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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
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Cas号索引 1
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Cas号索引 1
1421373-62-7 | MDK3627
(Catalog# : 187161)
MDK3627,也被称为突变EGFR抑制剂,是一种选择性和强效突变的EGFR抑
1303607-07-9 | MI-773
(Catalog# : 185251)
MI-773是一种新型的口服MDM2拮抗剂。
1417997-93-3 | MDK-7933
(Catalog# : 184161)
MDK-7933,也称为HDAC8-IN-1,是一种HDAC8 抑制剂,在癌症细胞器的IC50
1448189-80-7 | MDK7526盐酸盐
(Catalog# : 184104)
MDK7526, 也称为VHL Ligand 1,Protein degrader 1是一种有效的、选择性的蛋
1190379-70-4 | MRT68921
(Catalog# : 184103)
MRT68921是ULK1和ULK2的抑制剂(IC50 分别为= 2.9和1.1 nM)。
1870916-87-2 | Mc-Val-Ala-PAB
(Catalog# : 184219)
Mc-Val-Ala-PAB 是一种用于靶向药物传递的药物-药物结合剂(ADC)的有用
111797-22-9 | MDK7229
(Catalog# : 184211)
MDK7229, also known as MD2-IN-1 is a MD2 (Myeloid differentiation protein 2) inhibito
1215310-75-0 | 4-methylsulfonyl-2-(trifluoromethyl)benzaldehyde
(Catalog# : 1712293)
4-methylsulfonyl-2-(trifluoromethyl)benzaldehyde isa building blocks.
1187990-87-9 | MK-8617
(Catalog# : 1710163)
MK-8617是一种缺氧诱导因子(HIF脯氨酰羟化酶1−3 PHD1−3),具有强效
1883423-59-3 | MSC2530818
(Catalog# : 1710135)
MSC2530818是一种强效、选择性,口服生物利用度与抑制剂的IC50 = 2.
132819-92-2 | MDK19922
(Catalog# : 1791512)
MDK19922,也称为NOD-IN-1或化合物4,是一种有效的核苷酸结合寡聚化
137975-06-5 | 游离莫扎伐普坦
(Catalog# : 179154)
莫扎伐普坦,又名OPC 31260,是由大冢销售的血管加压素受体拮抗剂
1016535-83-3 | MDK35833
(Catalog# : 179114)
MDK35833又称为Oct3/4-inducer-1,是一种有效率的Oct3/4诱导者。MDK35833可
1991986-30-1 | ML364
(Catalog# : 179833)
ML364是具有潜在抗癌活性的小分子抑制剂的去泛素化酶USP2。
1422269-30-4 | ML-18
(Catalog# : 179810)
ML-18是蛙皮素受体亚型3(BRS-3)拮抗剂(IC50 = 4.8μm)。ML-18抑制肺
1207253-08-4 | MK-1064
(Catalog# : 16123054)
MK-1064是一种有效的、选择性和口服的Orexin OX2受体拮抗剂,用于治
1857417-13-0 | MI-503
(Catalog# : 178908)
MI-503是一种具有IC50为14.7 nM的有效和选择性的menin - mll抑制剂。在
1206799-15-6 | Merestinib (LY2801653)
(Catalog# : 178905)
Merestinib,又名LY2801653,是一种可口服的小分子抑制剂,原癌基因
1628317-18-9 | MI-463
(Catalog# : 17031006)
MI-463是一种Menin-MLL强力抑制剂,与IC50值15.3 nM相互作用。
1221186-53-3 | ML-265
(Catalog# : 17030804)
ML265是一个强有力的PKM2活化剂诱导四聚体,降低肿瘤的形成和大小
1346528-06-0 | ML241
(Catalog# : 17030714)
ML241是一种p97 ATPase有效的选择性抑制剂。ML241抑制p97 ATPase的IC(50)值
198821-22-6 | Merimepodib
(Catalog# : 17030308)
Merimepodib, 也称为VX-497,是有效的口服生物IMPDH抑制剂,它可以抑制
1550008-55-3 | ML-264
(Catalog# : 17030302)
ML-264是一种Krüppel-like因子5(KLF5)抑制剂,能有效抑制结直肠癌的生
1030612-90-8 | MK-8245
(Catalog# : 17030109)
MK-8245是一种有效的、以肝脏为靶点的SCD抑制剂,具有临床前抗糖
1268454-23-4 | MLN-1117
(Catalog# : 17030101)
Serabelisib(又名MLN1117,INK1117,TAK- 117)是一类具有潜在抗肿瘤活性的磷
1404437-62-2 | ML-281
(Catalog# : 17022811)
ML-281是一种有效的选择性STK33抑制剂(IC50 = 14nm)。与其他STK33抑制剂
1502816-23-0 | MS049
(Catalog# : 17021313)
MS049是PRMT4和PRMT6的一种有效的选择性抑制剂,IC50分别为34 nM和43 n
1313883-00-9 | Miransertib(ARQ 092)
(Catalog# : 17021301)
ARQ 092是一种新型的口服生物可用性和选择性AKT通路抑制剂,在晚
1399840-35-7 | MT-DADMe-ImmA(MTDIA HCl)
(Catalog# : 712101)
MT-DADMe-ImmA(MTDIA盐酸盐)是一种新型的MTAP抑制剂,具有治疗头颈部和
110448-33-4 | ML-7
(Catalog# : 17011107)
ML-7是平滑肌肌球蛋白轻链激酶的抑制剂(MLCK),Ki值为0.3μM。
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2750001-23-9 | AZD0095
(Catalog# : 237072)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2101538-28-5 | 2-MNG
(Catalog# : 24129)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
2439277-80-0 | MAT2A-IN-9
(Catalog# : 25147)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
1898206-17-1 | Safusidenib
(Catalog# : 25149)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
2669009-92-9 | Atebimetinib
(Catalog# : 25148)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
2242751-53-5 | Acoramidis hydrochloride
(Catalog# : 24068)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
2230263-60-0 | Crelosidenib
(Catalog# : 24101)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
2833703-74-3 | LOXO-435
(Catalog# : 25080)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
2446928-30-7 | Gridegalutamide
(Catalog# : 25138)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
1256349-48-0 | Chiauranib
(Catalog# : 25146)
Chiauranib also known as orally available, small molecule inhibitor of select serine-