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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
PROTAC
Antibody-drug Conjugate/ADC Related
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Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
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Chiral Compounds
Deuterated
Fluorides
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Cas号索引 1
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Cas号索引 1
1263373-43-8 | NVP-2
(Catalog# : 193205)
NVP-2是细胞周期蛋白依赖性激酶CDK9的抑制剂。
1566-81-0 | NS-1652
(Catalog# : 19361)
NS-1652是一种阴离子电导抑制剂。
1434639-57-2 | ND-646
(Catalog# : 191102)
ND-646是ACC酶ACC1和ACC2的变构抑制剂,可阻止ACC亚基二聚化,在体内
1434635-54-7 | ND-630
(Catalog# : 19133)
ND-630,也称为GS-0976, NDI-010976和firsocostat, 是一种有效的ACC抑制剂。
1448232-80-1 | Naquotinib游离
(Catalog# : 1812297)
Naquotinib,又称ASP8273,是一种口服、不可逆、第三代、突变选择、
1208315-24-5 | N6022
(Catalog# : 1811304)
N6022是一种有效、选择性、可逆性和有效性的s -亚硝基谷胱甘肽还
1253584-84-7 | NMS-E973
(Catalog# : 1810293)
NMS-E973是一种新型、选择性和强效的热休克蛋白90 (Hsp90)抑制剂。
153587-01-0 | NS1619
(Catalog# : 1810227)
NS1619是一种Bkca开启工具或大电导Ca2+活化钾(Bkca, KCa1.1)通道激活器
1452458-86-4 | Nacubactam
(Catalog# : 185169)
Nacubactam, 也称为RG-6080, FPI-1459, 和OP-0595, 是一种β-内酰胺酶抑制剂
108852-90-0 | Nemorubicin
(Catalog# : 185167)
Nemorubicin,又名PNU152243A,是一种不同于其母体药物的doxorubicin衍生
152946-68-4 | Nolatrexed盐酸盐
(Catalog# : 185166)
Nolatrexed,也叫AG337,是一种具有潜在抗癌活性的胸腺嘧啶合成酶抑
1773489-72-7 | Nidufexor
(Catalog# : 184288)
Nidufexor是一个法呢醇X受体(FXR)激动剂。
1422144-42-0 | Netarsudil(Mesylate)
(Catalog# : 712181)
Netarsudil( AR-11324) is a Rho-associated protein kinase inhibitor. Netarsudil is pot
1140844-63-8 | nor-NOHA醋酸盐
(Catalog# : 1710169)
nor-NOHA是一种强效、选择性、竞争性、以及精氨酸酶的高亲和力抑
1262417-51-5 | NMS-P118
(Catalog# : 17101311)
NMS-P118是一种有效的、可口服、高选择性PARP-1抑制剂具有优良的AD
1508250-71-2 | Nazartinib (EGF816)
(Catalog# : 1781004)
Nazartinib,也被称为EGF816,是一种口服可用,不可逆转的、第三代、
1254032-66-0 | Netarsudil
(Catalog# : 1781001)
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1676893-24-5 | NSC781406
(Catalog# : 20178810)
NSC781406是一种高效针对PI3K的IC50为2 nM的PI3K和mTOR抑制剂。
1916571-90-8 | NCT-503
(Catalog# : 2017888)
NCT-503是一种3 -磷酸甘油酸脱氢酶(PHGDH)抑制剂,抑制丝氨酸合成3 -磷
1304630-27-0 | NGP-555
(Catalog# : 2017875)
NGP 555正在被作为一种预防疾病老年痴呆症的治疗。
147149-76-6 | 诺拉曲特
(Catalog# : 17030908)
诺拉曲特,也叫AG337,是一种具有潜在抗癌活性的百里香酶抑制剂
1221713-92-3 | NPS-1034
(Catalog# : 17030907)
NPS-1034是一种新型的MET抑制剂,它能抑制活化的MET受体及其具有结
1400-61-9 | 制霉菌素
(Catalog# : 17030905)
制霉菌素是一种多烯抗真菌药物,含有三种生物活性成分的抗生素
1354744-91-4 | 聚乙二醇纳诺醇
(Catalog# : 17030202)
Naloxegol,也称为NKTR-118和AZ-13337019,是一种选择性的阿片拮抗剂,用于
1038915-64-8 | 尼拉帕尼盐酸盐
(Catalog# : 17030114)
尼拉帕尼, 也称为MK-4827, 是一种具有潜在抗肿瘤活性的聚(ADP-核糖
1698878-14-6 | Nampt-IN-1
(Catalog# : 17022705)
Nampt-IN-1是NAMPT的一种新型抑制剂,IC50分别为18 nM(NCI- H1155细胞),4
102586-30-1 | NSC12
(Catalog# : 17021317)
NSC12是一种可用于抑制FGF2 / FGFR相互作用并具有良好的抗肿瘤活性
123653-11-2 | NS-398 (NS398)
(Catalog# : 17011106)
NS-398是一种cyclooxygenase-2 (COX-2)的选择性抑制剂。
1253952-02-1 | Netarsudil (AR-13324) 2HCl
(Catalog# : 1710901)
Netarsudil (a.k.a. AR-13324)是一种ROCK抑制剂,Ki值为 0.2-10.3 nM。它目前
1313363-54-0 | NVP-CGM097
(Catalog# : 16122789)
NVP-CGM097 is a highly potent and selective MDM2 inhibitor. It binds to the p53 bindi
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
-- PROTAC
----
Molecular Glues
--
Antibody-drug Conjugate/ADC Related
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2102501-84-6 | PF-06835919 ( MDK-1846 )
(Catalog# : 193264)
MDK1846是一种强效的酮己糖激酶(KHK)抑制剂。
2671128-05-3 | FHD-286
(Catalog# : 20471)
FHD-286 is an oral, small-molecule, selective, allosteric inhibitor of BRG1 and BRM i
3002056-30-3 | NST-628
(Catalog# : 24058)
NST-628 是具有血脑屏障渗透性的 MAPK 通路分子胶,能够抑制 RAF 磷
2893778-31-7 | PHGDH-IN-3
(Catalog# : 25077)
PHGDH-IN-3 is an orally active phosphoglycerate dehydrogenase (PHGDH) inhibitor.
2882165-79-7 | CFT1946
(Catalog# : 25078)
CFT1946 是一种口服生物可利用的小分子降解剂,可降解实体瘤中的
68238-36-8 | 异硫蓝
(Catalog# : 178017)
Isosulfan blue 是一种用于淋巴管造影中淋巴管识别的蓝色染料。Isos
2803470-63-3 | HC-7366
(Catalog# : 25076)
HC-7366 is a potent and selective activator of the general control nonderepressible 2
2226636-04-8 | Soquelitinib ( CPI-818 )
(Catalog# : 20671)
Soquelitinib(CPI-818)是一种高度选择性的共价白细胞介素-2诱导的T
2230263-60-0 | Crelosidenib
(Catalog# : 24101)
Crelosidenib is an isocitrate dehydrogenase 1 (IDH1) inhibitor. It is an antineoplast
1260247-42-4 | LLL12
(Catalog# : 25075)
LLL12 is a potent STAT3 inhibitor. LLL12 inhibits colony formation and cell migration