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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
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产品名字索引 M
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产品名字索引 M
MDK7229
(Catalog# : 184211, Cas# :
111797-22-9
)
MDK7229, also known as MD2-IN-1 is a MD2 (Myeloid differentiation protein 2) inhibito
MDK6574
(Catalog# : 18421, Cas# :
2102196-57-4
)
MDK6574,也称为FAA1 agonist-1,FAA1受体激动剂。
2-甲基-7-氮杂吲哚
(Catalog# : 183131, Cas# :
23612-48-8
)
2-甲基-7-氮杂吲哚是一种医药中间体。
4-methylsulfonyl-2-(trifluoromethyl)benzaldehyde
(Catalog# : 1712293, Cas# :
1215310-75-0
)
4-methylsulfonyl-2-(trifluoromethyl)benzaldehyde isa building blocks.
MK-8617
(Catalog# : 1710163, Cas# :
1187990-87-9
)
MK-8617是一种缺氧诱导因子(HIF脯氨酰羟化酶1−3 PHD1−3),具有强效
MSC2530818
(Catalog# : 1710135, Cas# :
1883423-59-3
)
MSC2530818是一种强效、选择性,口服生物利用度与抑制剂的IC50 = 2.
MDK19922
(Catalog# : 1791512, Cas# :
132819-92-2
)
MDK19922,也称为NOD-IN-1或化合物4,是一种有效的核苷酸结合寡聚化
游离莫扎伐普坦
(Catalog# : 179154, Cas# :
137975-06-5
)
莫扎伐普坦,又名OPC 31260,是由大冢销售的血管加压素受体拮抗剂
ML-141
(Catalog# : 179152, Cas# :
71203-35-5
)
ML-141,也称为CID2950007,是Cdc42抑制剂(EC50 = 2.1μm)。
MDK30165
(Catalog# : 179138, Cas# :
2060530-16-5
)
MDK30165,也称为K-Ras(G12C)抑制剂6。
单甲基澳瑞他汀 D
(Catalog# : 20179132, Cas# :
203849-91-6
)
MMAD又称为单甲基澳瑞他汀 D,是一种高效的微管蛋白抑制剂。MMAD
ML-385
(Catalog# : 179119, Cas# :
846557-71-9
)
ML-385是强有力的和有选择性的Nrf2抑制剂(IC50 = 1.9μNrf2;M)。ML-3
ML-277
(Catalog# : 179115, Cas# :
516480-79-8
)
ML-277,又名Chk2抑制剂II,是Chk2(检查点激酶2)抑制剂。ML-277凋亡
MDK35833
(Catalog# : 179114, Cas# :
1016535-83-3
)
MDK35833又称为Oct3/4-inducer-1,是一种有效率的Oct3/4诱导者。MDK35833可
ML241 HCl
(Catalog# : 179111, Cas# :
2070015-13-1
)
ML241是强有力的和有选择性的蛋白酶抑制剂。ML241抑制P97 ATPase与IC
ML364
(Catalog# : 179833, Cas# :
1991986-30-1
)
ML364是具有潜在抗癌活性的小分子抑制剂的去泛素化酶USP2。
盐酸米托蒽醌
(Catalog# : 179827, Cas# :
70476-82-3
)
盐酸米托蒽醌是一种蒽醌抗生素,具有抗肿瘤活性的盐酸盐。米托
ML311
(Catalog# : 179826, Cas# :
315698-17-0
)
ML311,也被称为EU-5346,是强有力的和有选择性的Mcl-1和Bim蛋白相互
ML-18
(Catalog# : 179810, Cas# :
1422269-30-4
)
ML-18是蛙皮素受体亚型3(BRS-3)拮抗剂(IC50 = 4.8μm)。ML-18抑制肺
1-甲基咪唑烷-2,4,5-三酮
(Catalog# : 1781501, Cas# :
3659-97-0
)
1-甲基咪唑烷-2,4,5-三酮;1-MethyliMidazolidine-2,4,5-Trione
MK-1064
(Catalog# : 16123054, Cas# :
1207253-08-4
)
MK-1064是一种有效的、选择性和口服的Orexin OX2受体拮抗剂,用于治
MI-503
(Catalog# : 178908, Cas# :
1857417-13-0
)
MI-503是一种具有IC50为14.7 nM的有效和选择性的menin - mll抑制剂。在
Merestinib (LY2801653)
(Catalog# : 178905, Cas# :
1206799-15-6
)
Merestinib,又名LY2801653,是一种可口服的小分子抑制剂,原癌基因
米格鲁特盐酸盐
(Catalog# : 2017824, Cas# :
210110-90-0
)
米格鲁特, 也称为OGT 918,是Actelion开发的一种药物,主要用于治疗I
MK-0812
(Catalog# : 2017080111, Cas# :
624733-88-6
)
MK-0812是一种有效、选择性的CCR2拮抗剂。趋化因子受体2(CCR2)是单核
红曲素
(Catalog# : 201708015, Cas# :
21516-68-7
)
它是一种有效的抑制剂,是由car纤维组织形成来测量不利的化学或
美芬妥因
(Catalog# : 174161, Cas# :
50-12-4
)
美芬妥因是一个乙内酰脲,用作抗惊厥剂。美芬妥因(CAS 50-12- 4)是
MT-DADMe-ImmA
(Catalog# : 703301, Cas# :
653592-04-2
)
Methylthio-DADMe-immucillin-A (MT-DADMe-ImmA) 是一种5 -甲基硫腺苷磷酸化酶
MI-463
(Catalog# : 17031006, Cas# :
1628317-18-9
)
MI-463是一种Menin-MLL强力抑制剂,与IC50值15.3 nM相互作用。
ML-098
(Catalog# : 17030910, Cas# :
878978-76-8
)
ML-098, 也叫 CID- 7345532,是GTP结合蛋白Rab7(EC50 = 77.6 nM)的激活剂。
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
ECI830
(Catalog# : 26A031, Cas# :
3054692-62-2
)
ECI830是一种实验性的CDK2抑制剂。
GNE-317
(Catalog# : 52282, Cas# :
1394076-92-6
)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
DPTX-3186
(Catalog# : 26A010, Cas# :
3118994-80-9
)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108, Cas# :
435327-40-5
)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
Iclepertin (BI-425809)
(Catalog# : 24084, Cas# :
1421936-85-7
)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
Kartogenin ( KGN )
(Catalog# : 52215, Cas# :
4727-31-5
)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602, Cas# :
218791-21-0
)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
Apecotrep (BI 764198)
(Catalog# : 26A048, Cas# :
2311863-36-0
)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
BH-30643
(Catalog# : 26A047, Cas# :
3062177-59-4
)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制