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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
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产品名字索引 F
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产品名字索引 F
FM19G11
(Catalog# : 192211, Cas# :
329932-55-0
)
FM19G11是缺氧诱导因子α的抑制剂(HIFα),据报道,影响干细胞的自我更
Fmk
(Catalog# : 188102, Cas# :
821794-92-7
)
强效不可逆RSK1/2抑制剂(IC50 = 15nm)。灭活C端自激酶域活性。
Fezolinetant
(Catalog# : 18722, Cas# :
1629229-37-3
)
Fezolinetant,也被称为ESN-364,是一种神经kinin-3 (NK-3)受体拮抗剂,已
FRAX486
(Catalog# : 18721, Cas# :
1232030-35-1
)
FRAX486是一种有效的p21激活激酶(PAK)抑制剂(PAK1、PAK2、PAK3和PAK4的IC
非阿尿苷
(Catalog# : 184283, Cas# :
69123-98-4
)
非阿尿苷,又名FIAU, DRG-0098,是一种DNA定向DNA聚合酶抑制剂,可用
Fonadelpar
(Catalog# : 18445, Cas# :
515138-06-4
)
Fonadelpar是一个强有力的和选择性的过氧物酶体扩散者激活受体δ(
FM-381
(Catalog# : 18436, Cas# :
unknown
)
FM-381是JAK3和JAK3特定可逆共价抑制剂的化学探针。
Fmoc-Val-Ala-PAB
(Catalog# : 18431, Cas# :
1394238-91-5
)
Fmoc-Val-Ala-PAB, also known as Fmoc-Val-Ala-PAB-OH, is a useful linker for making An
Ferrostatin-1
(Catalog# : 184210, Cas# :
347174-05-4
)
Ferrostatin-1 (Fer-1) is a lipophilic antioxidant that effectively blocks ferroptosis
Fostemsavir
(Catalog# : 1712155, Cas# :
864953-29-7
)
Fostemsavir,也称为BMS-663068,是一种口服,安全有效的 HIV- 1附着抑
Farampator
(Catalog# : 179156, Cas# :
211735-76-1
)
Farampator,也称为ORG-24448;CX-691,是AMPA受体阳性变构调节剂可能用
FRAX1036
(Catalog# : 1791315, Cas# :
1432908-05-8
)
frax1036是强有力的和有选择性的激酶抑制剂。
FITM
(Catalog# : 17989, Cas# :
932737-65-0
)
FITM是一种有效的mGlu1 抑制剂。
Fluralaner
(Catalog# : 178309, Cas# :
864731-61-3
)
Fluralaner也称为AH252723,是一种经口服给药的系统杀虫剂和杀螨剂。
4-氟-2-甲氧基-5-硝基苯胺
(Catalog# : 521191, Cas# :
1075705-01-9
)
AZD9291中间体1
4-FORMYL-2-METHOXY-3-NITROPHENYL ACETATE
(Catalog# : 178225, Cas# :
2698-69-3
)
4-FORMYL-2-METHOXY-3-NITROPHENYL ACETATE
1-(3-Fluorophenyl)-cyclohexanamine HCl
(Catalog# : 178221, Cas# :
125802-18-8
)
1-(3-Fluorophenyl)-cyclohexanamine HCl
FPS-ZM1
(Catalog# : 16123002, Cas# :
945714-67-0
)
FPS-ZM1 is a high-affinity RAGE-specific blocker that inhibits amyloid- binding to RA
Flutamide
(Catalog# : 16123001, Cas# :
13311-84-7
)
Flutamide, also known as SCH13521, is a toluidine derivative and nonsteroidal antiand
Firategrast
(Catalog# : 16122946, Cas# :
402567-16-2
)
Firategrast, also known as SB-683699 or T-0047, is an orally bioavailable alpha4 beta
FIIN-3
(Catalog# : 16122945, Cas# :
1637735-84-2
)
FIIN-3 is a potent, selective, irreversible and the next-generation covalent FGFR inh
FGFR4-IN-1
(Catalog# : 16122813, Cas# :
1708971-72-5
)
FGFR4-IN-1 is a potent and selective FGFR4 inhibitor. FGFR4 may be a novel therapeuti
FG-2216
(Catalog# : 16122812, Cas# :
223387-75-5
)
FG-2216, also known as YM311, is orally bioavailable HIF-prolyl hydroxylase inhibitor
FH535
(Catalog# : 16122788, Cas# :
108409-83-2
)
FH535 is a Wnt/-catenin signaling inhibitor and also a dual PPAR and PPAR antagonist.
FLLL32
(Catalog# : 16122709, Cas# :
1226895-15-3
)
FLLL32 is a potent JAK2/STAT3 inhibitor with IC50 of <5 M.In MDA-MB-231 breast and
Fevipiprant ( NVP-QAW039 )
(Catalog# : 90102, Cas# :
872365-14-5
)
Fevipiprant (QAW039; NVP-QAW039) is a selective, potent, reversible competitive CRTh2
Filanesib
(Catalog# : 16071102, Cas# :
885060-09-3
)
Filanesib, also known as ARRY-520, is a synthetic, small molecule targeting the kines
FK866(APO866,Daporinad)
(Catalog# : 1662306, Cas# :
658084-64-1
)
FK866 is a highly specific noncompetitive inhibitor of nicotinamide phosphoribosyltra
FIIN-2
(Catalog# : 16062117, Cas# :
1633044-56-0
)
FIIN-2 is a potent, selective, irreversible and the next-generation covalent FGFR inh
FPH2
(Catalog# : 032513, Cas# :
957485-64-2
)
Coming soon!
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
ECI830
(Catalog# : 26A031, Cas# :
3054692-62-2
)
ECI830是一种实验性的CDK2抑制剂。
GNE-317
(Catalog# : 52282, Cas# :
1394076-92-6
)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
DPTX-3186
(Catalog# : 26A010, Cas# :
3118994-80-9
)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108, Cas# :
435327-40-5
)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
Iclepertin (BI-425809)
(Catalog# : 24084, Cas# :
1421936-85-7
)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
Kartogenin ( KGN )
(Catalog# : 52215, Cas# :
4727-31-5
)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602, Cas# :
218791-21-0
)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
Apecotrep (BI 764198)
(Catalog# : 26A048, Cas# :
2311863-36-0
)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
BH-30643
(Catalog# : 26A047, Cas# :
3062177-59-4
)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制