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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
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产品名字索引 C
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产品名字索引 C
CAY10602
(Catalog# : 191285, Cas# :
374922-43-7
)
CAY10602是SIRT1激活剂。CAY10602是通过高通量筛选增加sirt1介导的特定
Cilofexor ( GS-9674 )
(Catalog# : 19132, Cas# :
1418274-28-8
)
Cilofexor(也称为 GS-9674)是一种非甾体法尼醇 X 受体(FXR)激动剂
CCT241736
(Catalog# : 1812283, Cas# :
1402709-93-6
)
CCT241736是一种有效且具有口服活性的日常FLT3-Aurora抑制剂。
CA-4948
(Catalog# : 1811292, Cas# :
1801343-74-7
)
CA-4948是一种生物活性化学物。
CCT129202
(Catalog# : 1810291, Cas# :
942947-93-5
)
CCT129202是Aurora激酶活性的抑制剂,在临床前研究中表现出良好的抗
CBM 301940
(Catalog# : 1810232, Cas# :
902146-11-6
)
CBM 301940是一种有效的丙二酰辅酶a脱羧酶抑制剂,具有口服生物有
CID16020046
(Catalog# : 1810225, Cas# :
834903-43-4
)
CID16020046是一种选择性GPR55逆激动剂。
10-Cl-BBQ
(Catalog# : 1810161, Cas# :
23982-76-5
)
10-Cl-BBQ是芳烃受体(AhR)配体。
CGP-71683A盐酸盐
(Catalog# : 18792, Cas# :
192322-50-2
)
CGP 71683A是一种有效且高选择性的NPY Y(5)受体的非肽拮抗剂,在肥胖
卡卢莫南钠
(Catalog# : 18752, Cas# :
86832-68-0
)
卡卢莫南钠,也被称为Amasulin和AMA-1080,是一种单异戊巴丁与青霉
CEP-40783
(Catalog# : 186281, Cas# :
1437321-24-8
)
CEP-40783,又称RXDX-106,是AXL和c-Met的一种有效、选择性和口服的抑
CD437
(Catalog# : 185316, Cas# :
125316-60-1
)
CD437合成维生素a是一个RARγ-selective受体激动剂。
CB-1158
(Catalog# : 185315, Cas# :
1345810-21-0
)
CB-1158,又称INCB01158,是一种有效的精氨酸酶抑制剂。
西洛司特
(Catalog# : 185291, Cas# :
153259-65-5
)
西洛司特是一种用于治疗呼吸系统疾病,如哮喘和慢性阻塞性肺病
CNX-1351
(Catalog# : 185174, Cas# :
1276105-89-5
)
CNX-1351是PI3K的选择性共价抑制剂。
CGP60474
(Catalog# : 185171, Cas# :
164658-13-3
)
CGP60474是一种有效的双cdk1/cdk2抑制剂(IC50值分别为20和50 nM)。
COH29
(Catalog# : 184127, Cas# :
1190932-38-7
)
COH29是一种可口服的、芳香的取代噻唑和人核糖核苷酸还原酶(RNR)
CIL56
(Catalog# : 18491, Cas# :
300802-28-2
)
CIL56是一种YAP1抑制剂。它的作用是诱导非凋亡细胞死亡,触发细胞
Casopitant甲磺酸盐
(Catalog# : 18444, Cas# :
414910-30-8
)
Casopitant甲磺酸盐是一种中枢作用的神经激肽(NK1)受体拮抗剂,具有
COTI-2
(Catalog# : 184320, Cas# :
1039455-84-9
)
COTI-2是P53基因调制器和AKT2抑制剂。OTI-2在体外和体内都对多种人类
CBL0137
(Catalog# : 184319, Cas# :
314761-14-3
)
CBL0137激活p53并抑制NF-kB,它还能抑制组蛋白分子伴侣FACT,FACT促进染
CPI-444
(Catalog# : 18439, Cas# :
1202402-40-1
)
CPI-444,又名V81444,是一种腺苷A2A受体的口服拮抗剂。
CCG-203971
(Catalog# : 18437, Cas# :
1443437-74-8
)
CCG-203971是前列腺癌细胞系PC-3中SRE活化的抑制剂(IC50 = 6.4 μM),能够
CP-376395 free base
(Catalog# : 184213, Cas# :
175140-00-8
)
CP-376395 is a CRF1-selective antagonist. CRF1 receptor signaling regulates food and
Copanlisib HCl
(Catalog# : 18351, Cas# :
1402152-13-9
)
Copanlisib也称为BAY 80 - 6946,是一个强有力的磷酸肌醇3-激酶(PI3K)抑制
CB-03-01
(Catalog# : 1712153, Cas# :
19608-29-8
)
CB-03-01, also known as cortexolone 17alpha-propionate, is a topical and peripherally
Cenicriviroc ( TAK-652 )
(Catalog# : S510902, Cas# :
497223-25-3
)
Cenicriviroc(TAK-652, TBR-652) 是一种CCR2和CCR5受体抑制剂,临床上它被用
CHIR99021 HCl
(Catalog# : 179825, Cas# :
1797989-42-4
)
CHIR99021,又被称为 CT99021,是糖原合成酶激酶3β(GSK3β)抑制剂,
CDDO
(Catalog# : 92304, Cas# :
218600-44-3
)
CDDO是一种合成的齐墩果烷型三萜阻断诱导型一氧化氮合酶和诱导
CVT-10216
(Catalog# : 179818, Cas# :
1005334-57-5
)
CVT-10216是强有力的和有选择性的,乙醛脱氢酶2(ALDH2)的可逆性抑
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
ECI830
(Catalog# : 26A031, Cas# :
3054692-62-2
)
ECI830是一种实验性的CDK2抑制剂。
GNE-317
(Catalog# : 52282, Cas# :
1394076-92-6
)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
DPTX-3186
(Catalog# : 26A010, Cas# :
3118994-80-9
)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108, Cas# :
435327-40-5
)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
Iclepertin (BI-425809)
(Catalog# : 24084, Cas# :
1421936-85-7
)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
Kartogenin ( KGN )
(Catalog# : 52215, Cas# :
4727-31-5
)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602, Cas# :
218791-21-0
)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
Apecotrep (BI 764198)
(Catalog# : 26A048, Cas# :
2311863-36-0
)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
BH-30643
(Catalog# : 26A047, Cas# :
3062177-59-4
)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制