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抑制剂/受体激动剂
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Cas号索引 2
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Cas号索引 2
2097938-73-1 | MBQ-167
(Catalog# : 181152)
MBQ-167是一种有效的双Rac/Cdc42抑制剂,IC50分别为103/78 nM,用于转移
2109805-78-7 | MU-380
(Catalog# : 181022)
MU-380是一种有效且具有选择性的CHK1抑制剂。
2036044-77-4 | MDK-4774
(Catalog# : 18961)
MDK-4774, 又名Porcupine-IN-1, 是一种Porcupine抑制剂。
2080306-21-2 | MRT68921盐酸盐
(Catalog# : 184102)
MRT68921是ULK1和ULK2的抑制剂(IC50分别为 = 2.9和1.1 nM)。
2102196-57-4 | MDK6574
(Catalog# : 18421)
MDK6574,也称为FAA1 agonist-1,FAA1受体激动剂。
23612-48-8 | 2-甲基-7-氮杂吲哚
(Catalog# : 183131)
2-甲基-7-氮杂吲哚是一种医药中间体。
2060530-16-5 | MDK30165
(Catalog# : 179138)
MDK30165,也称为K-Ras(G12C)抑制剂6。
203849-91-6 | 单甲基澳瑞他汀 D
(Catalog# : 20179132)
MMAD又称为单甲基澳瑞他汀 D,是一种高效的微管蛋白抑制剂。MMAD
2070015-13-1 | ML241 HCl
(Catalog# : 179111)
ML241是强有力的和有选择性的蛋白酶抑制剂。ML241抑制P97 ATPase与IC
210110-90-0 | 米格鲁特盐酸盐
(Catalog# : 2017824)
米格鲁特, 也称为OGT 918,是Actelion开发的一种药物,主要用于治疗I
21516-68-7 | 红曲素
(Catalog# : 201708015)
它是一种有效的抑制剂,是由car纤维组织形成来测量不利的化学或
23007-85-4 | MPTP hydrochloride
(Catalog# : 16122796)
MPTP hydrochloride is a dopaminergic neurotoxin and cause selective destruction of do
2029049-79-2 | ML390
(Catalog# : 16122749)
ML390 is a human DHODH inhibitor that induces differentiation in acute myeloid leukem
219832-49-2 | MP-A08
(Catalog# : 6111524)
MP-A08 is a highly selective ATP competitive SK inhibitor that targets both SK1 and S
292057-76-2 | Mcl1-IN-2
(Catalog# : 6111404)
Mcl1-IN-2 is a Mcl-1 inhibitor without reported IC50 value.
256373-96-3 | MCC950 sodium
(Catalog# : 6111014)
MCC950 (CP 456773) sodium is a potent, selective, small molecule inhibitor of NLRP3 w
29906-67-0 | 1-METHYL-5-NITRO-1H-INDOLE
(Catalog# : 169701)
1-METHYL-5-NITRO-1H-INDOLE CAS#29906-67-0
210826-40-7 | MCC950
(Catalog# : 030101)
MCC950 is a potent, selective, small-molecule inhibitor of NLRP3 with IC50 of 7.5 nM
208538-73-2 | Micafungin sodium
(Catalog# : 120712)
Micafungin is an antifungal drug that belongs to the antifungal class of compounds kn
23012-17-1 | 2-Methyl-1,3-oxazole-4-carboxylic acid
(Catalog# : 91828)
Coming soon!
24623-20-9 | 6-methyl-2,3-dihydroinden-1-one
(Catalog# : 81929)
Coming soon!
24644-78-8 | 4-methyl-2,3-dihydroinden-1-one
(Catalog# : 81923)
Coming soon!
29415-97-2 | Methyl 3-bromo-4-hydroxybenzoate
(Catalog# : 80319)
Coming soon!
2227154-23-4 | N-Methylamisulpride ( 别名: LB-102 )
(Catalog# : 26A058)
N-甲基咪唑胺(同义词:LB-102)是一种多巴胺D2和D3受体拮抗剂和血
2794195-73-4 | Nomelcitinib ( D-2570 )
(Catalog# : 26A036)
Nomelcitinib (D-2570) 是一种新型TYK2变构抑制剂。
2351225-46-0 | NSD1 抑制剂 BT5
(Catalog# : 25207)
BT5可有效抑制NSD1,与细胞中的SET结构域结合,并降低H3K36me2水平。
2272917-13-0 | NT-0796
(Catalog# : 25153)
NT-0796 是一种抑制 NLRP3 炎症小体的口服小分子。
2443487-67-8 | Nivegacetor ( 别名: RG-6289, RO-7269162)
(Catalog# : 25151)
Nivegacetor(RG-6289,RO-7269162)是一种口服γ分泌酶调节剂。
2375840-87-0 | NDI-091143
(Catalog# : 24057)
NDI-091143 is a novel potent inhibitor of human ATP-citrate lyase, indirectly disrupt
2354321-33-6 | NMD670
(Catalog# : 24050)
NMD670 is an orally bioavailable skeletal muscle-specific chloride ion channel (ClC-1
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----
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----
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----
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抑制剂/受体激动剂
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新产品
天然化合物
最新产品
2765593-43-7 | Linafexor (别名: CS-0159)
(Catalog# : 26A089)
Linafexor(同义词:CS-0159)是法尼醇X受体(FXR)的强效非胆汁酸激
2569008-99-5 | Prifetrastat (Synonyms: PF-07248144)
(Catalog# : 26A088)
Prifetrastat (Synonyms: PF-07248144) 是一款首创、选择性、口服活性的
2417489-10-0 | Camonsertib
(Catalog# : 24052)
Camonsertib,也称为RP 3500,是一种新型、强效和选择性的ATR抑制剂,
1429882-07-4 | MRX-2843
(Catalog# : 26A087)
MRX-2843 是一种口服可用的双受体酪氨酸激酶(RTKs)抑制剂,作用
1637394-01-4 | GDC-0134
(Catalog# : 20432)
GDC-0134是一种MAP3K12(DLK)抑制剂。
2128698-24-6 | BI-847325
(Catalog# : 25046)
BI-847325是一种新型的、可口服的、竞争ATP结合位点的Aurora激酶和M
3137699-54-5 | GDD-261
(Catalog# : 26A084)
GDD-261是一种口服活性的磷酸甘油酸脱氢酶变构抑制剂(IC50=61nM)
2669009-92-9 | Atebimetinib
(Catalog# : 25148)
Atebimetinib(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制剂
3062177-59-4 | BH-30643
(Catalog# : 26A047)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制
2490431-16-6 | ERAS-801 ( JGK-068S )
(Catalog# : 20635)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。