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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
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Cas号索引 4
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Cas号索引 4
497223-15-1 | 5-(chloromethyl)-1-propyl-1H-imidazole hydrochloride
(Catalog# : 2091502)
5-(chloromethyl)-1-propyl-1H-imidazole hydrochloride 是合成 Cenicriviroc ( TAK-652
407587-33-1 | CaCCinh-A01
(Catalog# : 2061702)
CaCCinh-A01, also known as TMEM16 Blocker I, is a TMEM16 Blocker. CaCCinh-A01 is a no
41179-33-3 | CMPD1
(Catalog# : 2061307)
CMPD1 is an inhibitor of MK2 activation, primarily inhibiting tubulin polymerisation
497223-28-6 | Cenicriviroc Mesylate
(Catalog# : S510901)
Cenicriviroc(代号TAK-652,TBR-652)是用于治疗HIV感染的实验候选药物
414910-30-8 | Casopitant甲磺酸盐
(Catalog# : 18444)
Casopitant甲磺酸盐是一种中枢作用的神经激肽(NK1)受体拮抗剂,具有
497223-25-3 | Cenicriviroc ( TAK-652 )
(Catalog# : S510902)
Cenicriviroc(TAK-652, TBR-652) 是一种CCR2和CCR5受体抑制剂,临床上它被用
432001-19-9 | C188-9
(Catalog# : 2017873)
C188-9是一种生物活性化学品。
442912-55-2 | CY5.5-SE
(Catalog# : 20177314)
2-[5-[3-[6-[(2,5-Dioxo-1-pyrrolidinyl)oxy]-6-oxohexyl]-1,3-dihydro-1,1-dimethyl-6,8-d
464-49-3 | (±)-樟脑
(Catalog# : 17021401)
(±)-樟脑是烹饪中的一种成分,作为一种用于医药用途的防腐液体
440662-09-9 | CeMMEC1
(Catalog# : 17021308)
CeMMEC1是N-methylisoquinolinone导数,抑制第二溴域 TAF1(IC50 = 0.9μM)。
474012-90-3 | CAL-130 Racemate
(Catalog# : 611824)
CAL-130 racemate is a novel phosphoinositide 3-kinase (PI3K) inhibitor. It is reporte
481-74-3 | Chrysophanic acid
(Catalog# : 161009017)
Chrysophanic acid preferentially blocked proliferation in SNU-C5 cells but not in oth
40641-90-5 | 4-cyclopropylphenylacetic acid
(Catalog# : 032509)
Coming soon!
415903-37-6 | CJ-023423
(Catalog# : 012601)
CJ-023423 is a novel, potent and selective prostaglandin EP4 receptor antagonist with
425399-05-9 | CASIN
(Catalog# : 122844)
CASIN is an inhibitor of Cdc42 GTPase, a small GTPase of the Rho-subfamily that plays
42287-94-5 | 3-(4-CYANOPHENYL)PROPANOIC ACID
(Catalog# : 90612)
Coming soon!
42287-97-8 | 3-Cyanobenzenepropanoic acid
(Catalog# : 90611)
Coming soon!
4903-09-7 | 3-Chloro-4-methoxybenzaldehyde
(Catalog# : 81004)
Cooming soon!
474-25-9 | Chenodeoxycholic Acid
(Catalog# : 52781)
Chenodeoxycholic Acid (CDCA), is a hydrophobic primary bile acid that activates nucle
442632-72-6 | CK-636
(Catalog# : 52544)
CK-636(CK-0944636) is a small molecule inhibitor of Arp2/3 complex; Inhibitor of acti
476-34-6 | Clemizole
(Catalog# : 52520)
Clemizole is a H1 histamine receptor antagonist.Recently, researchers have identified
49745-95-1 | 多巴酚丁胺盐酸盐
(Catalog# : 17030803)
多巴酚丁胺是一种交感神经药物,用于治疗心力衰竭和心源性休克
405169-16-6 | Dovitinib
(Catalog# : 16071106)
Dovitinib, also known as TKI-258 or CHIR-258, is an orally bioavailable FGFR3 inhibit
444606-18-2 | Dilmapimod
(Catalog# : 011312)
Dilmapimod is p38 MAPK inhibitor. SB-681323 inhibited the p38 MAPK pathway to a great
496807-64-8 | EN460
(Catalog# : 20603)
EN460 is an endoplasmic reticulum oxidoreductase (ERO1) inhibitor. EN460 showed a dos
441045-17-6 | Eribulin Mesylate
(Catalog# : 20354)
Eribulin is an anticancer drug marketed by Eisai Co. under the trade name Halaven. Er
491833-29-5 | 依利格鲁司特
(Catalog# : 17022718)
依利格鲁司特, 也叫Genz-112638, 是一种有效的选择性的葡萄糖酰胺合
488832-69-5 | Elesclomol
(Catalog# : 16071025)
Elesclomol, also known as STA-4783, is a HSP-90 Inhibitor, and is a small-molecule bi
426842-85-5 | 3-氟-6-甲氧基喹啉
(Catalog# : 20433)
402567-16-2 | Firategrast
(Catalog# : 16122946)
Firategrast, also known as SB-683699 or T-0047, is an orally bioavailable alpha4 beta
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
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----
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----
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----
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----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
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----
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----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
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----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
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--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
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--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
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--
Other Heterocycles
--
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--
On Sale
新产品
天然化合物
最新产品
1497439-74-3 | AD-8007
(Catalog# : 26A018)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
1802650-31-2 | ZY-444
(Catalog# : 26A020)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
2306525-79-9 | AD-5584
(Catalog# : 26A019)
AD-5584是一种新型脑渗透性ACSS2抑制剂。
3079716-11-0 | IDB-003
(Catalog# : 26A017)
IDB-003在体内抑制MDA-MB-231肿瘤生长。
1357362-02-7 | Vafidemstat
(Catalog# : 18891)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
1260247-42-4 | LLL12
(Catalog# : 25075)
LLL12是一种强效的STAT3抑制剂。LLL12在小鼠异种移植物模型中显示出
2758659-09-3 | ECC-5004
(Catalog# : 26A015)
ECC5004是一款每日一次、低剂量、小分子GLP-1受体激动剂。
2911585-37-8 | SILA-123
(Catalog# : 26A014)
SILA-123是一种II型FLT3抑制剂,对FLT3-WT(IC50=2.1 nM)和FLT3-ITD(IC50=1
1214922-52-7 | Encaleret sulfate
(Catalog# : 26A013)
Encaleret是一种正在研究的钙敏感受体的小分子拮抗剂,用于钙稳态
1431303-72-8 | Iadademstat ( ORY-1001 ) hydrochloride
(Catalog# : 26A011)
Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