武汉永璨生物科技有限公司
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
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分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
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联系我们
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产品名字索引 C
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产品名字索引 C
CB-6644
(Catalog# : 41788, Cas# :
2316817-88-4
)
CB-6644 acts as a noncompetitive ATPase inhibitor. Additionally, it can inhibit RUVBL
Coralyne chloride
(Catalog# : 20111601, Cas# :
38989-38-7
)
Coralyne chloride is a a protoberberine alkaloid, can be used as a fluorescent DNA-ba
4-chloro-1H-pyrrolo[2,3-b]pyridine-5-carbaldehyde
(Catalog# : 20103005, Cas# :
958230-19-8
)
5-(chloromethyl)-1-propyl-1H-imidazole hydrochloride
(Catalog# : 2091502, Cas# :
497223-15-1
)
5-(chloromethyl)-1-propyl-1H-imidazole hydrochloride 是合成 Cenicriviroc ( TAK-652
2-氯-4-(4-氟苯基)-5-噻唑甲腈
(Catalog# : 2091202, Cas# :
1628265-17-7
)
CL2A-SN38 DCA
(Catalog# : 2071556, Cas# :
1279680-68-0
)
CL2A-SN38 is a SN38 derivative with a peptide-linker which can easily react with anti
Cariprazine HCl
(Catalog# : 2071544, Cas# :
839712-12-8
)
Cariprazine, also known as RGH-188 and MP-214, is an antipsychotic drug received FDA
CM-272
(Catalog# : 2071538, Cas# :
1846570-31-7
)
CM-272 is a first-in-class reversible dual small molecule inhibitor against G9a and D
2-Cyano-4-fluorobenzaldehyde
(Catalog# : 2062317, Cas# :
77532-90-2
)
3-chloro-1-benzothiophene-2-carbonyl chloride
(Catalog# : 2062306, Cas# :
21815-91-8
)
5-chloro-2,6-dimethoxy-4-methyl-8-nitroquinoline
(Catalog# : 2062026, Cas# :
189746-21-2
)
4-(3-Chloro-2-fluoroanilino)-6-hydroxy-7-methoxyquinazoline
(Catalog# : 2062022, Cas# :
612501-52-7
)
2-chloro-6-methoxy-4-methylquinoline
(Catalog# : 2062014, Cas# :
6340-55-2
)
CaCCinh-A01
(Catalog# : 2061702, Cas# :
407587-33-1
)
CaCCinh-A01, also known as TMEM16 Blocker I, is a TMEM16 Blocker. CaCCinh-A01 is a no
CLEFMA
(Catalog# : 615201, Cas# :
1246964-32-8
)
CLEFMA has anti-proliferative activity in H441 cells. CLEFMA may induce autophagic ce
CMPD1
(Catalog# : 2061307, Cas# :
41179-33-3
)
CMPD1 is an inhibitor of MK2 activation, primarily inhibiting tubulin polymerisation
CGP52411
(Catalog# : 2061306, Cas# :
145915-58-8
)
CGP52411, also known as DAPH, is a selective inhibitor of the epidermal growth factor
CADD522
(Catalog# : 2051505, Cas# :
199735-88-1
)
CADD522 is a potent inhibitor of runt-related transcription factor-2 (RUNX2)-DNA bind
2-氯-7-氟喹啉-3-甲醛
(Catalog# : S-204160, Cas# :
745830-16-4
)
铜色树碱
(Catalog# : S-203042, Cas# :
524-63-0
)
CC-885
(Catalog# : 2041501, Cas# :
1010100-07-8
)
CC-885 is a potent Cereblon Modulator with potent antitumor activity mediated through
CC-90009
(Catalog# : 203071, Cas# :
1860875-51-9
)
CC-90009 是一种 cereblon (CRBN) E3 连接酶调节剂。CC-90009 与 CRBN 特异性
5-氯-2,6-二甲氧基-4-甲基喹啉
(Catalog# : 4281903, Cas# :
189746-19-8
)
5-氯-2,6-二甲氧基-4-甲基喹啉是一个他非诺喹原料药合成中非常关
Cenicriviroc Mesylate
(Catalog# : S510901, Cas# :
497223-28-6
)
Cenicriviroc(代号TAK-652,TBR-652)是用于治疗HIV感染的实验候选药物
CLP-290
(Catalog# : 193286, Cas# :
1181083-81-7
)
CLP-290是一种新型的KCC2调制器和CLP-257的前药,对KCC2相关的Cl-转运
氯非铵甲苯磺酸盐
(Catalog# : 193181, Cas# :
92953-10-1
)
氯非铵甲苯磺酸盐是一种K+通道阻滞剂、心脏抑制剂和抗心律失常
Cevipabulin fumarate
(Catalog# : 193124, Cas# :
849550-67-0
)
Cevipabulin fumarate (TTI-237 fumarate) 是一种口服活性微管活性抗肿瘤化
Conteltinib
(Catalog# : 19342, Cas# :
1384860-29-0
)
Conteltinib是一种酪氨酸激酶抑制剂和抗肿瘤药。
C25-140
(Catalog# : 192274, Cas# :
1358099-18-9
)
C25-140是环-E3连接酶(TRAF6) / E2酶(Ubc13)结合的一级蛋白-蛋白相互作用
CCT-137690
(Catalog# : 192192, Cas# :
1095382-05-0
)
CCT137690是一种极光激酶抑制剂CCT137690,是一种高选择性的口服生物
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive-Oxygen-Species-ROS
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Mitoquinol mesylate (MitoQ)
(Catalog# : 26A042, Cas# :
845959-55-9
)
Mitoquinol mesylate (MitoQ) 是一种线粒体靶向抗氧化剂,具体而言,它
SPG-601 ( VSN-16R )
(Catalog# : 24042, Cas# :
1246960-09-7
)
SPG-601(原名VSN-16R)是一种口服给药、同类首创的小分子药物,是
LY3039478 ( Crenigacestat )
(Catalog# : 17021601, Cas# :
1421438-81-4
)
LY3039478 ( Crenigacestat ) 是一种选择性 NOTCH1 抑制剂,通过阻断 VEGFA/
PF-9366
(Catalog# : 184107, Cas# :
72882-78-1
)
PF-9366是一种新型的人蛋氨酸腺苷转移酶2A (Mat2A),肝外同种型。
MAT2A-IN-22
(Catalog# : 26A021, Cas# :
2925330-18-1
)
MAT2A-IN-22 (Compound 29-1) 是一种可透过血脑屏障的和口服有效的 MAT2A
Pantothenate kinase-IN-3
(Catalog# : 26A041)
泛酸激酶-IN-3(亦称化合物21,https://doi.org/10.1021/acs.jmedchem.5c03452)
Claziprotamidum ( Claziprotamide ; BBP-671 )
(Catalog# : 26A040, Cas# :
2361124-03-8
)
Claziprotamidum(Claziprotamide;BBP-671)是一种强效、口服有效且能透过
PZ-3022
(Catalog# : 26A039, Cas# :
2170608-85-0
)
PZ-3022是一种别构型的PanK激活剂,能够抵消C3-CoA的抑制作用。
PZ-2891
(Catalog# : 193282, Cas# :
2170608-82-7
)
PZ-2891是一种强效的、选择性的、口服活性泛酸激酶(PANK)调制剂,
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,