武汉永璨生物科技有限公司
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Epigenetics
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Bromides
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
PROTAC
Antibody-drug Conjugate/ADC Related
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
中间体
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定制合成
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Cas号索引 1
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Cas号索引 1
1312941-07-3 | 3-methoxy-4-(2-morpholinoethoxy)benzoic acid hydrochloride
(Catalog# : 2062018)
1417700-13-0 | ML188
(Catalog# : 2051506)
ML188 is a Potent Noncovalent Small Molecule Inhibitor of the Severe Acute Respirator
1401242-74-7 | ML277
(Catalog# : 2051504)
ML277 is a potent activator of KCNQ1 (Kv7.1) channels with >100-fold selectivity v
1201935-85-4 | 3-甲氧基-1-甲基-4-硝基-1H-吡唑
(Catalog# : 523192)
Sun-shine Chemical provides 3-methoxy-1-methyl-4-nitro-1H-pyrazole(CAS 1201935-85-4)
1260075-17-9 | Mitapivat
(Catalog# : 192191)
Mitapivat,又称PKM2激活剂1020,是一种治疗丙酮酸激酶缺乏症的PKM2激
1219737-12-8 | MK-3903
(Catalog# : 192183)
MK-3903是一种有效的选择性AMPK激活剂(EC50 = 8 nM)。
1049704-18-8 | MA242 TFA
(Catalog# : 191256)
MA242是MDM2和NFAT1在胰腺癌治疗中的双重抑制剂。无论p53状态如何,
1799631-75-6 | MIK665
(Catalog# : 191252)
MIK665,又称s64315,诱导骨髓白血病细胞分化蛋白(mcl1;Bcl2-L-3),具有
183721-13-3 | MRS1177
(Catalog# : 1812296)
MRS1177是一种生物活性化学物。
1642288-47-8 | Mavacamten
(Catalog# : 181255)
Mavacamten,又称SAR-439152和MYK-461,是一种潜在的治疗肥厚性心肌病的
147116-67-4 | 马罗皮坦
(Catalog# : 1811261)
马罗皮坦,又称CJ11972,是一种神经激肽(NK1)受体拮抗剂。
183721-15-5 | MRS1220
(Catalog# : 1810228)
MRS1220是人A3腺苷受体的一种有效且高度选择性的拮抗剂。
1445251-22-8 | ME0328
(Catalog# : 1810174)
ME0328是一种PARP-3的抑制剂(IC50 = 0.89 μM)。
1908414-82-3 | MDK-4823
(Catalog# : 18962)
MDK-4823,又称LMPTP抑制剂1;是低分子量酪氨酸磷酸酶(LMPTP)的有效抑
1644342-14-2 | ML-792
(Catalog# : 18941)
ML-792是一种有效的选择性SAE抑制剂,在细胞检测中具有纳米极的效
1883510-31-3 | ML327
(Catalog# : 187162)
ML327是MYC的阻滞剂。ML327介导了E-cadherin的转录去抑制和对上皮-间充
1421373-62-7 | MDK3627
(Catalog# : 187161)
MDK3627,也被称为突变EGFR抑制剂,是一种选择性和强效突变的EGFR抑
1303607-07-9 | MI-773
(Catalog# : 185251)
MI-773是一种新型的口服MDM2拮抗剂。
1417997-93-3 | MDK-7933
(Catalog# : 184161)
MDK-7933,也称为HDAC8-IN-1,是一种HDAC8 抑制剂,在癌症细胞器的IC50
1448189-80-7 | MDK7526盐酸盐
(Catalog# : 184104)
MDK7526, 也称为VHL Ligand 1,Protein degrader 1是一种有效的、选择性的蛋
1190379-70-4 | MRT68921
(Catalog# : 184103)
MRT68921是ULK1和ULK2的抑制剂(IC50 分别为= 2.9和1.1 nM)。
1870916-87-2 | Mc-Val-Ala-PAB
(Catalog# : 184219)
Mc-Val-Ala-PAB 是一种用于靶向药物传递的药物-药物结合剂(ADC)的有用
111797-22-9 | MDK7229
(Catalog# : 184211)
MDK7229, also known as MD2-IN-1 is a MD2 (Myeloid differentiation protein 2) inhibito
1215310-75-0 | 4-methylsulfonyl-2-(trifluoromethyl)benzaldehyde
(Catalog# : 1712293)
4-methylsulfonyl-2-(trifluoromethyl)benzaldehyde isa building blocks.
1187990-87-9 | MK-8617
(Catalog# : 1710163)
MK-8617是一种缺氧诱导因子(HIF脯氨酰羟化酶1−3 PHD1−3),具有强效
1883423-59-3 | MSC2530818
(Catalog# : 1710135)
MSC2530818是一种强效、选择性,口服生物利用度与抑制剂的IC50 = 2.
132819-92-2 | MDK19922
(Catalog# : 1791512)
MDK19922,也称为NOD-IN-1或化合物4,是一种有效的核苷酸结合寡聚化
137975-06-5 | 游离莫扎伐普坦
(Catalog# : 179154)
莫扎伐普坦,又名OPC 31260,是由大冢销售的血管加压素受体拮抗剂
1016535-83-3 | MDK35833
(Catalog# : 179114)
MDK35833又称为Oct3/4-inducer-1,是一种有效率的Oct3/4诱导者。MDK35833可
1991986-30-1 | ML364
(Catalog# : 179833)
ML364是具有潜在抗癌活性的小分子抑制剂的去泛素化酶USP2。
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
-- PROTAC
----
Molecular Glues
--
Antibody-drug Conjugate/ADC Related
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2102501-84-6 | PF-06835919 ( MDK-1846 )
(Catalog# : 193264)
MDK1846是一种强效的酮己糖激酶(KHK)抑制剂。
2671128-05-3 | FHD-286
(Catalog# : 20471)
FHD-286 is an oral, small-molecule, selective, allosteric inhibitor of BRG1 and BRM i
3002056-30-3 | NST-628
(Catalog# : 24058)
NST-628 是具有血脑屏障渗透性的 MAPK 通路分子胶,能够抑制 RAF 磷
2893778-31-7 | PHGDH-IN-3
(Catalog# : 25077)
PHGDH-IN-3 is an orally active phosphoglycerate dehydrogenase (PHGDH) inhibitor.
2882165-79-7 | CFT1946
(Catalog# : 25078)
CFT1946 是一种口服生物可利用的小分子降解剂,可降解实体瘤中的
68238-36-8 | 异硫蓝
(Catalog# : 178017)
Isosulfan blue 是一种用于淋巴管造影中淋巴管识别的蓝色染料。Isos
2803470-63-3 | HC-7366
(Catalog# : 25076)
HC-7366 is a potent and selective activator of the general control nonderepressible 2
2226636-04-8 | Soquelitinib ( CPI-818 )
(Catalog# : 20671)
Soquelitinib(CPI-818)是一种高度选择性的共价白细胞介素-2诱导的T
2230263-60-0 | Crelosidenib
(Catalog# : 24101)
Crelosidenib is an isocitrate dehydrogenase 1 (IDH1) inhibitor. It is an antineoplast
1260247-42-4 | LLL12
(Catalog# : 25075)
LLL12 is a potent STAT3 inhibitor. LLL12 inhibits colony formation and cell migration