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抑制剂/受体激动剂
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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
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分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
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Deuterated
Fluorides
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Pyrimidines
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Cas号索引 2
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Cas号索引 2
2630904-45-7 | MRTX1719
(Catalog# : 262401)
MRTX1719 is a potent and selective binder to the PRMT5•MTA complex and selectively
2326521-71-3 | MRTX849
(Catalog# : 20611)
Adagrasib, also known as MRTX849, is a potent, highly selective, oral available KRAS
2377352-49-1 | Migoprotafib
(Catalog# : 20592)
Migoprotafib, also known as GDC-1971 and RLY-1971, is a SHP2 allosteric inhibitor. GD
2861190-30-7 | Mtb-IN-2
(Catalog# : 20572)
Mtb-IN-2 (compound 10c) is an antimicrobial agent against Mycobacterium tuberculosis
2565656-70-2 | muvalaplin
(Catalog# : 20528)
2747162-85-0 | MCUF-651
(Catalog# : 20470)
MCUF-651 is a small molecule guanylyl cyclase A receptor positive allosteric modulato
2654743-22-1 | MRTX0902
(Catalog# : 171462)
MRTX0902 是一种口服有效的 SOS1 的抑制剂,IC50 为 46 nM。
210113-85-2 | 4-(2-氨基乙氧基)苯甲酸甲酯盐酸盐
(Catalog# : 20407)
235748-94-4 | methyl (3-chloropyrazin-2-yl)acetate
(Catalog# : 20395)
2385682-18-6 | methyl 3-bromo-4-ethoxy-5-formylbenzoate
(Catalog# : 20364)
24589-99-9 | 3-醛基-4-羟基苯甲酸甲酯
(Catalog# : 20362)
2621928-55-8 | MRTX1133
(Catalog# : 20291)
MRTX1133 is a potent and selective KRAS G12D inhibitor. MRTX1133 targets the KRAS G12
2416417-65-5 | MYF-01-37
(Catalog# : 20261)
MYF-01-37 is a novel covalent inhibitor of TEAD targeting Cys380 when incubated with
2144491-78-9 | MUN91789
(Catalog# : 21245)
MUN91789, also known as CPD77, is a potent inhibitor of SARS-CoV-2 main protease. MUN
2379438-80-7 | MVN38807
(Catalog# : 21243)
MVN38807, also known as Y-1, is neuraminidase (NA) inhibitor used in preparation of d
2095128-17-7 | MA-0204
(Catalog# : 2071518)
MA-0204 is a highly potent and selective PPARd modulator (PPARδ EC50 = 0.4 nM; PPARa
24673-56-1 | 3-methyl-1-benzofuran-2-carboxylic acid
(Catalog# : 2062303)
2286411-30-9 | MBX-4132
(Catalog# : 2051511)
MBX-4132 inhibit trans translation by binding to the bacterial ribosome.
215610-30-3 | 3-甲氧基-1H-吡唑
(Catalog# : 523191)
Sun-shine Chemical provides 3-methoxy-1H-pyrazole (CAS 215610-30-3) with high quality
2086689-91-8 | methyl 2-bromo-5-fluoro-3-(4-methylphenylsulfonamido)benzoate
(Catalog# : 4281905)
methyl 2-bromo-5-fluoro-3-(4-methylphenylsulfonamido)benzoate
264622-53-9 | MRS1706
(Catalog# : 19131)
MRS1706是一种选择性腺苷A2B受体逆激动剂,人类A2B、A1、A2A、A3受体
2097938-73-1 | MBQ-167
(Catalog# : 181152)
MBQ-167是一种有效的双Rac/Cdc42抑制剂,IC50分别为103/78 nM,用于转移
2109805-78-7 | MU-380
(Catalog# : 181022)
MU-380是一种有效且具有选择性的CHK1抑制剂。
2036044-77-4 | MDK-4774
(Catalog# : 18961)
MDK-4774, 又名Porcupine-IN-1, 是一种Porcupine抑制剂。
2080306-21-2 | MRT68921盐酸盐
(Catalog# : 184102)
MRT68921是ULK1和ULK2的抑制剂(IC50分别为 = 2.9和1.1 nM)。
2102196-57-4 | MDK6574
(Catalog# : 18421)
MDK6574,也称为FAA1 agonist-1,FAA1受体激动剂。
23612-48-8 | 2-甲基-7-氮杂吲哚
(Catalog# : 183131)
2-甲基-7-氮杂吲哚是一种医药中间体。
2060530-16-5 | MDK30165
(Catalog# : 179138)
MDK30165,也称为K-Ras(G12C)抑制剂6。
203849-91-6 | 单甲基澳瑞他汀 D
(Catalog# : 20179132)
MMAD又称为单甲基澳瑞他汀 D,是一种高效的微管蛋白抑制剂。MMAD
2070015-13-1 | ML241 HCl
(Catalog# : 179111)
ML241是强有力的和有选择性的蛋白酶抑制剂。ML241抑制P97 ATPase与IC
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
1497439-74-3 | AD-8007
(Catalog# : 26A018)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
1802650-31-2 | ZY-444
(Catalog# : 26A020)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
2306525-79-9 | AD-5584
(Catalog# : 26A019)
AD-5584是一种新型脑渗透性ACSS2抑制剂。
3079716-11-0 | IDB-003
(Catalog# : 26A017)
IDB-003在体内抑制MDA-MB-231肿瘤生长。
1357362-02-7 | Vafidemstat
(Catalog# : 18891)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
1260247-42-4 | LLL12
(Catalog# : 25075)
LLL12是一种强效的STAT3抑制剂。LLL12在小鼠异种移植物模型中显示出
2758659-09-3 | ECC-5004
(Catalog# : 26A015)
ECC5004是一款每日一次、低剂量、小分子GLP-1受体激动剂。
2911585-37-8 | SILA-123
(Catalog# : 26A014)
SILA-123是一种II型FLT3抑制剂,对FLT3-WT(IC50=2.1 nM)和FLT3-ITD(IC50=1
1214922-52-7 | Encaleret sulfate
(Catalog# : 26A013)
Encaleret是一种正在研究的钙敏感受体的小分子拮抗剂,用于钙稳态
1431303-72-8 | Iadademstat ( ORY-1001 ) hydrochloride
(Catalog# : 26A011)
Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