武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
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Nitro Compounds
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Peg Linkers
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Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
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定制合成
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产品名字索引 N
NVS-PAK1-1
(Catalog# : 21231, Cas# :
1783816-74-9
)
NVS-PAK1-1 is a a specific allosteric PAK1 inhibitor.
Niraparib tosylate hydrate
(Catalog# : 2021115, Cas# :
1613220-15-7
)
Niraparib, also know as MK-4827, is an inhibitor of poly (ADP-ribose) polymerase (PAR
N-(8-Benzyl-8-azabicyclo[3.2.1]oct-3-yl-exo)-2-methylpropanamide
(Catalog# : 2071632, Cas# :
376348-67-3
)
NCC007
(Catalog# : 2071529)
NCC007 is a novel CKIα and CKIδ dual inhibitor. NCC007 that showed stronger period
N-tert-butyl-3-[(2-chloro-5-methylpyrimidin-4-yl)amino]benzenesulfonamide
(Catalog# : 2062304, Cas# :
936092-53-4
)
N,N-dibenzyl-6-chloro-5-nitropyrimidine-4-amine
(Catalog# : 2062033, Cas# :
882272-97-1
)
N-(3,5-dimethoxyphenyl)-3-(1-methyl-1H-pyrazol-4-yl)quinoxalin-6-amine
(Catalog# : 2062032, Cas# :
1346133-39-8
)
N-(2-methylbenzyl)-4,5-dihydro-1H-imidazol-2-amine
(Catalog# : 2062031, Cas# :
38941-29-6
)
5-(N-PHTHALIMIDO)-2-PENTANONE
(Catalog# : 2062010, Cas# :
3197-25-9
)
N-Fmoc-O-[3,4,6-tri-O-acetyl-2-(acetylamino)-2-deoxy-α-D-galactopyranosyl]-L-serine
(Catalog# : 2061601, Cas# :
120173-57-1
)
NTP42
(Catalog# : 2051509, Cas# :
2055599-51-2
)
NTP42 is a novel antagonist of the thromboxane prostanoid receptor (TP), currently in
N-Boc-吡咯
(Catalog# : S-204153, Cas# :
5176-27-2
)
N-(4-戊炔基)酞酰亚胺
(Catalog# : S-204150, Cas# :
6097-07-0
)
N-benzyl-2,4-dichloropyrimidine-5-carboxamide
(Catalog# : 197101, Cas# :
1019115-13-9
)
NVS-ZP7-4
(Catalog# : 204506, Cas# :
2349367-89-9 (free base)
)
NVS-ZP7-4 is a potent ZIP7 Inhibitor, which inhibits Notch signaling with IC50 of 0.1
NVP-2
(Catalog# : 193205, Cas# :
1263373-43-8
)
NVP-2是细胞周期蛋白依赖性激酶CDK9的抑制剂。
NS-1652
(Catalog# : 19361, Cas# :
1566-81-0
)
NS-1652是一种阴离子电导抑制剂。
NCT-506
(Catalog# : 19354, Cas# :
2231098-99-8
)
NCT-506是一种口服生物可利用醛脱氢酶1A1 (ALDH1A1)抑制剂,IC50为7nm。
Nelotanserin
(Catalog# : 191121, Cas# :
839713-36-9
)
Nelotanserin( APD125) is a potent and selective human 5-hydroxytryptamine2A inverse a
ND-646
(Catalog# : 191102, Cas# :
1434639-57-2
)
ND-646是ACC酶ACC1和ACC2的变构抑制剂,可阻止ACC亚基二聚化,在体内
ND-630
(Catalog# : 19133, Cas# :
1434635-54-7
)
ND-630,也称为GS-0976, NDI-010976和firsocostat, 是一种有效的ACC抑制剂。
Naquotinib游离
(Catalog# : 1812297, Cas# :
1448232-80-1
)
Naquotinib,又称ASP8273,是一种口服、不可逆、第三代、突变选择、
N6022
(Catalog# : 1811304, Cas# :
1208315-24-5
)
N6022是一种有效、选择性、可逆性和有效性的s -亚硝基谷胱甘肽还
Nexinhib20
(Catalog# : 1811152, Cas# :
331949-35-0
)
Nexinhib20是一种Rab27抑制剂,可以抑制中性粒细胞的胞外活动,在体
NGI-1
(Catalog# : 181171, Cas# :
790702-57-7
)
NGI-1,又称ML414,是低聚糖转移酶(OST)的一种细胞渗透性抑制剂。
NMS-E973
(Catalog# : 1810293, Cas# :
1253584-84-7
)
NMS-E973是一种新型、选择性和强效的热休克蛋白90 (Hsp90)抑制剂。
NCT-505
(Catalog# : 1810261, Cas# :
2231079-74-4
)
NCT-505是一种口服生物有效醛脱氢酶1A1 (ALDH1A1)抑制剂,具有较强的
NVP-BGG463
(Catalog# : 1810233, Cas# :
890129-26-7
)
NVP-BGG463是一种新型的II型激酶抑制剂,靶向CDK2。
NS1619
(Catalog# : 1810227, Cas# :
153587-01-0
)
NS1619是一种Bkca开启工具或大电导Ca2+活化钾(Bkca, KCa1.1)通道激活器
Nacubactam
(Catalog# : 185169, Cas# :
1452458-86-4
)
Nacubactam, 也称为RG-6080, FPI-1459, 和OP-0595, 是一种β-内酰胺酶抑制剂
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
CT1812 ( Zervimesine )
(Catalog# : 193283, Cas# :
1802632-22-9
)
CT-1812是一种同类首创的、可口服的sigma-2/PGRMC1拮抗剂(αβ寡聚体
BLU-808
(Catalog# : 26A024, Cas# :
3041025-10-6
)
BLU-808是一种针对肥大细胞疾病的野生型c-KIT的强效且具有选择性的
Zedoresertib
(Catalog# : 26A023, Cas# :
2243882-74-6
)
Zedoresertib(Debio 0123)是一种脑渗透剂,高选择性WEE1激酶抑制剂。
BEN-28010
(Catalog# : 26A022, Cas# :
3033961-38-2
)
BEN-28010是一种自由脑渗透剂,强效且具有选择性的CHK1抑制剂。
4-((2-(甲氨基)-6-(2,2,2-三氟乙基)噻吩并[2,3-d]嘧啶-4-基)氨基)哌啶-1-甲酸叔丁酯
(Catalog# : 26B007, Cas# :
3107291-07-3
)
Muvalaplin
(Catalog# : 20528, Cas# :
2565656-70-2
)
Muvalaplin是一种小分子,通过干扰载脂蛋白(a)与载脂蛋白B100的结合
MAT2A-IN-22
(Catalog# : 26A021, Cas# :
2925330-18-1
)
MAT2A-IN-22 (Compound 29-1) 是一种可透过血脑屏障的和口服有效的 MAT2A
AD-8007
(Catalog# : 26A018, Cas# :
1497439-74-3
)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
ZY-444
(Catalog# : 26A020, Cas# :
1802650-31-2
)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
AD-5584
(Catalog# : 26A019, Cas# :
2306525-79-9
)
AD-5584是一种新型脑渗透性ACSS2抑制剂。