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sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
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Cytoskeleton
DNA Damage
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Cas号索引 2
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Cas号索引 2
2094810-82-7 | HFY-4A
(Catalog# : 20661)
HFY-4A is a HDAC inhibitor. HFY-4A inhibits breast cancer cell proliferation, migrati
257943-19-4 | Hynic-TOC
(Catalog# : 20658)
Hynic-TOC is a ligand for making 99mTc-Hynic-TOC as an imaging agent in the diagnosti
2071224-39-8 | HDAC-IN-58
(Catalog# : 20568)
HDAC-IN-58 is a HDAC inhibitor.
28194-09-4 | 4,5-二碘-1H-1H-1,2,3-三氮唑
(Catalog# : 20521)
2569527-64-4 | HM43239
(Catalog# : 20517)
HM43239 is an orally active small molecule inhibitor of FLT3 that selectively inhibit
27192-20-7 | 5-溴-6-环丙基嘧啶-4-醇
(Catalog# : 20482)
2086183-72-2 | 1H-Indazole-1-acetic acid, 3-acetyl-5-bromo-, 1,1-dimethylethyl ester
(Catalog# : 20422)
221675-35-0 | 1H-吡咯并[2,3-B]吡啶-2-羧酸乙酯
(Catalog# : 20388)
201847-54-3 | H-BETA-ALA-AMC TFA
(Catalog# : 2071633)
2158197-70-5 | HS-1371
(Catalog# : 192223)
HS-1371是一种新型的RIP3-介导坏死性凋亡激酶抑制剂。HS-1371以ATP-竞
271-47-6 | 1H-吡唑并[3,4-C]吡啶
(Catalog# : 1781503)
1H-吡唑并[3,4-C]吡啶,1H-pyrazolo[3,4-c]pyridine
218791-21-0 | Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
2463893-46-9 | iMQT_020
(Catalog# : 26A016)
iMQT_020是一种特异性小分子抑制剂,靶向线粒体SLC1A5_var(谷氨酰胺
2244136-58-9 | Irafamdastat (Synonyms: BMS-986368)
(Catalog# : 25154)
Irafamdastat (BMS-986368;以前称为 ABX-1772) 是一种口服、中枢神经渗透
2408840-26-4 | Imlunestrant
(Catalog# : 25104)
Imlunestrant is a biochemical
2230974-62-4 | Irpagratinib
(Catalog# : 25089)
Irpagratinib是一种口服生物可利用的人成纤维细胞生长因子受体4(
259657-09-5 | Ivospemin Hydrochloride
(Catalog# : 25044)
Ivospemin is an antineoplastic spermine analogue.
2246607-08-7 | Inupadenant
(Catalog# : 24138)
Inupadenant, also known as EOS-850, is a highly selective small molecule antagonist o
2448172-22-1 | Icovamenib
(Catalog# : 24097)
This product was removed for commercial reasons.
2059148-82-0 | IMP-1088
(Catalog# : 24029)
IMP-1088 是一种有效的人 N-肉豆蔻酰转移酶 NMT1 和 NMT2 双重抑制剂。
2563892-44-2 | IK-930
(Catalog# : 20656)
IK-930 是一种新型选择性小分子 TEAD 抑制剂,可防止棕榈酸结合,
2447007-60-3 | Iptacopan hydrochloride hydrate
(Catalog# : 20649)
Iptacopan hydrochloride hydrate is a highly potent and highly selective factor B inhi
21321-89-1 | Itruvone
(Catalog# : 20623)
Itruvone is an antidepressant.
2404604-06-2 | ITK inhibitor 6
(Catalog# : 20591)
2741-16-4 | 1-ISOPROPOXYBENZENE
(Catalog# : 20406)
2160546-07-4 | IACS-13909
(Catalog# : 822221)
IACS-13909 是一种特异性且有效的 SHP2 变构抑制剂,可抑制通过 MAPK
252870-53-4(free base) | Ispronicline
(Catalog# : 20288)
Ispronicline, also known as AZD3480; TC 1734; TC-0173, and RJR 1734, is a alpha4beta2
2231259-57-5 | IACS-9439
(Catalog# : 20911)
IACS-9439是一种有效的,高选择性和口服生物利用度的CSF1R抑制剂。
2074607-48-8 | IWP-O1
(Catalog# : 186222)
IWP-O1是一种高效的Porcn抑制剂,对Wnt蛋白的分泌至关重要,它有助
22503-72-6 | IDRA-21
(Catalog# : 179134)
IDRA-21是一种阳性的AMPA受体调节剂。IDRA-21抑制突触和突触外NMDA受
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
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--
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--
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On Sale
新产品
天然化合物
最新产品
3054692-62-2 | ECI830
(Catalog# : 26A031)
ECI830是一种实验性的CDK2抑制剂。
1394076-92-6 | GNE-317
(Catalog# : 52282)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
3118994-80-9 | DPTX-3186
(Catalog# : 26A010)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
435327-40-5 | Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
1421936-85-7 | Iclepertin (BI-425809)
(Catalog# : 24084)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
4727-31-5 | Kartogenin ( KGN )
(Catalog# : 52215)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
218791-21-0 | Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
2311863-36-0 | Apecotrep (BI 764198)
(Catalog# : 26A048)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
902614-04-4 | Pantothenate kinase-IN-2
(Catalog# : 26A038)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
3062177-59-4 | BH-30643
(Catalog# : 26A047)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制