Apecotrep (BI 764198) is a potential first-in-class, oral, selective TRPC6 inhibitor.
For research use only. We do not sell to patients.
| Name | Apecotrep (BI 764198) |
|---|---|
| Iupac Chemical Name | (4-(6-aminopyridazin-3-yl)piperidin-1-yl)(5-(4-fluorophenoxy)-4-methoxypyridin-2-yl)methanone |
| Synonyms | Apecotrep; BI 764198; BI764198; BI-764198; TRPC6-IN-3 |
| Molecular Formula | C22H22FN5O3 |
| Molecular Weight | 423.4 |
| Smile | O=C(N1CCC(C2=NN=C(N)C=C2)CC1)C3=NC=C(OC4=CC=C(F)C=C4)C(OC)=C3 |
| InChiKey | JUALOUHZJJERQT-UHFFFAOYSA-N |
| InChi | InChI=1S/C22H22FN5O3/c1-30-19-12-18(25-13-20(19)31-16-4-2-15(23)3-5-16)22(29)28-10-8-14(9-11-28)17-6-7-21(24)27-26-17/h2-7,12-14H,8-11H2,1H3,(H2,24,27) |
| CAS Number | 2311863-36-0 |
| Related CAS | 2311863-36-0 |
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Solid powder |
|---|---|
| Purity | ≧98.0% |
| Storage | Dry, dark and at 0 - 4℃ for short term (days to weeks) or -20℃ for long term (months to years). |
| Solubility | Soluble in DMSO (DMSO : ≥ 100 mg/mL) |
| Handling | Refer to MSDS |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| HS Code | 2934200090 |
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |