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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
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Amino Acids
Anilines
Boronic Acids
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Deuterated
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Pyrimidines
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产品名字索引 C
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产品名字索引 C
CM-579
(Catalog# : 2017874, Cas# :
1846570-40-8
)
CM-579是一种生物活性化学药品 。
C188-9
(Catalog# : 2017873, Cas# :
432001-19-9
)
C188-9是一种生物活性化学品。
5-氯-2-氰基苯硼酸
(Catalog# : 20178120, Cas# :
1072946-52-1
)
5-氯-2-氰基苯硼酸
CY5.5-SE
(Catalog# : 20177314, Cas# :
442912-55-2
)
2-[5-[3-[6-[(2,5-Dioxo-1-pyrrolidinyl)oxy]-6-oxohexyl]-1,3-dihydro-1,1-dimethyl-6,8-d
头孢曲松钠
(Catalog# : 17032406, Cas# :
73384-59-5
)
头孢曲松是一种用于治疗多种细菌感染的抗生素。
头孢布烯
(Catalog# : 17032405, Cas# :
97519-39-6
)
头孢布烯(Sch39720)是第三代头孢菌素类抗生素。
头孢他啶
(Catalog# : 17032404, Cas# :
72558-82-8
)
头孢他啶(GR20263)是一种用于治疗多种细菌感染的抗生素。
头孢拉定
(Catalog# : 17032403, Cas# :
38821-53-3
)
头孢拉定是第一代头孢菌素类抗生素。
头孢唑兰
(Catalog# : 17032402, Cas# :
113359-04-9
)
头孢唑兰(SCE 2787)是第四代头孢菌素。
头孢噻利
(Catalog# : 17032401, Cas# :
122841-10-5
)
头孢噻利是一种广泛使用于β-内酰胺的抗生素。
CC-122
(Catalog# : 17030313, Cas# :
1015474-32-4
)
CC-122是一种具有潜在抗肿瘤活性的多向性通路调制器。
CP21R7
(Catalog# : 17022715, Cas# :
125314-13-8
)
CP21R7,也称CP21,是一个强有力的和选择性GSK-3β抑制剂。
Citarinostat
(Catalog# : 17022701, Cas# :
1316215-12-9
)
Citarinostat是一种HDAC6特异性抑制剂,HDAC6和HDAC3的IC50分别为4nM和76
(±)-樟脑
(Catalog# : 17021401, Cas# :
464-49-3
)
(±)-樟脑是烹饪中的一种成分,作为一种用于医药用途的防腐液体
CeMMEC1
(Catalog# : 17021308, Cas# :
440662-09-9
)
CeMMEC1是N-methylisoquinolinone导数,抑制第二溴域 TAF1(IC50 = 0.9μM)。
CA-074 methyl ester (CA-074 Me)
(Catalog# : 17011104, Cas# :
147859-80-1
)
CA-074 Me是CA- 074的一种膜-渗透性衍生物,作为一种不可逆转的蛋白
CZ415
(Catalog# : 17011101, Cas# :
1429639-50-8
)
CZ415,是一种有效的ATP-竞争性mTOR抑制剂,拥有非常好的细胞渗透率
CPI-455
(Catalog# : 17109005, Cas# :
1628208-23-0
)
CPI-455是一种特殊的KDM5抑制剂,提高了H3K4三甲基化(H3K4me3)的全球水
Cytosporone B
(Catalog# : 16122924, Cas# :
321661-62-5
)
Cytosporone B is the first naturally occurring agonist for nuclear orphan receptor Nu
CVT-313
(Catalog# : 16122923, Cas# :
199986-75-9
)
CVT-313 is a potent and selective inhibitor of CDK2 that prevents neointimal prolifer
CTP354
(Catalog# : 16122922, Cas# :
1213669-91-0
)
CTP354, also known as C-21191, a novel deuterated subtype-selective GABA(A) modulator
Ciliobrevin A
(Catalog# : 16122921, Cas# :
302803-72-1
)
Ciliobrevin A, also known as HPI-4 and Hedgehog Pathway Inhibitor 4, is a Hedgehog pa
CID5721353
(Catalog# : 16122920, Cas# :
301356-95-6
)
CID5721353 is a B-Cell Lymphoma 6 Inhibitor (BCL6 inhibitor).
Cetilistat
(Catalog# : 16122918, Cas# :
282526-98-1
)
Cetilistat, also known as ATL-962, is a drug designed to treat obesity. It acts in th
Cerdulatinib (PRT062070)
(Catalog# : 16122917, Cas# :
1198300-79-6
)
Cerdulatinib, also known as PRT2070 and PRT062070, is a n ovel, oral, dual spleen tyr
Cefotetan Sodium
(Catalog# : 16122916, Cas# :
74356-00-6
)
Cefotetan Sodium, also known as ICI-156834 and YM-09330, is a second-generation cepha
C-DIM12
(Catalog# : 16122915, Cas# :
178946-89-9
)
C-DIM12 is a novel synthetic activator of Nurr1. C-DIM12 induces dopaminergic gene ex
CCG215022
(Catalog# : 16122914, Cas# :
1813527-81-9
)
CCG215022 is a potent GRK2 and GRK5 inhibitor. CCG215022 exhibited nanomolar IC50 val
CB-839
(Catalog# : 16122913, Cas# :
1439399-58-2
)
CB-839 an is orally bioavailable inhibitor of glutaminase, with potential antineoplas
CAY10683
(Catalog# : 16122912, Cas# :
1477949-42-0
)
CAY10683, also known as Santacruzamate A, is a potent and selective histone deacetyla
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AZD0095
(Catalog# : 237072, Cas# :
2750001-23-9
)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2-MNG
(Catalog# : 24129, Cas# :
2101538-28-5
)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
MAT2A-IN-9
(Catalog# : 25147, Cas# :
2439277-80-0
)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
Acoramidis hydrochloride
(Catalog# : 24068, Cas# :
2242751-53-5
)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
Crelosidenib
(Catalog# : 24101, Cas# :
2230263-60-0
)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
LOXO-435
(Catalog# : 25080, Cas# :
2833703-74-3
)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
Gridegalutamide
(Catalog# : 25138, Cas# :
2446928-30-7
)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
Chiauranib
(Catalog# : 25146, Cas# :
1256349-48-0
)
Chiauranib also known as orally available, small molecule inhibitor of select serine-