武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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Amines
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Boronic Acids
Bromides
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Deuterated
Fluorides
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Indoles and Oxindoles
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
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产品名字索引 N
Navarixin
(Catalog# : 185168, Cas# :
473727-83-2
)
Navarixin, 也称为SCH527123, PS291822和MK-7123, 是一种有效的CXCR2拮抗剂。
Nemorubicin
(Catalog# : 185167, Cas# :
108852-90-0
)
Nemorubicin,又名PNU152243A,是一种不同于其母体药物的doxorubicin衍生
Nolatrexed盐酸盐
(Catalog# : 185166, Cas# :
152946-68-4
)
Nolatrexed,也叫AG337,是一种具有潜在抗癌活性的胸腺嘧啶合成酶抑
Nucleozin
(Catalog# : 185164, Cas# :
341001-38-5
)
Nucleozin是一种杀毒剂。它的目标是一种核蛋白(NP),这是一种病毒
Nidufexor
(Catalog# : 184288, Cas# :
1773489-72-7
)
Nidufexor是一个法呢醇X受体(FXR)激动剂。
1NM-PP1
(Catalog# : 184174, Cas# :
221244-14-0
)
1NM-PP1 是一种有效的突变激酶抑制剂。
Netarsudil(Mesylate)
(Catalog# : 712181, Cas# :
1422144-42-0
)
Netarsudil( AR-11324) is a Rho-associated protein kinase inhibitor. Netarsudil is pot
nor-NOHA醋酸盐
(Catalog# : 1710169, Cas# :
1140844-63-8
)
nor-NOHA是一种强效、选择性、竞争性、以及精氨酸酶的高亲和力抑
NMS-P118
(Catalog# : 17101311, Cas# :
1262417-51-5
)
NMS-P118是一种有效的、可口服、高选择性PARP-1抑制剂具有优良的AD
盐酸萘替芬
(Catalog# : 1791514, Cas# :
65473-14-5
)
萘替芬是一种丙烯胺抗真菌药物的局部治疗足癣、股癣、体癣(真
Neflamapimod
(Catalog# : 1791317, Cas# :
209410-46-8
)
Neflamapimod,也称为VX-745,VRT-031745和VD-31745,是高度有效的和选择性
盐酸纳洛酮
(Catalog# : 178305, Cas# :
357-08-4
)
纳洛酮是一种μ-opioid受体(MOR)逆受体激动剂。纳洛酮针对在中枢神
3-Nitrosalicylic Acid Methyl Ester
(Catalog# : 178224, Cas# :
22621-41-6
)
3-Nitrosalicylic Acid Methyl Ester
N-甲氧基-N-甲基乙酰胺
(Catalog# : 178223, Cas# :
78191-00-1
)
N-Methoxy-N-methylacetamide
N-(4-(benzyloxy)-3-methoxybenzyl)-5-phenyl-N-(2-(pyridin-2-yl)ethyl)pentanamide
(Catalog# : 1781506, Cas# :
521310-51-0
)
N-(4-(Benzyloxy)-3-methoxybenzyl)-5-phenyl-N-(2-(pyridin-2-yl)ethyl)pentanamide
NIH-12848
(Catalog# : 1781103, Cas# :
959551-10-1
)
NIH-12848是一种普遍认为的磷脂酰肌醇5 -磷酸四激酶(PI5P4K)抑制剂。
Nazartinib (EGF816)
(Catalog# : 1781004, Cas# :
1508250-71-2
)
Nazartinib,也被称为EGF816,是一种口服可用,不可逆转的、第三代、
Netarsudil
(Catalog# : 1781001, Cas# :
1254032-66-0
