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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
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Bromides
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Deuterated
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Pyrimidines
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Cas号索引 1
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Cas号索引 1
118414-82-7 | MK 886
(Catalog# : 122217)
MK 886 is a leukotriene antagonist. It may perform this by blocking the 5-lipoxygenas
1430213-30-1 | ML216
(Catalog# : 122101)
ML216 is a potent inhibitor of the DNA unwinding activity of BLM helicase; showing si
1010085-13-8 | MK-5108
(Catalog# : 121504)
MK-5108 is a highly selective Aurora A inhibitor with IC50 of 0.064 nM; 220- and 190-
115550-35-1 | Marbofloxacin
(Catalog# : 121425)
Marbofloxacin is a potent antibiotic of which depends upon its inhibition of DNA-gyra
1162656-22-5 | MCB-613
(Catalog# : 111305)
Coming soon!
133407-82-6 | MG-132
(Catalog# : 111303)
MG-132 is an inhibitor of proteasome with IC50 of 100 nM, and also inhibits calpain w
1303607-60-4 | MI-773
(Catalog# : 102207)
MI-773 is an orally available spiro-oxindole HDM2 (human double minute 2) antagonist
1265905-21-2 | methyl 2-((1R,3S)-3-amino-1-hydroxy-4-methylpentyl)thiazole-4-carboxylate
(Catalog# : 91809)
Coming soon!
1206524-85-7 | MK-5172 intermediate
(Catalog# : 91802)
MK-5172(Grazoprevir) intermediate
1206524-84-6 | Methyl (1aR,5S,8S,10R,22aR)-5-tert-butyl-14-methoxy-3,6-dioxo-
(Catalog# : 91801)
MK-5172(Grazoprevir) intermediate
183429-63-2 | METHYL 1-AMINO-1-CYCLOHEPTANECARBOXYLATE
(Catalog# : 83111)
Coming soon!
13623-25-1 | 6-Methoxy-1-indanone
(Catalog# : 81924)
Coming soon!
18372-22-0 | methyl 2-(1H-indol-3-yl)-2-oxoacetate
(Catalog# : 81921)
Coming soon!
196929-78-9 | 2-methylpropane-2-sulfinamide
(Catalog# : 81914)
Coming soon!
129799-08-2 | Methyl 4-Boc-Piperazine-2-Carboxylate
(Catalog# : 81704)
Coming soon!
1131594-45-0 | Methyl 3-bromo-4-(trifluoromethoxy)benzoate
(Catalog# : 81018)
Coming soon!
14034-08-3 | Methyl 3-bromo-4-(tert-butyl)benzoate
(Catalog# : 81013)
Coming soon!
113642-05-0 | Methyl 3-bromo-4-ethylbenzoate
(Catalog# : 81007)
Coming soon!
1131587-97-7 | Methyl 5-bromo-2-methoxy-4-(trifluoromethyl)benzoate
(Catalog# : 80310)
Coming soon!
152849-72-4 | Methyl 5-bromo-2,4-dimethylbenzoate
(Catalog# : 80309)
Coming soon!
121917-57-5 | (-)-MK801(maleate)
(Catalog# : 71902)
(-)-MK801 is a elective and non-competitive NMDA receptor antagonist. Less active ena
1246529-32-7 | MPI-0479605
(Catalog# : 62907)
MPI-0479605, a small-molecule inhibitor of the mitotic kinase Mps1.Cells treated with
151767-02-1 | Montelukast sodium
(Catalog# : 52809)
Montelukast Sodium(Singulair) is a potent, selective, anti-inflammatory CysLT1 recept
1201902-80-8 | MLN9708
(Catalog# : 52749)
MLN9708 immediately hydrolyzed to MLN2238, which is an N-capped dipeptidyl leucine bo
1062368-49-3 | ML347
(Catalog# : 52742)
ML347(DN193719) is a highly selective ALK1/ALK2 inhibitor with IC50s of 46/32 nM; sho
1228960-69-7 | MLN0905
(Catalog# : 52827)
MLN0905 is a small-molecule and potent inhibitor of PLK1 with IC50 of 2 nM.
1032350-13-2 | MK 2206
(Catalog# : 51505)
MK-2206 (Merck, Whitehouse Station, NJ) is an investigational oral allosteric AKT inh
130798-51-5 | MDL-29951
(Catalog# : 52545)
MDL-29951 is a novel glycine antagonist of NMDA receptor activation (Ki=0.14 mM, [3H]
1395084-25-9 | MS436
(Catalog# : 52317)
MS436 is a diazobenzene-based small-molecule inhibitor for the BRD4 bromodomains with
13116-77-3 | NSC624206
(Catalog# : 26A028)
NSC624206是一种泛素E1抑制剂,它特异性地抑制泛素(Ub)和泛素连
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
----
SSTR
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
----
Hemoglobin
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2417955-18-9 | Osivelotor (别名: GBT-601; GBT-021601)
(Catalog# : 26A061)
Osivelotor(同义词:GBT-601;GBT-021601)是下一代镰状血红蛋白(HbS)
2389060-50-6 | Linvemastat (别名: FP-020)
(Catalog# : 26A060)
Linvemastat(FP-020)是一种高效、选择性口服MMP-12抑制剂。
3041025-10-6 | BLU-808
(Catalog# : 26A024)
BLU-808是一种针对肥大细胞疾病的野生型c-KIT的强效且具有选择性的
1695564-98-7 | SCO-240
(Catalog# : 26A059)
SCO-240是一种研究性、口服活性和选择性生长抑素受体亚型5(SSTR5
2227154-23-4 | N-Methylamisulpride ( 别名: LB-102 )
(Catalog# : 26A058)
N-甲基咪唑胺(同义词:LB-102)是一种多巴胺D2和D3受体拮抗剂和血
1898207-64-1 | Safusidenib Erbumine
(Catalog# : 25178)
DS-1001 是一种口服的脑渗透性突变 IDH1 选择性抑制剂。
2837993-05-0 | Repinatrabit ( 别称: JNT-517 )
(Catalog# : 26A056)
Repinatrabit(JNT-517)是一种针对Phe转运蛋白SLC6A19的研究性、选择性
1361200-34-1 | Privosegtor ( 别名: OCS-05, ACT-01 )
(Catalog# : 26A055)
Privosegtor(OCS-05,ACT-01)是一种小分子拟肽、BDNF/NT-3生长因子受体
2923356-52-7 | ART-6043
(Catalog# : 26A054)
ART-6043是一种口服的DNA聚合酶θ(POLQ)小分子抑制剂。
2756333-39-6 | Palacaparib ( Synonyms: AZD-9574 )
(Catalog# : 26A053)
Palacioparib(AZD-9574)是一种口服的中枢神经系统渗透剂PARP-1抑制剂