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抑制剂/受体激动剂
Angiogenesis
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Aldehydes
Amines
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Boronic Acids
Bromides
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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
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分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
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Indoles and Oxindoles
Iodos
Nitro Compounds
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Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
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Other Azoles
Other Heterocycles
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Cas号索引 2
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Cas号索引 2
2072057-17-9 | RG7834
(Catalog# : 19355)
RG7834,也称为RO7020322,是一种新型口服HBV病毒基因表达抑制剂阻断病
252889-88-6 | RWJ-56110
(Catalog# : 19353)
RWJ-56110是一种选择性蛋白酶活化受体-1 (PAR1)拮抗剂。它阻断凝血酶
259188-38-0 | Rebimastat
(Catalog# : 192254)
Rebimastat,又名BMS275291,是一种具有潜在抗肿瘤活性的巯基第二代
2172651-73-7 | RMC-4550
(Catalog# : 186251)
RMC-4550一种有效且具有选择性的SHP2抑制剂。
2133832-83-2 | R-IMPP
(Catalog# : 18413)
R-IMPP是PCSK9的转化抑制剂。
2003234-63-5 | R-GNE-140
(Catalog# : 18432)
R-GNE-140是一种新型高效的乳酸脱氢酶(LDHA)抑制剂,LDHA的IC50为3nM,
2097334-19-3 | (2R,14R)-4-((R)-1-((R)-4-benzyl-2-oxooxazolidin-3-yl)-3-(tert-butoxycarbonyl)-1-oxopropan-2-yl)benzyl 2,4-dimethylbenzoate
(Catalog# : 183217)
(2R,14R)-4-((R)-1-((R)-4-benzyl-2-oxooxazolidin-3-yl)-3-(tert-butoxycarbonyl)-1-oxopr
2097334-18-2 | (R)-4-(2-(4-benzyl-2-oxooxazolidin-3-yl)-2-oxoethyl)benzyl 2,4-dimethylbenzoate
(Catalog# : 183216)
(R)-4-(2-(4-benzyl-2-oxooxazolidin-3-yl)-2-oxoethyl)benzyl 2,4-dimethylbenzoate是一
269730-03-2 | RPI-1
(Catalog# : 17030301)
RPI-1是一种ATP依赖的RET激酶抑制剂。通过口服RPI-1,导致生长阻滞
283173-50-2 | Rucaparib
(Catalog# : 123005)
Rucaparib is an inhibitor of PARP with Ki of 1.4 nM for PARP1, also showing binding a
27298-99-3 | (1R)-1-(4-chlorophenyl)ethanamine
(Catalog# : 91124)
Coming soon!
239105-47-6 | (1R)-1-(4-methylphenyl)propan-1-amine,hydrochloride
(Catalog# : 91106)
Coming soon!
23844-66-8 | (1R)-2-methyl-1-phenylpropan-1-amine
(Catalog# : 91103)
Coming soon!
278788-60-6 | (2R)-1-[(2-methylpropan-2-yl)oxycarbonyl]piperazine-2-carboxylic acid
(Catalog# : 81724)
Coming soon!
213261-59-7 | RITA
(Catalog# : 52526)
RITA(NSC 652287) induced both DNA-protein and DNA-DNA cross-links with no detectable
2260969-36-4 | Selnoflast (别名:RO-7486967 ; IZD334)
(Catalog# : 25167)
Selnoflast,也称为 RO-7486967 或 IZD334,是一种抑制 NLRP3 炎症小体的强
2521285-05-0 | Sevabertinib ( 别名:BAY-2927088 )
(Catalog# : 25079)
Sevabertinib ( BAY-2927088 )是一种口服非共价酪氨酸激酶受体抑制剂(
2805997-46-8 | Survodutide
(Catalog# : 25043)
2097938-74-2 | Stafib-2
(Catalog# : 24142)
Stafib-2 is a potent and selctive inhibitor of the transcription factor STAT5b, with
2589531-76-8 | Saruparib
(Catalog# : 24100)
Saruparib, also known as AZD5305 is a potent, selective and oral active PARP inhibito
2274723-90-7 | SPG-302
(Catalog# : 24065)
Phenylbenzothiazole-PEG4-OH (compound 1) can treat spinal cord injury and promote spi
2226636-04-8 | Soquelitinib ( CPI-818 )
(Catalog# : 20671)
Soquelitinib(CPI-818)是一种高度选择性的共价白细胞介素-2诱导的T
2222138-31-8 (HCl) | Sotuletinib HCl
(Catalog# : 20663)
Sotuletinib, also known as BLZ945, is a potent and selective CSF-1R kinase inhibitor.
