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抑制剂/受体激动剂
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
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产品名字索引 M
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产品名字索引 M
4-methylsulfonyl-2-(trifluoromethyl)benzaldehyde
(Catalog# : 1712293, Cas# :
1215310-75-0
)
4-methylsulfonyl-2-(trifluoromethyl)benzaldehyde isa building blocks.
MK-8617
(Catalog# : 1710163, Cas# :
1187990-87-9
)
MK-8617是一种缺氧诱导因子(HIF脯氨酰羟化酶1−3 PHD1−3),具有强效
MSC2530818
(Catalog# : 1710135, Cas# :
1883423-59-3
)
MSC2530818是一种强效、选择性,口服生物利用度与抑制剂的IC50 = 2.
MDK19922
(Catalog# : 1791512, Cas# :
132819-92-2
)
MDK19922,也称为NOD-IN-1或化合物4,是一种有效的核苷酸结合寡聚化
游离莫扎伐普坦
(Catalog# : 179154, Cas# :
137975-06-5
)
莫扎伐普坦,又名OPC 31260,是由大冢销售的血管加压素受体拮抗剂
ML-141
(Catalog# : 179152, Cas# :
71203-35-5
)
ML-141,也称为CID2950007,是Cdc42抑制剂(EC50 = 2.1μm)。
MDK30165
(Catalog# : 179138, Cas# :
2060530-16-5
)
MDK30165,也称为K-Ras(G12C)抑制剂6。
单甲基澳瑞他汀 D
(Catalog# : 20179132, Cas# :
203849-91-6
)
MMAD又称为单甲基澳瑞他汀 D,是一种高效的微管蛋白抑制剂。MMAD
ML-385
(Catalog# : 179119, Cas# :
846557-71-9
)
ML-385是强有力的和有选择性的Nrf2抑制剂(IC50 = 1.9μNrf2;M)。ML-3
ML-277
(Catalog# : 179115, Cas# :
516480-79-8
)
ML-277,又名Chk2抑制剂II,是Chk2(检查点激酶2)抑制剂。ML-277凋亡
MDK35833
(Catalog# : 179114, Cas# :
1016535-83-3
)
MDK35833又称为Oct3/4-inducer-1,是一种有效率的Oct3/4诱导者。MDK35833可
ML241 HCl
(Catalog# : 179111, Cas# :
2070015-13-1
)
ML241是强有力的和有选择性的蛋白酶抑制剂。ML241抑制P97 ATPase与IC
ML364
(Catalog# : 179833, Cas# :
1991986-30-1
)
ML364是具有潜在抗癌活性的小分子抑制剂的去泛素化酶USP2。
盐酸米托蒽醌
(Catalog# : 179827, Cas# :
70476-82-3
)
盐酸米托蒽醌是一种蒽醌抗生素,具有抗肿瘤活性的盐酸盐。米托
ML311
(Catalog# : 179826, Cas# :
315698-17-0
)
ML311,也被称为EU-5346,是强有力的和有选择性的Mcl-1和Bim蛋白相互
ML-18
(Catalog# : 179810, Cas# :
1422269-30-4
)
ML-18是蛙皮素受体亚型3(BRS-3)拮抗剂(IC50 = 4.8μm)。ML-18抑制肺
1-甲基咪唑烷-2,4,5-三酮
(Catalog# : 1781501, Cas# :
3659-97-0
)
1-甲基咪唑烷-2,4,5-三酮;1-MethyliMidazolidine-2,4,5-Trione
MK-1064
(Catalog# : 16123054, Cas# :
1207253-08-4
)
MK-1064是一种有效的、选择性和口服的Orexin OX2受体拮抗剂,用于治
MI-503
(Catalog# : 178908, Cas# :
1857417-13-0
)
MI-503是一种具有IC50为14.7 nM的有效和选择性的menin - mll抑制剂。在
Merestinib (LY2801653)
(Catalog# : 178905, Cas# :
1206799-15-6
)
Merestinib,又名LY2801653,是一种可口服的小分子抑制剂,原癌基因
米格鲁特盐酸盐
(Catalog# : 2017824, Cas# :
210110-90-0
)
米格鲁特, 也称为OGT 918,是Actelion开发的一种药物,主要用于治疗I
MK-0812
(Catalog# : 2017080111, Cas# :
624733-88-6
)
MK-0812是一种有效、选择性的CCR2拮抗剂。趋化因子受体2(CCR2)是单核
红曲素
(Catalog# : 201708015, Cas# :
21516-68-7
)
它是一种有效的抑制剂,是由car纤维组织形成来测量不利的化学或
美芬妥因
(Catalog# : 174161, Cas# :
50-12-4
)
美芬妥因是一个乙内酰脲,用作抗惊厥剂。美芬妥因(CAS 50-12- 4)是
MT-DADMe-ImmA
(Catalog# : 703301, Cas# :
653592-04-2
)
Methylthio-DADMe-immucillin-A (MT-DADMe-ImmA) 是一种5 -甲基硫腺苷磷酸化酶
MI-463
(Catalog# : 17031006, Cas# :
1628317-18-9
)
MI-463是一种Menin-MLL强力抑制剂,与IC50值15.3 nM相互作用。
ML-098
(Catalog# : 17030910, Cas# :
878978-76-8
)
ML-098, 也叫 CID- 7345532,是GTP结合蛋白Rab7(EC50 = 77.6 nM)的激活剂。
ML-265
(Catalog# : 17030804, Cas# :
1221186-53-3
)
ML265是一个强有力的PKM2活化剂诱导四聚体,降低肿瘤的形成和大小
MN-64
(Catalog# : 17030717, Cas# :
92831-11-3
)
MN-64 是一种有效的、选择性的Tankyrase 1和2抑制剂(IC50值分别为6和
ML241
(Catalog# : 17030714, Cas# :
1346528-06-0
)
ML241是一种p97 ATPase有效的选择性抑制剂。ML241抑制p97 ATPase的IC(50)值
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AD-8007
(Catalog# : 26A018, Cas# :
1497439-74-3
)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
ZY-444
(Catalog# : 26A020, Cas# :
1802650-31-2
)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
AD-5584
(Catalog# : 26A019, Cas# :
2306525-79-9
)
AD-5584是一种新型脑渗透性ACSS2抑制剂。
IDB-003
(Catalog# : 26A017, Cas# :
3079716-11-0
)
IDB-003在体内抑制MDA-MB-231肿瘤生长。
Vafidemstat
(Catalog# : 18891, Cas# :
1357362-02-7
)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
LLL12
(Catalog# : 25075, Cas# :
1260247-42-4
)
LLL12是一种强效的STAT3抑制剂。LLL12在小鼠异种移植物模型中显示出
ECC-5004
(Catalog# : 26A015, Cas# :
2758659-09-3
)
ECC5004是一款每日一次、低剂量、小分子GLP-1受体激动剂。
SILA-123
(Catalog# : 26A014, Cas# :
2911585-37-8
)
SILA-123是一种II型FLT3抑制剂,对FLT3-WT(IC50=2.1 nM)和FLT3-ITD(IC50=1
Encaleret sulfate
(Catalog# : 26A013, Cas# :
1214922-52-7
)
Encaleret是一种正在研究的钙敏感受体的小分子拮抗剂,用于钙稳态
Iadademstat ( ORY-1001 ) hydrochloride
(Catalog# : 26A011, Cas# :
1431303-72-8
)
Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