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抑制剂/受体激动剂
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Metabolism
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Deuterated
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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
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Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
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Chiral Compounds
Deuterated
Fluorides
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Iodos
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Oxazoles
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Pyrimidines
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Cas号索引 1
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Cas号索引 1
1246964-32-8 | CLEFMA
(Catalog# : 615201)
CLEFMA has anti-proliferative activity in H441 cells. CLEFMA may induce autophagic ce
145915-58-8 | CGP52411
(Catalog# : 2061306)
CGP52411, also known as DAPH, is a selective inhibitor of the epidermal growth factor
199735-88-1 | CADD522
(Catalog# : 2051505)
CADD522 is a potent inhibitor of runt-related transcription factor-2 (RUNX2)-DNA bind
1010100-07-8 | CC-885
(Catalog# : 2041501)
CC-885 is a potent Cereblon Modulator with potent antitumor activity mediated through
1713240-67-5 | CM4620
(Catalog# : 204504)
CM4620是一种选择性的Orai1抑制剂,可防止Ca2 +进入腺泡细胞。CM4620
1860875-51-9 | CC-90009
(Catalog# : 203071)
CC-90009 是一种 cereblon (CRBN) E3 连接酶调节剂。CC-90009 与 CRBN 特异性
189746-19-8 | 5-氯-2,6-二甲氧基-4-甲基喹啉
(Catalog# : 4281903)
5-氯-2,6-二甲氧基-4-甲基喹啉是一个他非诺喹原料药合成中非常关
1181083-81-7 | CLP-290
(Catalog# : 193286)
CLP-290是一种新型的KCC2调制器和CLP-257的前药,对KCC2相关的Cl-转运
1802632-22-9 | CT-1812
(Catalog# : 193283)
CT-1812是一类口服的sigma-2/PGRMC1拮抗剂(α-β-低聚物受体拮抗剂),目
1384860-29-0 | Conteltinib
(Catalog# : 19342)
Conteltinib是一种酪氨酸激酶抑制剂和抗肿瘤药。
1358099-18-9 | C25-140
(Catalog# : 192274)
C25-140是环-E3连接酶(TRAF6) / E2酶(Ubc13)结合的一级蛋白-蛋白相互作用
1095382-05-0 | CCT-137690
(Catalog# : 192192)
CCT137690是一种极光激酶抑制剂CCT137690,是一种高选择性的口服生物
1418274-28-8 | Cilofexor ( GS-9674 )
(Catalog# : 19132)
Cilofexor(也称为 GS-9674)是一种非甾体法尼醇 X 受体(FXR)激动剂
1402709-93-6 | CCT241736
(Catalog# : 1812283)
CCT241736是一种有效且具有口服活性的日常FLT3-Aurora抑制剂。
1801343-74-7 | CA-4948
(Catalog# : 1811292)
CA-4948是一种生物活性化学物。
192322-50-2 | CGP-71683A盐酸盐
(Catalog# : 18792)
CGP 71683A是一种有效且高选择性的NPY Y(5)受体的非肽拮抗剂,在肥胖
1437321-24-8 | CEP-40783
(Catalog# : 186281)
CEP-40783,又称RXDX-106,是AXL和c-Met的一种有效、选择性和口服的抑
125316-60-1 | CD437
(Catalog# : 185316)
CD437合成维生素a是一个RARγ-selective受体激动剂。
1345810-21-0 | CB-1158
(Catalog# : 185315)
CB-1158,又称INCB01158,是一种有效的精氨酸酶抑制剂。
153259-65-5 | 西洛司特
(Catalog# : 185291)
西洛司特是一种用于治疗呼吸系统疾病,如哮喘和慢性阻塞性肺病
1276105-89-5 | CNX-1351
(Catalog# : 185174)
CNX-1351是PI3K的选择性共价抑制剂。
164658-13-3 | CGP60474
(Catalog# : 185171)
CGP60474是一种有效的双cdk1/cdk2抑制剂(IC50值分别为20和50 nM)。
1190932-38-7 | COH29
(Catalog# : 184127)
COH29是一种可口服的、芳香的取代噻唑和人核糖核苷酸还原酶(RNR)
1039455-84-9 | COTI-2
(Catalog# : 184320)
COTI-2是P53基因调制器和AKT2抑制剂。OTI-2在体外和体内都对多种人类
1202402-40-1 | CPI-444
(Catalog# : 18439)
CPI-444,又名V81444,是一种腺苷A2A受体的口服拮抗剂。
1443437-74-8 | CCG-203971
(Catalog# : 18437)
CCG-203971是前列腺癌细胞系PC-3中SRE活化的抑制剂(IC50 = 6.4 μM),能够
175140-00-8 | CP-376395 free base
(Catalog# : 184213)
CP-376395 is a CRF1-selective antagonist. CRF1 receptor signaling regulates food and
1402152-13-9 | Copanlisib HCl
(Catalog# : 18351)
Copanlisib也称为BAY 80 - 6946,是一个强有力的磷酸肌醇3-激酶(PI3K)抑制
19608-29-8 | CB-03-01
(Catalog# : 1712153)
CB-03-01, also known as cortexolone 17alpha-propionate, is a topical and peripherally
1797989-42-4 | CHIR99021 HCl
(Catalog# : 179825)
CHIR99021,又被称为 CT99021,是糖原合成酶激酶3β(GSK3β)抑制剂,
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2365193-22-0 | Zelasudil
(Catalog# : 24014)
Zelasudil 是一种有效的、高选择性的口服活性抑制剂,针对 Rho 相关
2134675-36-6 | Ziftomenib ( KO-539 )
(Catalog# : 24013)
Ziftomenib 是一种口服、有效、选择性的小分子抑制剂,针对 menin 和
1640282-42-3 | Zunsemetinib
(Catalog# : 24012)
Zunsemetinib是一种在研口服丝裂原活化蛋白激酶活化蛋白激酶2(MK2
2728667-27-2 | Zongertinib ( BI 1810631 )
(Catalog# : 24011)
Zongertinib [BI 1810631] 是一种人表皮生长因子受体 2 (HER2) 抑制剂。
2272904-53-5 | Zasocitinib
(Catalog# : 24010)
Zasocitinib是一种作用于非受体酪氨酸蛋白激酶 (TYK2)靶点的抑制
2503036-46-0 | RNK-05047
(Catalog# : 24008)
RNK-05047 为BRD4降解剂,其在小鼠荷瘤异种移植模型中展现出显著抑
1001288-58-9 | Asengeprast (FT011)
(Catalog# : 24009)
Asengeprast (FT011) 是一种抗纤维化剂,降低胶原蛋白 I 和 III 的 mRNA
2490431-16-6 | ERAS-801 ( JGK-068S )
(Catalog# : 20635)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。
209746-59-8 | T-1095
(Catalog# : 24004)
T-1095 is a potent and selective inhibitor of Na+-glucose cotransporters (SGLTs).
2739866-40-9 | NVL-655 ( ALK-IN-27 )
(Catalog# : 24003)
NVL-655是一种新型脑渗透性ALK选择性抑制剂,旨在解决目前可用的