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首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
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产品名字索引 C
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产品名字索引 C
卡米诺霉素盐酸盐
(Catalog# : 17914, Cas# :
52794-97-5
)
卡米诺霉素盐酸盐是一种蒽环类抗肿瘤抗生素类的洋红色马杜拉细
Cambinol
(Catalog# : 178313, Cas# :
14513-15-6
)
Cambinol是一种SIRT抑制剂。它能抑制促炎性细胞因子的表达,提高模
2-氯-4-(甲基氨基)-5-嘧啶甲醛
(Catalog# : 1781601, Cas# :
839708-50-8
)
2-氯-4-(甲基氨基)-5-嘧啶甲醛;2-chloro-4-(methylamino) pyrimidine-5-carbaldeh
2-吗啉-4-基-6-噻蒽-1-基吡喃-4-酮
(Catalog# : 1781504, Cas# :
119671-47-5
)
2-吗啉-4-基-6-噻蒽-1-基吡喃-4-酮;2-Chloro-6-morpholinopyran-4-one
CCT196969
(Catalog# : 178913, Cas# :
1163719-56-9
)
CCT196969,是一种pan-RAF / SFK抑制剂对治疗单纯的BRAF和NRAS突变型黑色
CCT365623
(Catalog# : 2017876)
CCT365623是一种赖氨酰化氧抑制剂。
CM-579
(Catalog# : 2017874, Cas# :
1846570-40-8
)
CM-579是一种生物活性化学药品 。
C188-9
(Catalog# : 2017873, Cas# :
432001-19-9
)
C188-9是一种生物活性化学品。
5-氯-2-氰基苯硼酸
(Catalog# : 20178120, Cas# :
1072946-52-1
)
5-氯-2-氰基苯硼酸
CY5.5-SE
(Catalog# : 20177314, Cas# :
442912-55-2
)
2-[5-[3-[6-[(2,5-Dioxo-1-pyrrolidinyl)oxy]-6-oxohexyl]-1,3-dihydro-1,1-dimethyl-6,8-d
头孢曲松钠
(Catalog# : 17032406, Cas# :
73384-59-5
)
头孢曲松是一种用于治疗多种细菌感染的抗生素。
头孢布烯
(Catalog# : 17032405, Cas# :
97519-39-6
)
头孢布烯(Sch39720)是第三代头孢菌素类抗生素。
头孢他啶
(Catalog# : 17032404, Cas# :
72558-82-8
)
头孢他啶(GR20263)是一种用于治疗多种细菌感染的抗生素。
头孢拉定
(Catalog# : 17032403, Cas# :
38821-53-3
)
头孢拉定是第一代头孢菌素类抗生素。
头孢唑兰
(Catalog# : 17032402, Cas# :
113359-04-9
)
头孢唑兰(SCE 2787)是第四代头孢菌素。
头孢噻利
(Catalog# : 17032401, Cas# :
122841-10-5
)
头孢噻利是一种广泛使用于β-内酰胺的抗生素。
CC-122
(Catalog# : 17030313, Cas# :
1015474-32-4
)
CC-122是一种具有潜在抗肿瘤活性的多向性通路调制器。
CP21R7
(Catalog# : 17022715, Cas# :
125314-13-8
)
CP21R7,也称CP21,是一个强有力的和选择性GSK-3β抑制剂。
Citarinostat
(Catalog# : 17022701, Cas# :
1316215-12-9
)
Citarinostat是一种HDAC6特异性抑制剂,HDAC6和HDAC3的IC50分别为4nM和76
(±)-樟脑
(Catalog# : 17021401, Cas# :
464-49-3
)
(±)-樟脑是烹饪中的一种成分,作为一种用于医药用途的防腐液体
CeMMEC1
(Catalog# : 17021308, Cas# :
440662-09-9
)
CeMMEC1是N-methylisoquinolinone导数,抑制第二溴域 TAF1(IC50 = 0.9μM)。
CA-074 methyl ester (CA-074 Me)
(Catalog# : 17011104, Cas# :
147859-80-1
)
CA-074 Me是CA- 074的一种膜-渗透性衍生物,作为一种不可逆转的蛋白
CZ415
(Catalog# : 17011101, Cas# :
1429639-50-8
)
CZ415,是一种有效的ATP-竞争性mTOR抑制剂,拥有非常好的细胞渗透率
CPI-455
(Catalog# : 17109005, Cas# :
1628208-23-0
)
CPI-455是一种特殊的KDM5抑制剂,提高了H3K4三甲基化(H3K4me3)的全球水
Cytosporone B
(Catalog# : 16122924, Cas# :
321661-62-5
)
Cytosporone B is the first naturally occurring agonist for nuclear orphan receptor Nu
CVT-313
(Catalog# : 16122923, Cas# :
199986-75-9
)
CVT-313 is a potent and selective inhibitor of CDK2 that prevents neointimal prolifer
CTP354
(Catalog# : 16122922, Cas# :
1213669-91-0
)
CTP354, also known as C-21191, a novel deuterated subtype-selective GABA(A) modulator
Ciliobrevin A
(Catalog# : 16122921, Cas# :
302803-72-1
)
Ciliobrevin A, also known as HPI-4 and Hedgehog Pathway Inhibitor 4, is a Hedgehog pa
CID5721353
(Catalog# : 16122920, Cas# :
301356-95-6
)
CID5721353 is a B-Cell Lymphoma 6 Inhibitor (BCL6 inhibitor).
Cetilistat
(Catalog# : 16122918, Cas# :
282526-98-1
)
Cetilistat, also known as ATL-962, is a drug designed to treat obesity. It acts in th
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
ECI830
(Catalog# : 26A031, Cas# :
3054692-62-2
)
ECI830是一种实验性的CDK2抑制剂。
GNE-317
(Catalog# : 52282, Cas# :
1394076-92-6
)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
DPTX-3186
(Catalog# : 26A010, Cas# :
3118994-80-9
)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108, Cas# :
435327-40-5
)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
Iclepertin (BI-425809)
(Catalog# : 24084, Cas# :
1421936-85-7
)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
Kartogenin ( KGN )
(Catalog# : 52215, Cas# :
4727-31-5
)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602, Cas# :
218791-21-0
)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
Apecotrep (BI 764198)
(Catalog# : 26A048, Cas# :
2311863-36-0
)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
BH-30643
(Catalog# : 26A047, Cas# :
3062177-59-4
)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制