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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
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Cas号索引 2
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Cas号索引 2
2957874-18-7 | MAT2A inhibitor 5
(Catalog# : 25204)
MAT2A抑制剂5具有抑制MAT2A的高效力和对MTAP缺失的癌症细胞系的显著
2750895-97-5 | MTX115325
(Catalog# : 186264)
MTX115325是一种强效、选择性、脑渗透性USP30抑制剂,具有良好的类
2439277-80-0 | GSK4362676 ( MAT2A-IN-9 )
(Catalog# : 25147)
MAT2A-IN-9 ( GSK4362676 )是一种2-氧代喹唑啉衍生物,是一种强效的MAT2
2769008-22-0 | MEN-1703
(Catalog# : 25143)
228113-66-4 | Maralixibat Chloride
(Catalog# : 25126)
Maralixibat (also known as SHP625, LUM001, and lopixibat) is an ileal bile acid trans
2991818-13-2 | MGD-28
(Catalog# : 25073)
MGD-28 is a potent molecular glue degrader that demonstrates significant in vitro eff
2891709-58-1 | MS6105
(Catalog# : 25039)
2763252-25-9 | M3554
(Catalog# : 25017)
M3554,一种新型抗GD2抗体药物偶联物。
2990506-75-5 | ML353
(Catalog# : 24151)
ML353 is a selective ligand of mGlu5 silent allosteric modulator (SAM).
2630904-45-7 | MRTX1719
(Catalog# : 262401)
MRTX1719 is a potent and selective binder to the PRMT5•MTA complex and selectively
2326521-71-3 | MRTX849
(Catalog# : 20611)
Adagrasib, also known as MRTX849, is a potent, highly selective, oral available KRAS
2377352-49-1 | Migoprotafib
(Catalog# : 20592)
Migoprotafib, also known as GDC-1971 and RLY-1971, is a SHP2 allosteric inhibitor. GD
2861190-30-7 | Mtb-IN-2
(Catalog# : 20572)
Mtb-IN-2 (compound 10c) is an antimicrobial agent against Mycobacterium tuberculosis
2565656-70-2 | Muvalaplin
(Catalog# : 20528)
Muvalaplin是一种小分子,通过干扰载脂蛋白(a)与载脂蛋白B100的结合
2747162-85-0 | MCUF-651
(Catalog# : 20470)
MCUF-651 is a small molecule guanylyl cyclase A receptor positive allosteric modulato
2654743-22-1 | MRTX0902
(Catalog# : 171462)
MRTX0902 是一种口服有效的 SOS1 的抑制剂,IC50 为 46 nM。
210113-85-2 | 4-(2-氨基乙氧基)苯甲酸甲酯盐酸盐
(Catalog# : 20407)
235748-94-4 | methyl (3-chloropyrazin-2-yl)acetate
(Catalog# : 20395)
2385682-18-6 | methyl 3-bromo-4-ethoxy-5-formylbenzoate
(Catalog# : 20364)
24589-99-9 | 3-醛基-4-羟基苯甲酸甲酯
(Catalog# : 20362)
2621928-55-8 | MRTX1133
(Catalog# : 20291)
MRTX1133 is a potent and selective KRAS G12D inhibitor. MRTX1133 targets the KRAS G12
2416417-65-5 | MYF-01-37
(Catalog# : 20261)
MYF-01-37 is a novel covalent inhibitor of TEAD targeting Cys380 when incubated with
2144491-78-9 | MUN91789
(Catalog# : 21245)
MUN91789, also known as CPD77, is a potent inhibitor of SARS-CoV-2 main protease. MUN
2379438-80-7 | MVN38807
(Catalog# : 21243)
MVN38807, also known as Y-1, is neuraminidase (NA) inhibitor used in preparation of d
2095128-17-7 | MA-0204
(Catalog# : 2071518)
MA-0204 is a highly potent and selective PPARd modulator (PPARδ EC50 = 0.4 nM; PPARa
24673-56-1 | 3-methyl-1-benzofuran-2-carboxylic acid
(Catalog# : 2062303)
2286411-30-9 | MBX-4132
(Catalog# : 2051511)
MBX-4132 inhibit trans translation by binding to the bacterial ribosome.
215610-30-3 | 3-甲氧基-1H-吡唑
(Catalog# : 523191)
Sun-shine Chemical provides 3-methoxy-1H-pyrazole (CAS 215610-30-3) with high quality
2086689-91-8 | methyl 2-bromo-5-fluoro-3-(4-methylphenylsulfonamido)benzoate
(Catalog# : 4281905)
methyl 2-bromo-5-fluoro-3-(4-methylphenylsulfonamido)benzoate
264622-53-9 | MRS1706
(Catalog# : 19131)
MRS1706是一种选择性腺苷A2B受体逆激动剂,人类A2B、A1、A2A、A3受体
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
----
SSTR
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
----
Hemoglobin
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
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--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
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--
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--
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--
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--
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On Sale
新产品
天然化合物
最新产品
2765593-43-7 | Linafexor (别名: CS-0159)
(Catalog# : 26A089)
Linafexor(同义词:CS-0159)是法尼醇X受体(FXR)的强效非胆汁酸激
2569008-99-5 | Prifetrastat (Synonyms: PF-07248144)
(Catalog# : 26A088)
Prifetrastat (Synonyms: PF-07248144) 是一款首创、选择性、口服活性的
2417489-10-0 | Camonsertib
(Catalog# : 24052)
Camonsertib,也称为RP 3500,是一种新型、强效和选择性的ATR抑制剂,
1429882-07-4 | MRX-2843
(Catalog# : 26A087)
MRX-2843 是一种口服可用的双受体酪氨酸激酶(RTKs)抑制剂,作用
1637394-01-4 | GDC-0134
(Catalog# : 20432)
GDC-0134是一种MAP3K12(DLK)抑制剂。
2128698-24-6 | BI-847325
(Catalog# : 25046)
BI-847325是一种新型的、可口服的、竞争ATP结合位点的Aurora激酶和M
3137699-54-5 | GDD-261
(Catalog# : 26A084)
GDD-261是一种口服活性的磷酸甘油酸脱氢酶变构抑制剂(IC50=61nM)
2669009-92-9 | Atebimetinib
(Catalog# : 25148)
Atebimetinib(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制剂
3062177-59-4 | BH-30643
(Catalog# : 26A047)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制
2490431-16-6 | ERAS-801 ( JGK-068S )
(Catalog# : 20635)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。