武汉永璨生物科技有限公司
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抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
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Epigenetics
GPCR & G Protein
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MAPK
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Metabolism
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NF-κB
Protein Tyrosine Kinase
Proteases
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TGF-beta/Smad
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Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
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产品名字索引 N
NCH-51
(Catalog# : 17030716, Cas# :
848354-66-5
)
NCH-51, 也叫PTACH,是一种组蛋白去乙酰化酶(HDAC)抑制剂。NCH-51抑制
NS-1643
(Catalog# : 17030715, Cas# :
448895-37-2
)
NS-1643是一种人类ether-a-go-go相关基因(hERG)KV11.1通道激活剂(EC50 = 10.
Nifenalol HCl
(Catalog# : 17030705, Cas# :
5704-60-9
)
Nifenalol,也叫INPEA,是一种新型的β-肾上腺素受体拮抗剂。
聚乙二醇纳诺醇
(Catalog# : 17030202, Cas# :
1354744-91-4
)
Naloxegol,也称为NKTR-118和AZ-13337019,是一种选择性的阿片拮抗剂,用于
尼拉帕尼盐酸盐
(Catalog# : 17030114, Cas# :
1038915-64-8
)
尼拉帕尼, 也称为MK-4827, 是一种具有潜在抗肿瘤活性的聚(ADP-核糖
那可汀盐酸盐
(Catalog# : 17022711, Cas# :
912-60-7
)
那可汀, 也被称为麻醉药物,阿片烷,是一种来自罂粟科植物的be
Nampt-IN-1
(Catalog# : 17022705, Cas# :
1698878-14-6
)
Nampt-IN-1是NAMPT的一种新型抑制剂,IC50分别为18 nM(NCI- H1155细胞),4
NSC12
(Catalog# : 17021317, Cas# :
102586-30-1
)
NSC12是一种可用于抑制FGF2 / FGFR相互作用并具有良好的抗肿瘤活性
NS-398 (NS398)
(Catalog# : 17011106, Cas# :
123653-11-2
)
NS-398是一种cyclooxygenase-2 (COX-2)的选择性抑制剂。
Netarsudil (AR-13324) 2HCl
(Catalog# : 1710901, Cas# :
1253952-02-1
)
Netarsudil (a.k.a. AR-13324)是一种ROCK抑制剂,Ki值为 0.2-10.3 nM。它目前
Naftifine
(Catalog# : 16122834, Cas# :
65472-88-0
)
Naftifine is an allylamine antifungal drug for the topical treatment of tinea pedis,
Nafamostat mesylate
(Catalog# : 16122833, Cas# :
82956-11-4
)
Nafamostat, also known as FUT-175, is a serine protease inhibitor and an anticoagulan
NSC697923
(Catalog# : 16122791, Cas# :
343351-67-7
)
NSC697923 is a cell-permeable and selective inhibitor of the Ub-conjugating enzyme (E
NVP-CGM097
(Catalog# : 16122789, Cas# :
1313363-54-0
)
NVP-CGM097 is a highly potent and selective MDM2 inhibitor. It binds to the p53 bindi
NSC228155
(Catalog# : 16122779, Cas# :
113104-25-9
)
NSC228155 is an activator of EGFR, binding to the sEGFR dimerization domain II and mo
NQDI-1
(Catalog# : 16122772, Cas# :
175026-96-7
)
NQDI 1, an inhibitor of ASK1(apoptosis signal-regulating kinase 1), attenuates acute
Nitroxoline
(Catalog# : 16122719, Cas# :
4008-48-4
)
Nitroxoline is a urinary antibacterial agent active against susceptible gram-positive
Napabucasin
(Catalog# : 16122708, Cas# :
83280-65-3
)
Napabucasin is an orally available Stat3 and cancer cell stemness inhibitor.Napabucas
