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抑制剂/受体激动剂
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
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Pyridines
Pyrimidines
Quinolines
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产品名字索引 M
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产品名字索引 M
ML-265
(Catalog# : 17030804, Cas# :
1221186-53-3
)
ML265是一个强有力的PKM2活化剂诱导四聚体,降低肿瘤的形成和大小
MN-64
(Catalog# : 17030717, Cas# :
92831-11-3
)
MN-64 是一种有效的、选择性的Tankyrase 1和2抑制剂(IC50值分别为6和
ML241
(Catalog# : 17030714, Cas# :
1346528-06-0
)
ML241是一种p97 ATPase有效的选择性抑制剂。ML241抑制p97 ATPase的IC(50)值
ML348
(Catalog# : 17030712, Cas# :
899713-86-1
)
ML348,又称CID 3238952;SID 160654487,是一个可逆的LYPLA1抑制剂,IC50值
MMAF (Monomethyl auristatin F)
(Catalog# : 17030611, Cas# :
745017-94-1
)
一甲基澳瑞他汀 F(MMAF)是一种合成抗肿瘤药物。它是一些实验性抗
Merimepodib
(Catalog# : 17030308, Cas# :
198821-22-6
)
Merimepodib, 也称为VX-497,是有效的口服生物IMPDH抑制剂,它可以抑制
ML-264
(Catalog# : 17030302, Cas# :
1550008-55-3
)
ML-264是一种Krüppel-like因子5(KLF5)抑制剂,能有效抑制结直肠癌的生
MK-8245
(Catalog# : 17030109, Cas# :
1030612-90-8
)
MK-8245是一种有效的、以肝脏为靶点的SCD抑制剂,具有临床前抗糖
MLN-1117
(Catalog# : 17030101, Cas# :
1268454-23-4
)
Serabelisib(又名MLN1117,INK1117,TAK- 117)是一类具有潜在抗肿瘤活性的磷
ML-281
(Catalog# : 17022811, Cas# :
1404437-62-2
)
ML-281是一种有效的选择性STK33抑制剂(IC50 = 14nm)。与其他STK33抑制剂
马拉维若
(Catalog# : 17022804, Cas# :
376348-65-1
)
马拉维若(UK-427857; Selzentry; Celsentri) 是选择性CCR5拮抗剂(IC50 = 6.4 nM
单甲基奥立斯丁
(Catalog# : 17022403, Cas# :
474645-27-7
)
MMAE,又称单甲基奥立斯丁,是一种合成的抗肿瘤药物。
Monastrol
(Catalog# : 17021322, Cas# :
329689-23-8
)
Monastrol是一种细胞可渗透的小分子抑制剂,它对保持半纺锤的分离
MS049
(Catalog# : 17021313, Cas# :
1502816-23-0
)
MS049是PRMT4和PRMT6的一种有效的选择性抑制剂,IC50分别为34 nM和43 n
Miransertib(ARQ 092)
(Catalog# : 17021301, Cas# :
1313883-00-9
)
ARQ 092是一种新型的口服生物可用性和选择性AKT通路抑制剂,在晚
MT-DADMe-ImmA(MTDIA HCl)
(Catalog# : 712101, Cas# :
1399840-35-7
)
MT-DADMe-ImmA(MTDIA盐酸盐)是一种新型的MTAP抑制剂,具有治疗头颈部和
7-Methyl-7H-pyrrolo[2,3-d]pyriMidin-4-aMine
(Catalog# : 17011908, Cas# :
7752-54-7
)
7-Methyl-7H-pyrrolo[2,3-d]pyriMidin-4-aMine
ML-7
(Catalog# : 17011107, Cas# :
110448-33-4
)
ML-7是平滑肌肌球蛋白轻链激酶的抑制剂(MLCK),Ki值为0.3μM。
MX69
(Catalog# : 17011105, Cas# :
1005264-47-0
)
MX69是一种MDM2/XIAP抑制剂, 用于治疗癌症。
MK-571 sodium salt
(Catalog# : 16123055, Cas# :
115104-28-4
)
MK-571 is a selective, orally active CysLT1 receptor antagonist. It blocks the bindin
Mizoribine
(Catalog# : 16123053, Cas# :
50924-49-7
)
Mizoribine,Mizoribine (INN, trade name Bredinin) is an immunosuppressive drug. The co
Mivebresib
(Catalog# : 16123052, Cas# :
1445993-26-9
)
Mivebresib, also known as ABBV-075, is a potent BET inhibitor (bromodomain (BRD)-cont
Mitoxantrone HCl
(Catalog# : 16123051, Cas# :
65271-80-9
)
Mitoxantrone hydrochloride is the hydrochloride salt of an anthracenedione antibiotic
Mirin
(Catalog# : 16123049, Cas# :
1198097-97-0
)
Mirin is a Mre11-Rad50-Nbs1 (MRN)-ATM pathway inhibitor.
