武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
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产品名字索引 N
NVP-BGG463
(Catalog# : 1810233, Cas# :
890129-26-7
)
NVP-BGG463是一种新型的II型激酶抑制剂,靶向CDK2。
NS1619
(Catalog# : 1810227, Cas# :
153587-01-0
)
NS1619是一种Bkca开启工具或大电导Ca2+活化钾(Bkca, KCa1.1)通道激活器
Nacubactam
(Catalog# : 185169, Cas# :
1452458-86-4
)
Nacubactam, 也称为RG-6080, FPI-1459, 和OP-0595, 是一种β-内酰胺酶抑制剂
Navarixin
(Catalog# : 185168, Cas# :
473727-83-2
)
Navarixin, 也称为SCH527123, PS291822和MK-7123, 是一种有效的CXCR2拮抗剂。
Nemorubicin
(Catalog# : 185167, Cas# :
108852-90-0
)
Nemorubicin,又名PNU152243A,是一种不同于其母体药物的doxorubicin衍生
Nolatrexed盐酸盐
(Catalog# : 185166, Cas# :
152946-68-4
)
Nolatrexed,也叫AG337,是一种具有潜在抗癌活性的胸腺嘧啶合成酶抑
Nucleozin
(Catalog# : 185164, Cas# :
341001-38-5
)
Nucleozin是一种杀毒剂。它的目标是一种核蛋白(NP),这是一种病毒
Nidufexor
(Catalog# : 184288, Cas# :
1773489-72-7
)
Nidufexor是一个法呢醇X受体(FXR)激动剂。
1NM-PP1
(Catalog# : 184174, Cas# :
221244-14-0
)
1NM-PP1 是一种有效的突变激酶抑制剂。
Netarsudil(Mesylate)
(Catalog# : 712181, Cas# :
1422144-42-0
)
Netarsudil( AR-11324) is a Rho-associated protein kinase inhibitor. Netarsudil is pot
nor-NOHA醋酸盐
(Catalog# : 1710169, Cas# :
1140844-63-8
)
nor-NOHA是一种强效、选择性、竞争性、以及精氨酸酶的高亲和力抑
NMS-P118
(Catalog# : 17101311, Cas# :
1262417-51-5
)
NMS-P118是一种有效的、可口服、高选择性PARP-1抑制剂具有优良的AD
盐酸萘替芬
(Catalog# : 1791514, Cas# :
65473-14-5
)
萘替芬是一种丙烯胺抗真菌药物的局部治疗足癣、股癣、体癣(真
Neflamapimod
(Catalog# : 1791317, Cas# :
209410-46-8
)
Neflamapimod,也称为VX-745,VRT-031745和VD-31745,是高度有效的和选择性
盐酸纳洛酮
(Catalog# : 178305, Cas# :
357-08-4
)
纳洛酮是一种μ-opioid受体(MOR)逆受体激动剂。纳洛酮针对在中枢神
3-Nitrosalicylic Acid Methyl Ester
(Catalog# : 178224, Cas# :
22621-41-6
)
3-Nitrosalicylic Acid Methyl Ester
N-甲氧基-N-甲基乙酰胺
(Catalog# : 178223, Cas# :
78191-00-1
)
N-Methoxy-N-methylacetamide
N-(4-(benzyloxy)-3-methoxybenzyl)-5-phenyl-N-(2-(pyridin-2-yl)ethyl)pentanamide
(Catalog# : 1781506, Cas# :
521310-51-0
)
N-(4-(Benzyloxy)-3-methoxybenzyl)-5-phenyl-N-(2-(pyridin-2-yl)ethyl)pentanamide
NIH-12848
(Catalog# : 1781103, Cas# :
959551-10-1
)
NIH-12848是一种普遍认为的磷脂酰肌醇5 -磷酸四激酶(PI5P4K)抑制剂。
Nazartinib (EGF816)
(Catalog# : 1781004, Cas# :
1508250-71-2
)
Nazartinib,也被称为EGF816,是一种口服可用,不可逆转的、第三代、
Netarsudil
(Catalog# : 1781001, Cas# :
1254032-66-0
)
<span style="color:#34495E;font-family:" font-size:14px;background-color
NSC781406
(Catalog# : 20178810, Cas# :
1676893-24-5
)
NSC781406是一种高效针对PI3K的IC50为2 nM的PI3K和mTOR抑制剂。
NCT-503
(Catalog# : 2017888, Cas# :
1916571-90-8
)
NCT-503是一种3 -磷酸甘油酸脱氢酶(PHGDH)抑制剂,抑制丝氨酸合成3 -磷
NGP-555
(Catalog# : 2017875, Cas# :
1304630-27-0
)
NGP 555正在被作为一种预防疾病老年痴呆症的治疗。
N-反式-阿魏酰酪胺
(Catalog# : 201708019, Cas# :
66648-43-9
)
N-反式-阿魏酰酪胺|N-Trans-Feruloyltyramine|(E)-3-(4-hydroxy-3-Methoxy-phenyl)-
NDGA
(Catalog# : 17030909, Cas# :
500-38-9
)
去甲二氢愈创木酸(NDGA),也被称为masoprocol,是一种天然抗氧化剂dica
诺拉曲特
(Catalog# : 17030908, Cas# :
147149-76-6
)
诺拉曲特,也叫AG337,是一种具有潜在抗癌活性的百里香酶抑制剂
NPS-1034
(Catalog# : 17030907, Cas# :
1221713-92-3
)
NPS-1034是一种新型的MET抑制剂,它能抑制活化的MET受体及其具有结
NVP-BEP800
(Catalog# : 17030906, Cas# :
847559-80-2
)
NVP-BEP800, 也称为BEP-800,是一种新型的、完全合成的口服生物可用抑
制霉菌素
(Catalog# : 17030905, Cas# :
1400-61-9
)
制霉菌素是一种多烯抗真菌药物,含有三种生物活性成分的抗生素
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
ECI830
(Catalog# : 26A031, Cas# :
3054692-62-2
)
ECI830是一种实验性的CDK2抑制剂。
GNE-317
(Catalog# : 52282, Cas# :
1394076-92-6
)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
DPTX-3186
(Catalog# : 26A010, Cas# :
3118994-80-9
)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108, Cas# :
435327-40-5
)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
Iclepertin (BI-425809)
(Catalog# : 24084, Cas# :
1421936-85-7
)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
Kartogenin ( KGN )
(Catalog# : 52215, Cas# :
4727-31-5
)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602, Cas# :
218791-21-0
)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
Apecotrep (BI 764198)
(Catalog# : 26A048, Cas# :
2311863-36-0
)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
BH-30643
(Catalog# : 26A047, Cas# :
3062177-59-4
)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制