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Cytoskeletal Signaling
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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
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Boronic Acids
Bromides
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Chiral Compounds
Deuterated
Fluorides
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Nitro Compounds
Oxazoles
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Piperidines
Pyridines
Pyrimidines
Quinolines
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Trifluoroborates
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订购信息
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产品名字索引 C
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产品名字索引 C
4-氯-6-三氟甲基喹唑啉
(Catalog# : 20310, Cas# :
16499-64-2
)
4-氯甲基-1-环戊基-2-三氟甲基苯
(Catalog# : 20308, Cas# :
957208-65-0
)
1-cyanocyclohexyl 4-methylbenzenesulfonate
(Catalog# : 21075, Cas# :
90775-01-2
)
1-cyanocyclohexyl 4-methylbenzenesulfonate (CAS 90775-01-2 ) 是有机合成反应中
Caroverine HCl
(Catalog# : 20260, Cas# :
55750-05-5
)
Caroverine HCl is a nonselective NMDA and AMPA glutamate receptor antagonist, also ac
CRT0273750
(Catalog# : 20258, Cas# :
1979939-16-6
)
CRT0273750 modulates LPA levels in plasma and is suitable for in vivo studies.
Centanafadine ( free base )
(Catalog# : 21237, Cas# :
924012-43-1
)
Centanafadine (free base) is a dual norepinephrine-dopamine transporter inhibitor use
Centanafadine HCl
(Catalog# : 21236, Cas# :
923981-14-0
)
Centanafadine, also known as EB-1020, is an adrenergic uptake inhibitor and dopamine
CB-6644
(Catalog# : 41788, Cas# :
2316817-88-4
)
CB-6644 acts as a noncompetitive ATPase inhibitor. Additionally, it can inhibit RUVBL
Coralyne chloride
(Catalog# : 20111601, Cas# :
38989-38-7
)
Coralyne chloride is a a protoberberine alkaloid, can be used as a fluorescent DNA-ba
4-chloro-1H-pyrrolo[2,3-b]pyridine-5-carbaldehyde
(Catalog# : 20103005, Cas# :
958230-19-8
)
5-(chloromethyl)-1-propyl-1H-imidazole hydrochloride
(Catalog# : 2091502, Cas# :
497223-15-1
)
5-(chloromethyl)-1-propyl-1H-imidazole hydrochloride 是合成 Cenicriviroc ( TAK-652
2-氯-4-(4-氟苯基)-5-噻唑甲腈
(Catalog# : 2091202, Cas# :
1628265-17-7
)
CL2A-SN38 DCA
(Catalog# : 2071556, Cas# :
1279680-68-0
)
CL2A-SN38 is a SN38 derivative with a peptide-linker which can easily react with anti
Cariprazine HCl
(Catalog# : 2071544, Cas# :
839712-12-8
)
Cariprazine, also known as RGH-188 and MP-214, is an antipsychotic drug received FDA
CM-272
(Catalog# : 2071538, Cas# :
1846570-31-7
)
CM-272 is a first-in-class reversible dual small molecule inhibitor against G9a and D
2-Cyano-4-fluorobenzaldehyde
(Catalog# : 2062317, Cas# :
77532-90-2
)
3-chloro-1-benzothiophene-2-carbonyl chloride
(Catalog# : 2062306, Cas# :
21815-91-8
)
Carbamic acid,N-[(7S)-20-[[[(4-fluorophenyl)methyl]amino]carbonyl]-8-oxo-2,9,16,18,21-pentaazabicyclo[15.3.1]heneicosa-1(21),17,19-trien-7-yl]-, 1,1-dimethylethyl ester
(Catalog# : 2062029, Cas# :
2092998-71-3
)
5-chloro-2,6-dimethoxy-4-methyl-8-nitroquinoline
(Catalog# : 2062026, Cas# :
189746-21-2
)
4-(3-Chloro-2-fluoroanilino)-6-hydroxy-7-methoxyquinazoline
(Catalog# : 2062022, Cas# :
612501-52-7
)
2-chloro-6-methoxy-4-methylquinoline
(Catalog# : 2062014, Cas# :
6340-55-2
)
CaCCinh-A01
(Catalog# : 2061702, Cas# :
407587-33-1
)
CaCCinh-A01, also known as TMEM16 Blocker I, is a TMEM16 Blocker. CaCCinh-A01 is a no
CLEFMA
(Catalog# : 615201, Cas# :
1246964-32-8
)
CLEFMA has anti-proliferative activity in H441 cells. CLEFMA may induce autophagic ce
CMPD1
(Catalog# : 2061307, Cas# :
41179-33-3
)
CMPD1 is an inhibitor of MK2 activation, primarily inhibiting tubulin polymerisation
CGP52411
(Catalog# : 2061306, Cas# :
145915-58-8
)
CGP52411, also known as DAPH, is a selective inhibitor of the epidermal growth factor
CADD522
(Catalog# : 2051505, Cas# :
199735-88-1
)
CADD522 is a potent inhibitor of runt-related transcription factor-2 (RUNX2)-DNA bind
2-氯-7-氟喹啉-3-甲醛
(Catalog# : S-204160, Cas# :
745830-16-4
)
铜色树碱
(Catalog# : S-203042, Cas# :
524-63-0
)
CC-885
(Catalog# : 2041501, Cas# :
1010100-07-8
)
CC-885 is a potent Cereblon Modulator with potent antitumor activity mediated through
CM4620
(Catalog# : 204504, Cas# :
1713240-67-5
)
CM4620是一种选择性的Orai1抑制剂,可防止Ca2 +进入腺泡细胞。CM4620
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
PLX8394
(Catalog# : 20613, Cas# :
1393466-87-9
)
PLX8394 is an orally bioavailable inhibitor of serine/threonine-protein kinase B-raf
Zelasudil
(Catalog# : 24014, Cas# :
2365193-22-0
)
Zelasudil 是一种有效的、高选择性的口服活性抑制剂,针对 Rho 相关
Ziftomenib ( KO-539 )
(Catalog# : 24013, Cas# :
2134675-36-6
)
Ziftomenib 是一种口服、有效、选择性的小分子抑制剂,针对 menin 和
Zunsemetinib
(Catalog# : 24012, Cas# :
1640282-42-3
)
Zunsemetinib是一种在研口服丝裂原活化蛋白激酶活化蛋白激酶2(MK2
Zongertinib ( BI 1810631 )
(Catalog# : 24011, Cas# :
2728667-27-2
)
Zongertinib [BI 1810631] 是一种人表皮生长因子受体 2 (HER2) 抑制剂。
Zasocitinib
(Catalog# : 24010, Cas# :
2272904-53-5
)
Zasocitinib是一种作用于非受体酪氨酸蛋白激酶 (TYK2)靶点的抑制
RNK-05047
(Catalog# : 24008, Cas# :
2503036-46-0
)
RNK-05047 为BRD4降解剂,其在小鼠荷瘤异种移植模型中展现出显著抑
Asengeprast (FT011)
(Catalog# : 24009, Cas# :
1001288-58-9
)
Asengeprast (FT011) 是一种抗纤维化剂,降低胶原蛋白 I 和 III 的 mRNA
ERAS-801 ( JGK-068S )
(Catalog# : 20635, Cas# :
2490431-16-6
)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。
T-1095
(Catalog# : 24004, Cas# :
209746-59-8
)
T-1095 is a potent and selective inhibitor of Na+-glucose cotransporters (SGLTs).