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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
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Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
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Chiral Compounds
Deuterated
Fluorides
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Indoles and Oxindoles
Iodos
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Peg Linkers
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Piperidines
Pyridines
Pyrimidines
Quinolines
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Other Azoles
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Cas号索引 1
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Cas号索引 1
1508250-71-2 | Nazartinib (EGF816)
(Catalog# : 1781004)
Nazartinib,也被称为EGF816,是一种口服可用,不可逆转的、第三代、
1254032-66-0 | Netarsudil
(Catalog# : 1781001)
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1676893-24-5 | NSC781406
(Catalog# : 20178810)
NSC781406是一种高效针对PI3K的IC50为2 nM的PI3K和mTOR抑制剂。
1916571-90-8 | NCT-503
(Catalog# : 2017888)
NCT-503是一种3 -磷酸甘油酸脱氢酶(PHGDH)抑制剂,抑制丝氨酸合成3 -磷
1304630-27-0 | NGP-555
(Catalog# : 2017875)
NGP 555正在被作为一种预防疾病老年痴呆症的治疗。
147149-76-6 | 诺拉曲特
(Catalog# : 17030908)
诺拉曲特,也叫AG337,是一种具有潜在抗癌活性的百里香酶抑制剂
1221713-92-3 | NPS-1034
(Catalog# : 17030907)
NPS-1034是一种新型的MET抑制剂,它能抑制活化的MET受体及其具有结
1400-61-9 | 制霉菌素
(Catalog# : 17030905)
制霉菌素是一种多烯抗真菌药物,含有三种生物活性成分的抗生素
1354744-91-4 | 聚乙二醇纳诺醇
(Catalog# : 17030202)
Naloxegol,也称为NKTR-118和AZ-13337019,是一种选择性的阿片拮抗剂,用于
1038915-64-8 | 尼拉帕尼盐酸盐
(Catalog# : 17030114)
尼拉帕尼, 也称为MK-4827, 是一种具有潜在抗肿瘤活性的聚(ADP-核糖
1698878-14-6 | Nampt-IN-1
(Catalog# : 17022705)
Nampt-IN-1是NAMPT的一种新型抑制剂,IC50分别为18 nM(NCI- H1155细胞),4
102586-30-1 | NSC12
(Catalog# : 17021317)
NSC12是一种可用于抑制FGF2 / FGFR相互作用并具有良好的抗肿瘤活性
123653-11-2 | NS-398 (NS398)
(Catalog# : 17011106)
NS-398是一种cyclooxygenase-2 (COX-2)的选择性抑制剂。
1253952-02-1 | Netarsudil (AR-13324) 2HCl
(Catalog# : 1710901)
Netarsudil (a.k.a. AR-13324)是一种ROCK抑制剂,Ki值为 0.2-10.3 nM。它目前
1313363-54-0 | NVP-CGM097
(Catalog# : 16122789)
NVP-CGM097 is a highly potent and selective MDM2 inhibitor. It binds to the p53 bindi
113104-25-9 | NSC228155
(Catalog# : 16122779)
NSC228155 is an activator of EGFR, binding to the sEGFR dimerization domain II and mo
175026-96-7 | NQDI-1
(Catalog# : 16122772)
NQDI 1, an inhibitor of ASK1(apoptosis signal-regulating kinase 1), attenuates acute
1360614-48-7 | Necrosulfonamide
(Catalog# : 6111508)
Necrosulfonamide is a very specific and potent necrosis inhibitor and blocks mixed li
154447-35-5 | NU 7026
(Catalog# : 6118017)
NU 7026 is a novel and potential inhibitor of the DNA repair enzyme DNA-dependent pro
1449236-96-7 | NMS-859
(Catalog# : 161014001)
NMS-859 is a potent and specific small molecule covalent inhibitor of the ATPase VCP/
1802088-50-1 | NCT-501
(Catalog# : 16071414)
NCT-501 is a potent ALDH1A1 inhibitor. Aldehyde dehydrogenases (ALDHs) metabolize rea
140926-75-6 | NSC5844
(Catalog# : 16060601)
NSC5844
161058-83-9 | NU2058
(Catalog# : 032515)
Coming soon!
1599432-08-2 | NIBR189
(Catalog# : 012007)
NIBR189 is a small molecule antagonist of the Epstein-Barr virus-induced gene 2 (EBI2
1419949-20-4 | NVP-TNKS656
(Catalog# : 010408)
NVP-TNKS656 is a highly potent, selective, and orally active TNKS2 inhibitor with IC5
121032-29-9 | Nelarabine
(Catalog# : 010404)
Nelarabine is a Nucleoside Metabolic Inhibitor. The mechanism of action of nelarabine
104206-65-7 | Nitisinone
(Catalog# : 122526)
Nitisinone is a Hydroxyphenyl-Pyruvate Dioxygenase Inhibitor.
131060-14-5 | NB-598
(Catalog# : 121405)
NB-598 is a potent competitive inhibitor of squalene epoxidase (SE), which suppresses
101385-93-7 | N-Boc-3-Pyrrolidinone
(Catalog# : 90714)
Coming soon!
16642-79-8 | 3-(4-Nitrophenyl)propanoic acid
(Catalog# : 90618)
Coming soon!
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2750001-23-9 | AZD0095
(Catalog# : 237072)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2101538-28-5 | 2-MNG
(Catalog# : 24129)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
2439277-80-0 | MAT2A-IN-9
(Catalog# : 25147)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
1898206-17-1 | Safusidenib
(Catalog# : 25149)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
2669009-92-9 | Atebimetinib
(Catalog# : 25148)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
2242751-53-5 | Acoramidis hydrochloride
(Catalog# : 24068)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
2230263-60-0 | Crelosidenib
(Catalog# : 24101)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
2833703-74-3 | LOXO-435
(Catalog# : 25080)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
2446928-30-7 | Gridegalutamide
(Catalog# : 25138)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
1256349-48-0 | Chiauranib
(Catalog# : 25146)
Chiauranib also known as orally available, small molecule inhibitor of select serine-