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Name Index A

• APY29 (Catalog# : 011108, Cas# : 1216665-49-4)APY29 is an allosteric modulator of IRE1; inhibits IRE1 autophosphorylation (IC50 = 2
• AMG-47a (Catalog# : 011107, Cas# : 882663-88-9)AMG-47a is a potent inhibitor of Lck and T cell proliferation.
• ARQ-736 (Catalog# : 011104, Cas# : 1228237-57-7)ARQ 736 is a potent and selective BRAF inhibitor.
• AZD4547 (Catalog# : 010820, Cas# : 1035270-39-3)AZD4547 is a novel selective FGFR inhibitor targeting FGFR1/2/3 with IC50 of 0.2 nM/2
• AZD-1480 (Catalog# : 010816, Cas# : 935666-88-9)AZD1480 is a novel ATP-competitive JAK2 inhibitor with IC50 of 0.26 nM, selectivity a
• AZD8330 (Catalog# : 010809, Cas# : 869357-68-6)AZD8330 is a novel, selective, non-ATP competitive MEK 1/2 inhibitor with IC50 of 7 n
• AS703026 (Catalog# : 010808, Cas# : 1236699-92-5)AS703026 is an orally bioavailable small-molecule inhibitor of MEK1 and MEK2 (MEK1/2)
• AZ505 (Catalog# : 010803, Cas# : 1035227-43-0)AZ505 is a potent and highly selective inhibitor of the oncogenic protein SMYD2(IC50=
• AG-L-59687 (Catalog# : 010428, Cas# : 793035-88-8)Coming soon!
• AG1024 (Catalog# : 010422, Cas# : 65678-07-1)AG-1024 inhibits IGF-1R autophosphorylation with IC50 of 7 M, less potent to IR with
• Almotriptan (Catalog# : 010418, Cas# : 154323-57-6)Almotriptan is a 5-HT1B/1D-receptor agonist used to treat migraine.
• AM630 (Catalog# : 010410, Cas# : 164178-33-0)AM630 is a selectivity CB2 antagonist with Ki of 31.2 nM; > 150 fold selectivity o
• AZD-8055 (Catalog# : 123019, Cas# : 1009298-09-2)AZD-8055 is an inhibitor of the mammalian target of rapamycin (mTOR) with potential a
• Amuvatinib (Catalog# : 123016, Cas# : 850879-09-3)Amuvatinib is a potent and multi-targeted inhibitor of c-Kit, PDGFR and Flt3 with IC5
• AR-42 (Catalog# : 123009, Cas# : 935881-37-1)AR-42 is a novel, oral cancer therapy currently in early clinical development.
• A-966492 (Catalog# : 123006, Cas# : 934162-61-5)A-966492 is a novel and potent inhibitor of PARP1 and PARP2 with Ki of 1 nM and 1.5 n
• AMG 487 (Catalog# : 122942, Cas# : 473719-41-4)AMG 487 is a small molecule antagonist of the chemokine receptor CXCR3.
• Atosiban acetate (Catalog# : 122931, Cas# : 90779-69-4)Atosiban is a nonapeptide, desamino-oxytocin analogue, and a competitive vasopressin/
• AST-1306 (Catalog# : 122926, Cas# : 897383-62-9)AST-1306 is a novel irreversible inhibitor of EGFR and ErbB2 with IC50 of 0.5 nM and
• AZD8186 (Catalog# : 122925, Cas# : 1627494-13-6)AZD8186 is an isoform-specific small-molecule PI3K inhibitor, potently inhibits PI3K
• AG-120 (Catalog# : 122906, Cas# : 1448346-63-1)AG-120 is an orally available inhibitor of isocitrate dehydrogenase type 1 (IDH1), wi
• AZD-5423 (Catalog# : 122902, Cas# : 1034148-04-3)Coming soon!
• A 83-01 (Catalog# : 122843, Cas# : 909910-43-6)A 83-01 is a selective inhibitor of TGF- type I receptor ALK5 kinase, type I activin/
• AM251 (Catalog# : 122842, Cas# : 183232-66-8)AM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 3
• AZD2858 (Catalog# : 122838, Cas# : 486424-20-8)AZD2858 is a selective GSK-3 inhibitor with an IC50 of 68 nM, inhibits tau phosphoryl
• Adjudin (Catalog# : 122824, Cas# : 252025-52-8)Adjudin is a drug which is under development as a potential non-hormonal male contrac
• AdipoRon (Catalog# : 122822, Cas# : 924416-43-3)AdipoRon is a novel small-molecule AdipoR agonist; binds to both AdipoR1(Kd= 1.8 uM)
• Anamorelin (Catalog# : 122407, Cas# : 249921-19-5)Anamorelin is a synthetic orally active ghrelin receptor agonist which is under devel
• Atorvastatin sodium (Catalog# : 122303, Cas# : 134523-01-6)Atorvastatin has the potential to ameliorate arsenic-induced vascular dysfunction and
• Amrubicin (Catalog# : 122211, Cas# : 110267-81-7)Amrubicin is a novel anthracycline derivative for treatment of bladder carcinoma.