武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
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分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
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Chiral Compounds
Deuterated
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Iodos
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Oxazoles
Peg Linkers
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Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
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Other Heterocycles
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On Sale
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产品名字索引 L
LAU159
(Catalog# : 2071505, Cas# :
2055050-87-6
)
LAU159 is a potent modulator of α6β3γ2 GABAA receptor.
Lificiguat
(Catalog# : 2071502, Cas# :
170632-47-0
)
Lificiguat, also known as YC-1, is a inhibitor of Hypoxia-inducible factor-1alpha (HI
Lanraplenib
(Catalog# : 20732, Cas# :
1800046-95-0
)
GS-9876(lanraplenib)是一种高度选择性的口服SYK抑制剂,主要用于狼
Linperlisib free base
(Catalog# : 2061309, Cas# :
1702816-75-8
)
Linperlisib, also known as YY-20394 and PI3Kδ-IN-2, is a potent and selective PI3Kδ
L006235
(Catalog# : 2061307, Cas# :
294623-49-7
)
L006235 is a potent, reversible cathepsin K inhibitor (IC50 = 0.25 nM) that displays
LML-134
(Catalog# : 2051510, Cas# :
1542135-76-1
)
LML134 是一种具有口服活性,高选择性 H3R (组胺 3 受体) 反向激动剂
LUT-014
(Catalog# : 2042701, Cas# :
2274819-46-2
)
LUT-014 is a B-Raf Inhibitor. Leveraging the paradoxical effect of B-Raf Inhibitors,
LSZ102
(Catalog# : 2041502, Cas# :
2135600-76-7
)
LSZ102 is a potent ERα antagonist and degrader. LSZ102 showed ERα degradation IC50
LUN42589
(Catalog# : 204502, Cas# :
1848242-58-9
)
LUN42589,也称为PI3K / mTOR抑制剂2,是一种有效的双重pan-PI3K / mTOR抑
Lerociclib
(Catalog# : 204302, Cas# :
1628256-23-4 (free base)
)
Lerociclib,也称为G1T38,是一种口服,有效和选择性的CDK4 / 6抑制剂
Lemborexant (E-2006)
(Catalog# : 6111904, Cas# :
1369764-02-2
)
Lemborexant( E-2006, CAS 1369764-02-2)是食欲素OX 1和OX 2受体的双重拮抗
LY2794193
(Catalog# : 193262, Cas# :
2173037-97-1
)
LY2794193是一种高效选择性的mGlu3受体激动剂。
LY-3381916
(Catalog# : 193123, Cas# :
2166616-75-5
)
LY-3381916是一种强效的、选择性的、脑透性的IDO1活性抑制剂,与缺
LR-90
(Catalog# : 19364, Cas# :
245075-84-7
)
LR-90是一种晚期糖基化终产物(AGE)抑制剂,可抑制人单核细胞的炎
LCL521
(Catalog# : 19357, Cas# :
1226851-11-1
)
LCL521是一种酸性神经酰胺酶(ACDase)抑制剂。LCL521还抑制溶酶体酸鞘
Larotaxel
(Catalog# : 1922710, Cas# :
156294-36-9
)
Larotaxel是紫杉烷10-脱乙酰巴卡丁III的半合成衍生物,具有潜在的抗
Leniolisib
(Catalog# : 192271, Cas# :
1354690-24-6
)
Leniolisib,又名CDZ173,是一种有效的磷脂酰肌醇3激酶抑制剂(PI3K抑
Leuprolide Acetate
(Catalog# : 192261, Cas# :
74381-53-6
)
Leuprolide Acetate是一种合成的类似促性腺激素释放激素的非肽类似物
LOXO-292
(Catalog# : 192195, Cas# :
2222755-14-6
)
LOXO-292 (ARRY-192)是一种口服和临床开发的选择性研究药物,用于治
Lexibulin
(Catalog# : 19122, Cas# :
917111-49-0
)
Lexibulin,又称CYT997,是一种n型口服生物利用小分子,具有管蛋白
LP-211
(Catalog# : 1811302, Cas# :
1052147-86-0
)
LP-211是血清素5-HT7受体的选择性激动剂。
LXH254游离
(Catalog# : 1811213, Cas# :
1800398-38-2
)
LXH254是所有丝氨酸/苏氨酸蛋白激酶Raf家族成员的口服有效抑制剂
LY2828360
(Catalog# : 181172, Cas# :
1231220-79-3
)
LY2828360是一种新的有效的、选择性的、有效的CB2激动剂。
LP-533401盐酸盐
(Catalog# : 1810262, Cas# :
1040526-12-2
)
LP-533401 HCl是色氨酸羟化酶-1 (Tph-1)的抑制剂,Tph-1是内脏衍生血清
LP-922761
(Catalog# : 188101, Cas# :
1454808-95-7
)
LP-922761是一种强有力的和选择性AAK1抑制剂,在体外的IC50值为4.8±
LM22B-10
(Catalog# : 187165, Cas# :
342777-54-2
)
LM22B-10是TrkB和TrkC激动剂。LM22B-10表现为神经营养活性(EC50 = 200- 300
LY-3200882
(Catalog# : 186278, Cas# :
1898283-02-7
)
LY-3200882是一种口服TGFbeta抑制剂。LY3200882目标转化生长因子-beta (T
LX2761
(Catalog# : 186275, Cas# :
1610954-97-6
)
LX2761是一种局部作用的SGLT1抑制剂,体外强效,延缓体内肠道葡萄
L685458
(Catalog# : 186156, Cas# :
292632-98-5
)
L685458是一个强有力的和选择性γ分泌酶抑制剂。
Lometrexol disodium
(Catalog# : 186151, Cas# :
120408-07-3
)
Lometrexol是一种具有抗肿瘤活性的叶酸模拟抗代谢产物。
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Kartogenin ( KGN )
(Catalog# : 52215, Cas# :
4727-31-5
)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602, Cas# :
218791-21-0
)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
Apecotrep (BI 764198)
(Catalog# : 26A048, Cas# :
2311863-36-0
)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
BH-30643
(Catalog# : 26A047, Cas# :
3062177-59-4
)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制
Gridegalutamide
(Catalog# : 26A044, Cas# :
2446929-86-6
)
格列德加鲁胺是一种具有口服生物利用度的雄激素受体(AR)降解
BMS-986365 (别名: CC-94676 )
(Catalog# : 25138, Cas# :
2446928-30-7
)
BMS-986365,也称为 CC-94676,是一种口服生物可利用的雄激素受体 (A
CBR-5884
(Catalog# : 24109, Cas# :
681159-27-3
)
CBR 5884 是一种磷酸甘油酸脱氢酶 (PHGDH) 抑制剂,能够抑制过度表达
JHU-083
(Catalog# : 24108, Cas# :
1998725-11-3
)
JHU-083 选择性阻断大脑 CD11b+ 细胞中的谷氨酰胺酶活性,并防止慢
VAS3947
(Catalog# : 20302, Cas# :
869853-70-3
)
VAS3947是一种低微摩尔浓度的NADPH氧化酶活性的选择性抑制剂,既不