Necrosulfonamide
(Catalog# : 6111508, Cas# :
1360614-48-7
)
Necrosulfonamide is a very specific and potent necrosis inhibitor and blocks mixed li
Necrostatin 2 S enantiomer
(Catalog# : 6111412, Cas# :
852391-20-9
)
Necrostatin 2 is a potent necroptosis inhibitor with EC50 of 50 nM.Necrostatin 2 is a
Necrostatin 2 racemate
(Catalog# : 6111411, Cas# :
852391-15-2
)
Necrostatin 2 is a potent necroptosis inhibitor with EC50 of 50 nM.Necrostatin 2 is a
NBI-74330
(Catalog# : 6111112, Cas# :
855527-92-3
)
NBI-74330 is a small molecule antagonist for CXCR3, NBI-74330 demonstrates potent inh
Nastorazepide
(Catalog# : 6111110, Cas# :
209219-38-5
)
Nastorazepide (Z-360) is a selective, orally available, 1,5-benzodiazepine-derivative
NU6300
(Catalog# : 611923, Cas# :
2070015-09-5
)
NU6300 is a non-covalent ATP-competitive CDK2 inhibitor (IC50 = 0.16 mM). NU6300
NU 7026
(Catalog# : 6118017, Cas# :
154447-35-5
)
NU 7026 is a novel and potential inhibitor of the DNA repair enzyme DNA-dependent pro
NMS-859
(Catalog# : 161014001, Cas# :
1449236-96-7
)
NMS-859 is a potent and specific small molecule covalent inhibitor of the ATPase VCP/
NCT-501
(Catalog# : 16071414, Cas# :
1802088-50-1
)
NCT-501 is a potent ALDH1A1 inhibitor. Aldehyde dehydrogenases (ALDHs) metabolize rea
Naquotinib
(Catalog# : 16071107, Cas# :
448232-80-1
)
Naquotinib, also known as ASP8273, is an orally available, irreversible, third-genera
Necrostatin 2
(Catalog# : 16070914, Cas# :
852391-19-6
)
Necrostatin 2
Navitoclax (ABT-263)
(Catalog# : 16070102, Cas# :
923564-51-6
)
Navitoclax, also known as ABT-263, is an orally bioavailable, synthetic small-molecul
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive-Oxygen-Species-ROS
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Mitoquinol mesylate (MitoQ)
(Catalog# : 26A042, Cas# :
845959-55-9
)
Mitoquinol mesylate (MitoQ) 是一种线粒体靶向抗氧化剂,具体而言,它
SPG-601 ( VSN-16R )
(Catalog# : 24042, Cas# :
1246960-09-7
)
SPG-601(原名VSN-16R)是一种口服给药、同类首创的小分子药物,是
LY3039478 ( Crenigacestat )
(Catalog# : 17021601, Cas# :
1421438-81-4
)
LY3039478 ( Crenigacestat ) 是一种选择性 NOTCH1 抑制剂,通过阻断 VEGFA/
PF-9366
(Catalog# : 184107, Cas# :
72882-78-1
)
PF-9366是一种新型的人蛋氨酸腺苷转移酶2A (Mat2A),肝外同种型。
MAT2A-IN-22
(Catalog# : 26A021, Cas# :
2925330-18-1
)
MAT2A-IN-22 (Compound 29-1) 是一种可透过血脑屏障的和口服有效的 MAT2A
Pantothenate kinase-IN-3
(Catalog# : 26A041)
泛酸激酶-IN-3(亦称化合物21,https://doi.org/10.1021/acs.jmedchem.5c03452)
Claziprotamidum ( Claziprotamide ; BBP-671 )
(Catalog# : 26A040, Cas# :
2361124-03-8
)
Claziprotamidum(Claziprotamide;BBP-671)是一种强效、口服有效且能透过
PZ-3022
(Catalog# : 26A039, Cas# :
2170608-85-0
)
PZ-3022是一种别构型的PanK激活剂,能够抵消C3-CoA的抑制作用。
PZ-2891
(Catalog# : 193282, Cas# :
2170608-82-7
)
PZ-2891是一种强效的、选择性的、口服活性泛酸激酶(PANK)调制剂,
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,