)
<span style="color:#34495E;font-family:" font-size:14px;background-color
NSC781406
(Catalog# : 20178810, Cas# :
1676893-24-5
)
NSC781406是一种高效针对PI3K的IC50为2 nM的PI3K和mTOR抑制剂。
NCT-503
(Catalog# : 2017888, Cas# :
1916571-90-8
)
NCT-503是一种3 -磷酸甘油酸脱氢酶(PHGDH)抑制剂,抑制丝氨酸合成3 -磷
NGP-555
(Catalog# : 2017875, Cas# :
1304630-27-0
)
NGP 555正在被作为一种预防疾病老年痴呆症的治疗。
N-反式-阿魏酰酪胺
(Catalog# : 201708019, Cas# :
66648-43-9
)
N-反式-阿魏酰酪胺|N-Trans-Feruloyltyramine|(E)-3-(4-hydroxy-3-Methoxy-phenyl)-
NDGA
(Catalog# : 17030909, Cas# :
500-38-9
)
去甲二氢愈创木酸(NDGA),也被称为masoprocol,是一种天然抗氧化剂dica
诺拉曲特
(Catalog# : 17030908, Cas# :
147149-76-6
)
诺拉曲特,也叫AG337,是一种具有潜在抗癌活性的百里香酶抑制剂
NPS-1034
(Catalog# : 17030907, Cas# :
1221713-92-3
)
NPS-1034是一种新型的MET抑制剂,它能抑制活化的MET受体及其具有结
NVP-BEP800
(Catalog# : 17030906, Cas# :
847559-80-2
)
NVP-BEP800, 也称为BEP-800,是一种新型的、完全合成的口服生物可用抑
制霉菌素
(Catalog# : 17030905, Cas# :
1400-61-9
)
制霉菌素是一种多烯抗真菌药物,含有三种生物活性成分的抗生素
NCH-51
(Catalog# : 17030716, Cas# :
848354-66-5
)
NCH-51, 也叫PTACH,是一种组蛋白去乙酰化酶(HDAC)抑制剂。NCH-51抑制
NS-1643
(Catalog# : 17030715, Cas# :
448895-37-2
)
NS-1643是一种人类ether-a-go-go相关基因(hERG)KV11.1通道激活剂(EC50 = 10.
Nifenalol HCl
(Catalog# : 17030705, Cas# :
5704-60-9
)
Nifenalol,也叫INPEA,是一种新型的β-肾上腺素受体拮抗剂。
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Dencatistat (STP938)
(Catalog# : 25177, Cas# :
2377000-84-3
)
Dencatistat 是一种口服生物可利用的小分子胞苷三磷酸合酶 1 (CTPS1)
DS-1001b
(Catalog# : 25178, Cas# :
1898207-64-1
)
DS-1001 是一种口服的脑渗透性突变 IDH1 选择性抑制剂。
Z57346765
(Catalog# : 25191, Cas# :
1016340-64-9
)
Z57346765 是一种 PGK1 特异性抑制剂,可降低 PGK1 糖酵解中代谢酶的
CBR-470-1
(Catalog# : 25192, Cas# :
2416095-06-0
)
CBR-470-1 是诱导 Nrf2 活性的糖酵解酶 PGK1 的抑制剂。
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
HC-7366
(Catalog# : 25076, Cas# :
2803470-63-3
)
HC-7366 is a potent and selective activator of the general control nonderepressible 2
Flavopiridol ( 夫拉平度 )
(Catalog# : 237071, Cas# :
146426-40-6
)
Alvocidib is a synthetic dihydroxyflavone that is 5,7-dihydroxyflavone which is subst
AG-270
(Catalog# : 25176, Cas# :
2201056-66-6
)
MAT2A 抑制剂 AG-270 是一种口服的蛋氨酸腺苷转移酶 II α (MAT2A) 小分
AZD-5904
(Catalog# : 181121, Cas# :
618913-30-7
)
AZD5904是一个有效的口服生物利用率MPO抑制剂。在临床前研究中,AZ
ALT-007
(Catalog# : 25157, Cas# :
2035010-37-6
)
ALT-007 是一种口服生物可利用的 SPT 抑制剂,比多球菌素更有效,