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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
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On Sale
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联系我们
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产品名字索引 M
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产品名字索引 M
MDK19922
(Catalog# : 1791512, Cas# :
132819-92-2
)
MDK19922,也称为NOD-IN-1或化合物4,是一种有效的核苷酸结合寡聚化
游离莫扎伐普坦
(Catalog# : 179154, Cas# :
137975-06-5
)
莫扎伐普坦,又名OPC 31260,是由大冢销售的血管加压素受体拮抗剂
ML-141
(Catalog# : 179152, Cas# :
71203-35-5
)
ML-141,也称为CID2950007,是Cdc42抑制剂(EC50 = 2.1μm)。
MDK30165
(Catalog# : 179138, Cas# :
2060530-16-5
)
MDK30165,也称为K-Ras(G12C)抑制剂6。
单甲基澳瑞他汀 D
(Catalog# : 20179132, Cas# :
203849-91-6
)
MMAD又称为单甲基澳瑞他汀 D,是一种高效的微管蛋白抑制剂。MMAD
ML-385
(Catalog# : 179119, Cas# :
846557-71-9
)
ML-385是强有力的和有选择性的Nrf2抑制剂(IC50 = 1.9μNrf2;M)。ML-3
ML-277
(Catalog# : 179115, Cas# :
516480-79-8
)
ML-277,又名Chk2抑制剂II,是Chk2(检查点激酶2)抑制剂。ML-277凋亡
MDK35833
(Catalog# : 179114, Cas# :
1016535-83-3
)
MDK35833又称为Oct3/4-inducer-1,是一种有效率的Oct3/4诱导者。MDK35833可
ML241 HCl
(Catalog# : 179111, Cas# :
2070015-13-1
)
ML241是强有力的和有选择性的蛋白酶抑制剂。ML241抑制P97 ATPase与IC
ML364
(Catalog# : 179833, Cas# :
1991986-30-1
)
ML364是具有潜在抗癌活性的小分子抑制剂的去泛素化酶USP2。
盐酸米托蒽醌
(Catalog# : 179827, Cas# :
70476-82-3
)
盐酸米托蒽醌是一种蒽醌抗生素,具有抗肿瘤活性的盐酸盐。米托
ML311
(Catalog# : 179826, Cas# :
315698-17-0
)
ML311,也被称为EU-5346,是强有力的和有选择性的Mcl-1和Bim蛋白相互
ML-18
(Catalog# : 179810, Cas# :
1422269-30-4
)
ML-18是蛙皮素受体亚型3(BRS-3)拮抗剂(IC50 = 4.8μm)。ML-18抑制肺
1-甲基咪唑烷-2,4,5-三酮
(Catalog# : 1781501, Cas# :
3659-97-0
)
1-甲基咪唑烷-2,4,5-三酮;1-MethyliMidazolidine-2,4,5-Trione
MK-1064
(Catalog# : 16123054, Cas# :
1207253-08-4
)
MK-1064是一种有效的、选择性和口服的Orexin OX2受体拮抗剂,用于治
MI-503
(Catalog# : 178908, Cas# :
1857417-13-0
)
MI-503是一种具有IC50为14.7 nM的有效和选择性的menin - mll抑制剂。在
Merestinib (LY2801653)
(Catalog# : 178905, Cas# :
1206799-15-6
)
Merestinib,又名LY2801653,是一种可口服的小分子抑制剂,原癌基因
米格鲁特盐酸盐
(Catalog# : 2017824, Cas# :
210110-90-0
)
米格鲁特, 也称为OGT 918,是Actelion开发的一种药物,主要用于治疗I
MK-0812
(Catalog# : 2017080111, Cas# :
624733-88-6
)
MK-0812是一种有效、选择性的CCR2拮抗剂。趋化因子受体2(CCR2)是单核
红曲素
(Catalog# : 201708015, Cas# :
21516-68-7
)
它是一种有效的抑制剂,是由car纤维组织形成来测量不利的化学或
美芬妥因
(Catalog# : 174161, Cas# :
50-12-4
)
美芬妥因是一个乙内酰脲,用作抗惊厥剂。美芬妥因(CAS 50-12- 4)是
MT-DADMe-ImmA
(Catalog# : 703301, Cas# :
653592-04-2
)
Methylthio-DADMe-immucillin-A (MT-DADMe-ImmA) 是一种5 -甲基硫腺苷磷酸化酶
MI-463
(Catalog# : 17031006, Cas# :
1628317-18-9
)
MI-463是一种Menin-MLL强力抑制剂,与IC50值15.3 nM相互作用。
ML-098
(Catalog# : 17030910, Cas# :
878978-76-8
)
ML-098, 也叫 CID- 7345532,是GTP结合蛋白Rab7(EC50 = 77.6 nM)的激活剂。
ML-265
(Catalog# : 17030804, Cas# :
1221186-53-3
)
ML265是一个强有力的PKM2活化剂诱导四聚体,降低肿瘤的形成和大小
MN-64
(Catalog# : 17030717, Cas# :
92831-11-3
)
MN-64 是一种有效的、选择性的Tankyrase 1和2抑制剂(IC50值分别为6和
ML241
(Catalog# : 17030714, Cas# :
1346528-06-0
)
ML241是一种p97 ATPase有效的选择性抑制剂。ML241抑制p97 ATPase的IC(50)值
ML348
(Catalog# : 17030712, Cas# :
899713-86-1
)
ML348,又称CID 3238952;SID 160654487,是一个可逆的LYPLA1抑制剂,IC50值
MMAF (Monomethyl auristatin F)
(Catalog# : 17030611, Cas# :
745017-94-1
)
一甲基澳瑞他汀 F(MMAF)是一种合成抗肿瘤药物。它是一些实验性抗
Merimepodib
(Catalog# : 17030308, Cas# :
198821-22-6
)
Merimepodib, 也称为VX-497,是有效的口服生物IMPDH抑制剂,它可以抑制
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AZD0095
(Catalog# : 237072, Cas# :
2750001-23-9
)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2-MNG
(Catalog# : 24129, Cas# :
2101538-28-5
)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
MAT2A-IN-9
(Catalog# : 25147, Cas# :
2439277-80-0
)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
Acoramidis hydrochloride
(Catalog# : 24068, Cas# :
2242751-53-5
)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
Crelosidenib
(Catalog# : 24101, Cas# :
2230263-60-0
)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
LOXO-435
(Catalog# : 25080, Cas# :
2833703-74-3
)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
Gridegalutamide
(Catalog# : 25138, Cas# :
2446928-30-7
)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
Chiauranib
(Catalog# : 25146, Cas# :
1256349-48-0
)
Chiauranib also known as orally available, small molecule inhibitor of select serine-