2383086-06-2 | Sonrotoclax (BGB-11417)
(Catalog# : 20650)
Sonrotoclax is an antineoplastic.
2546091-70-5 | SOP1812 (QN-302)
(Catalog# : 20639)
QN-302 是一种 G4选择性转录抑制剂。
256414-75-2 | SEW2871
(Catalog# : 20604)
SEW2871 is a S1P1 agonist (sphingosine-1-phosphate type 1 receptor agonist). SEW2871
2765525-82-2 | STX-721
(Catalog# : 20576)
STX-721 is a next-generation, orally delivered therapy, designed with potential best-
2648257-56-9 | STC-15
(Catalog# : 20549)
STC-15 is a first-in-class inhibitor of RNA modification and is the first ever RNA me
2921961-53-5 | (S)-5-fluoro-3-methylbenzo[c][1,2]oxaborol-1(3H)-ol
(Catalog# : 20522)
2170746-98-0 | Spiro[cyclohexane-1,9'(6'H)-pyrazino[1',2':1,5]pyrrolo[2,3-d]pyrimidine]-7'(8'H)-carboxylic acid, 2'-(methylthio)-6'-oxo-5'-[[(trifluoromethyl)sulfonyl]oxy]-, 1,1-dimethylethyl ester
(Catalog# : 20412)
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2750895-97-5 | MTX115325
(Catalog# : 186264)
MTX115325是一种强效、选择性、脑渗透性USP30抑制剂,具有良好的类
2166616-75-5 | LY-3381916
(Catalog# : 193123)
LY-3381916是一种强效的、选择性的、脑透性的IDO1活性抑制剂,与缺
2376397-93-0 | Opakalim
(Catalog# : 25193)
Opakalim(BHV-7000)是Kv7.2/7.3钾通道(KCNQ2/3)的口服小分子激活剂,
2488609-21-6 | DS68591889
(Catalog# : 25158)
DS68591889 (PTDSS1i) 特异性抑制 PTDSS1,而 PTDSS1 可催化丝氨酸掺入 PC。
944808-88-2 | CAY 10566
(Catalog# : 10403)
CAY 10566是一种强效的选择性SCD-1抑制剂。
2308520-97-8 | Cadefrecitinib (GLPG-3667)
(Catalog# : 20509)
Cadefrecitinib(GLPG-3667)是一种口服小分子TYK2激酶抑制剂,目前正处
1802735-28-9 | QBS10072S
(Catalog# : 25190)
QBS10072S 是一种血脑屏障 (BBB) 渗透剂,由细胞毒性化疗结构域 N-双
2377000-84-3 | Dencatistat (STP938)
(Catalog# : 25177)
Dencatistat 是一种口服生物可利用的小分子胞苷三磷酸合酶 1 (CTPS1)
1898207-64-1 | DS-1001b
(Catalog# : 25178)
DS-1001 是一种口服的脑渗透性突变 IDH1 选择性抑制剂。
1016340-64-9 | Z57346765
(Catalog# : 25191)
Z57346765 是一种 PGK1 特异性抑制剂,可降低 PGK1 糖酵解中代谢酶的