agonist that elicits calcium influx in
GNE-131
(Catalog# : 2071509, Cas# :
1629063-81-5
)
GNE-131 is a Potent and Selective hNaV1.7 Inhibitor (Na V1.7 IC50 = 3 nM) for the Tre
GW284543
(Catalog# : 2061310, Cas# :
790186-68-4
)
GW284543, also known as UNC10225170;, is a potent and selective MEK5 inhibitor with t
G-1
(Catalog# : 206103, Cas# :
881639-98-1
)
G-1 is a selective agonist for GPER. It acts by blocking tubulin polymerization.
Glumetinib
(Catalog# : 203401, Cas# :
1642581-63-2
)
Glumetinib, also known as SCC244, is a novel, potent and highly selective inhibitor o
GNE-2861
(Catalog# : 111892, Cas# :
1394121-05-1
)
GNE-2861 is a potent and exquisitely kinase-selective Group II PAK inhibitor (PAK4 Ki
GSK-199
(Catalog# : 193293, Cas# :
1549811-53-1
)
GSK199是一种选择性的PAD4抑制剂,在不含钙的情况下,其半峰抑制
GS-626510
(Catalog# : 193221, Cas# :
1637770-13-8
)
GS-626510是一种有效的BET家族溴域抑制剂。它的作用是针对BRD2/3/4和
GSK2837808A
(Catalog# : 193194, Cas# :
1445879-21-9
)
GSK2837808A是一种高效、选择性的乳酸脱氢酶A(LDHA)抑制剂(LDHA和LDHB的
GSK-963
(Catalog# : 193185, Cas# :
2049868-46-2
)
GSK-963,也被称为GSK'963或GSK963,是一种有效的和选择性的RIP1激
GNE-9605
(Catalog# : 192284, Cas# :
1536200-31-3
)
GNE-9605是一种高效、选择性强、脑内渗透的氨基吡唑亮氨酸富集重
GSK3004774
(Catalog# : 192281, Cas# :
2138814-32-9
)
GSK3004774是一种有效的、不可吸收的CaSR激动剂,人、小鼠和大鼠Ca
GW-3965盐酸盐
(Catalog# : 192251, Cas# :
405911-17-3
)
GW-3965是一种肝脏X受体激动剂。GW3965抑制小鼠肥大细胞产生促炎细
GSK2334470
(Catalog# : 192224, Cas# :
1227911-45-6
)
GSK2334470是一种有效的3-磷酸肌苷依赖性蛋白激酶(PDK1)抑制剂(IC50 ~
GSK269962盐酸盐
(Catalog# : 192201, Cas# :
2095432-71-4
)
GSK269962是一种选择性ROCK抑制剂,对ROCK-I和ROCK- II的IC50值分别为1.6
GW-803430
(Catalog# : 192194, Cas# :
515141-51-2
)
GW-803430是一种强效、口服活性和选择性黑色素聚集激素受体1 (MCH1
GNE-477
(Catalog# : 192181, Cas# :
1032754-81-6
)
GNE-477是一种有效的双PI3K/mTOR抑制剂。
GSKJ1
(Catalog# : 191255, Cas# :
1373422-53-7
)
GSKJ1是一种具有选择性和有效的组蛋白脱甲基酶抑制剂(GSK-J1)有重
GSK2643943A
(Catalog# : 191144, Cas# :
//
)
GSK2643943A是一种有效的USP20抑制剂,IC50值为160 nM。
GSK-2807
(Catalog# : 19185, Cas# :
2245255-65-4
)
GSK-2807是一种有效且具有选择性的SMYD3的SAM-竞争性抑制剂。
GNE-6640
(Catalog# : 1812291, Cas# :
2009273-67-8
)
GNE-6640是一种新型选择性USP7抑制剂,可诱导肿瘤细胞死亡。GNE-664
GSK1940029
(Catalog# : 1812102, Cas# :
1150701-66-8
)
GSK1940029,又称SCD抑制剂1,是一种SCD抑制剂。GSK1940029能够潜在的局
GSK2814338
(Catalog# : 181241, Cas# :
1420367-28-7
)
GSK2814338,也称为Lp-PLA2 -IN-1,是一种Lp-PLA2抑制剂。
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AD-8007
(Catalog# : 26A018, Cas# :
1497439-74-3
)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
ZY-444
(Catalog# : 26A020, Cas# :
1802650-31-2
)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
AD-5584
(Catalog# : 26A019, Cas# :
2306525-79-9
)
AD-5584是一种新型脑渗透性ACSS2抑制剂。
IDB-003
(Catalog# : 26A017, Cas# :
3079716-11-0
)
IDB-003在体内抑制MDA-MB-231肿瘤生长。
Vafidemstat
(Catalog# : 18891, Cas# :
1357362-02-7
)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
LLL12
(Catalog# : 25075, Cas# :
1260247-42-4
)
LLL12是一种强效的STAT3抑制剂。LLL12在小鼠异种移植物模型中显示出
ECC-5004
(Catalog# : 26A015, Cas# :
2758659-09-3
)
ECC5004是一款每日一次、低剂量、小分子GLP-1受体激动剂。
SILA-123
(Catalog# : 26A014, Cas# :
2911585-37-8
)
SILA-123是一种II型FLT3抑制剂,对FLT3-WT(IC50=2.1 nM)和FLT3-ITD(IC50=1
Encaleret sulfate
(Catalog# : 26A013, Cas# :
1214922-52-7
)
Encaleret是一种正在研究的钙敏感受体的小分子拮抗剂,用于钙稳态
Iadademstat ( ORY-1001 ) hydrochloride
(Catalog# : 26A011, Cas# :
1431303-72-8
)
Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