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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
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Immunology & Inflammation
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Cas号索引 2
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Cas号索引 2
2088453-21-6 | OATD-01 (GLPG-4716)
(Catalog# : 208191)
OATD-01 (GLPG-4716)是一种有效的酸性哺乳动物几丁质酶(AMCase)和壳
253426-24-3 | 奥瑞布林盐酸盐
(Catalog# : 186291)
奥瑞布林是一种合成的水溶性类似物,与combrestyatin A4类似,源自
204697-65-4 | Olcegepant
(Catalog# : 185285)
Olcegepant,又称BIBN-4096或BIBN-4096BS,是降钙素基因相关肽1 (CGRP1)受体
288847-34-7 | OXi-4503钠
(Catalog# : 178308)
OXi-4503是一种二磷酸酯类药物,开始是从植物纤维中分离出来的,
216227-54-2 | ONT-093
(Catalog# : 17030901)
ONT-093, 也称为OC-144-093,是一种口服的P-糖蛋白泵抑制剂,用于治疗
29700-22-9 | 氧化白藜芦醇
(Catalog# : 17021324)
氧化白藜芦醇,一种天然存在的化合物,尤其在Morus alba L中发现。
202590-98-5 | OTX015
(Catalog# : 111012)
OTX-015 is a new potent BRD2/3/4 inhibitor with evident anti-proliferative activity i
270065-52-6 | 1-O-benzyl 2-O-ethyl (2S)-5-oxopyrrolidine-1,2-dicarboxylate
(Catalog# : 90103)
Coming soon!
252990-05-9 | 1-O-tert-butyl 2-O-methyl (2R)-piperazine-1,2-dicarboxylate
(Catalog# : 81726)
Coming soon!
2569008-99-5 | Prifetrastat (Synonyms: PF-07248144)
(Catalog# : 26A088)
Prifetrastat (Synonyms: PF-07248144) 是一款首创、选择性、口服活性的
2756333-39-6 | Palacaparib ( Synonyms: AZD-9574 )
(Catalog# : 26A053)
Palacioparib(AZD-9574)是一种口服的中枢神经系统渗透剂PARP-1抑制剂
2170608-85-0 | PZ-3022
(Catalog# : 26A039)
PZ-3022是一种别构型的PanK激活剂,能够抵消C3-CoA的抑制作用。
2759304-23-7 | Pimicotinib hydrochloride
(Catalog# : 26A003)
Pimicotinib (ABSK021) hydrochloride 是一种选择性且具有口服活性的 CSF1R
2892065-45-9 | PLX-4545
(Catalog# : 24111)
PLX-4545 是一种口服生物可利用的 IKZF2 分子胶降解剂,旨在破坏高
2416875-06-2 | 7-氯-5-(3-戊基)吡唑并[1,5-A]嘧啶
(Catalog# : 24081)
2893778-31-7 | PHGDH-IN-3
(Catalog# : 25077)
PHGDH-IN-3 is an orally active phosphoglycerate dehydrogenase (PHGDH) inhibitor.
2101700-15-4 | Pirtobrutinib
(Catalog# : 20618)
2904682-19-3 | PDS-0330
(Catalog# : 231106)
PDS-0330 是一种特异性、有效的Claudin-1抑制剂。PDS-0330 干扰 claudin-1
2253123-16-7 | Pimicotinib
(Catalog# : 20548)
Pimicotinib是一种新型的 CSF-1R 小分子抑制剂,可口服、高选择性、
260415-63-2 | PD-173955
(Catalog# : 20499)
PD-173955 is a src tyrosine kinase inhibitor. PD173955 inhibited Bcr-Abl-dependent ce
217171-01-2 | PD-173212
(Catalog# : 20468)
PD-173212 is a small molecule N-type calcium channel blocker. PD173212 fully reduced
2172870-89-0 | Paltusotine ( CRN-00808 )
(Catalog# : 20294)
Paltusotine 是一类新型的、口服、选择性、非肽类2型生长抑素受体
26305-03-3 | Pepstatin
(Catalog# : 2071607)
Pepstatin inhibits the aspartic protease endothiapepsin.
2227425-05-8 | PF-06869206
(Catalog# : 2071506)
PF-06869206 is an Orally Bioavailable Selective Inhibitors of the Sodium-Phosphate Co
26033-20-5 | 3-PHENYL-1H-PYRAZOLE-4-CARBALDEHYDE
(Catalog# : 2062020)
248282-01-1 | Paquinimod
(Catalog# : 2061706)
Paquinimod, also known as ABR‑215757, is a S100A9 inhibitor preventing S100A9 bindi
2170608-82-7 | PZ-2891
(Catalog# : 193282)
PZ-2891是一种强效的、选择性的、口服活性泛酸激酶(PANK)调制剂,
2102501-84-6 | PF-06835919 ( MDK-1846 )
(Catalog# : 193264)
MDK1846是一种强效的酮己糖激酶(KHK)抑制剂。
2185857-97-8 | PF-06873600
(Catalog# : 191145)
PF-06873600是一种口服生物利用的细胞周期蛋白依赖性激酶(CDK)抑制
2070014-93-4 | PF-CBP1盐酸
(Catalog# : 179112)
PF-CBP1,也称为 PF06670910,是强效、高选择性的CREB结合蛋白布罗莫
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产品分类
信号通路
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----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
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----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
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----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
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----
PKA
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LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
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----
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----
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----
SSTR
-- Immunology & Inflammation
----
PD-1
----
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----
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----
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----
Histamine Receptor
----
TLR
----
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----
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----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
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----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
----
Hemoglobin
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
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----
Melanocortin Receptor
----
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----
CGRP-Receptor
----
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-- NF-κB
----
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----
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----
IKK
----
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-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
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----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
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--
Chiral Compounds
--
Deuterated
--
Fluorides
--
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Indoles and Oxindoles
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Iodos
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Nitro Compounds
--
Oxazoles
--
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Phenols
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On Sale
新产品
天然化合物
最新产品
2765593-43-7 | Linafexor (别名: CS-0159)
(Catalog# : 26A089)
Linafexor(同义词:CS-0159)是法尼醇X受体(FXR)的强效非胆汁酸激
2569008-99-5 | Prifetrastat (Synonyms: PF-07248144)
(Catalog# : 26A088)
Prifetrastat (Synonyms: PF-07248144) 是一款首创、选择性、口服活性的
2417489-10-0 | Camonsertib
(Catalog# : 24052)
Camonsertib,也称为RP 3500,是一种新型、强效和选择性的ATR抑制剂,
1429882-07-4 | MRX-2843
(Catalog# : 26A087)
MRX-2843 是一种口服可用的双受体酪氨酸激酶(RTKs)抑制剂,作用
1637394-01-4 | GDC-0134
(Catalog# : 20432)
GDC-0134是一种MAP3K12(DLK)抑制剂。
2128698-24-6 | BI-847325
(Catalog# : 25046)
BI-847325是一种新型的、可口服的、竞争ATP结合位点的Aurora激酶和M
3137699-54-5 | GDD-261
(Catalog# : 26A084)
GDD-261是一种口服活性的磷酸甘油酸脱氢酶变构抑制剂(IC50=61nM)
2669009-92-9 | Atebimetinib
(Catalog# : 25148)
Atebimetinib(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制剂
3062177-59-4 | BH-30643
(Catalog# : 26A047)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制
2490431-16-6 | ERAS-801 ( JGK-068S )
(Catalog# : 20635)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。