Migalastat HCl
(Catalog# : 16123048, Cas# :
75172-81-5
)
Migalastat HCl, also known as AT1001 or GR181413A, is a pharmacological chaperone tha
MI-2 (MALT1 inhibitor)
(Catalog# : 16123047, Cas# :
1047953-91-2
)
MI-2 is a MALT1 inhibitor (IC50 = 5.84 M). MI-2 binds directly to MALT1 and irreversi
MG-101
(Catalog# : 16123046, Cas# :
110044-82-1
)
MG-101, also known as Calpain Inhibitor I and ALLN, is a calpain inhibitor (IC50 = 0.
Mertansine (DM1)
(Catalog# : 16123045, Cas# :
139504-50-0
)
Mertansine refers to the thiol-containing maytansinoid, DM1 (N2-deacetyl-N2-(3-mercap
MC-976
(Catalog# : 16122832, Cas# :
129831-99-8
)
MC-976 is an Vitamin D3 derivative.
Mafodotin
(Catalog# : 16122831, Cas# :
863971-19-1
)
Mafodotin, also known as mc-MMAF and SGD-1269 or Maleimidocaproyl monomethylauristati
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive-Oxygen-Species-ROS
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Mitoquinol mesylate (MitoQ)
(Catalog# : 26A042, Cas# :
845959-55-9
)
Mitoquinol mesylate (MitoQ) 是一种线粒体靶向抗氧化剂,具体而言,它
SPG-601 ( VSN-16R )
(Catalog# : 24042, Cas# :
1246960-09-7
)
SPG-601(原名VSN-16R)是一种口服给药、同类首创的小分子药物,是
LY3039478 ( Crenigacestat )
(Catalog# : 17021601, Cas# :
1421438-81-4
)
LY3039478 ( Crenigacestat ) 是一种选择性 NOTCH1 抑制剂,通过阻断 VEGFA/
PF-9366
(Catalog# : 184107, Cas# :
72882-78-1
)
PF-9366是一种新型的人蛋氨酸腺苷转移酶2A (Mat2A),肝外同种型。
MAT2A-IN-22
(Catalog# : 26A021, Cas# :
2925330-18-1
)
MAT2A-IN-22 (Compound 29-1) 是一种可透过血脑屏障的和口服有效的 MAT2A
Pantothenate kinase-IN-3
(Catalog# : 26A041)
泛酸激酶-IN-3(亦称化合物21,https://doi.org/10.1021/acs.jmedchem.5c03452)
Claziprotamidum ( Claziprotamide ; BBP-671 )
(Catalog# : 26A040, Cas# :
2361124-03-8
)
Claziprotamidum(Claziprotamide;BBP-671)是一种强效、口服有效且能透过
PZ-3022
(Catalog# : 26A039, Cas# :
2170608-85-0
)
PZ-3022是一种别构型的PanK激活剂,能够抵消C3-CoA的抑制作用。
PZ-2891
(Catalog# : 193282, Cas# :
2170608-82-7
)
PZ-2891是一种强效的、选择性的、口服活性泛酸激酶(PANK)调制剂,
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,