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+86-17702719238
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抑制剂/受体激动剂
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Anti-infection
Apoptosis
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Cas号索引 1
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Cas号索引 1
1034442-21-1 | Basimglurant
(Catalog# : 187121)
Basimglurant,又称RO 4917523和RG-7090,是一种新型的mGlu5阴性变构调制
1923833-60-6 | BMS-986205
(Catalog# : 185314)
BMS-986205是一种抗癌药物。
1260251-31-7 | Birinapant
(Catalog# : 185182)
Birinapant,也被称为TL32711,是一种合成的小分子,具有潜在的抗肿
1286279-29-5 | BMS-813160
(Catalog# : 1842812)
BMS-813160是一种有效的选择性CCR2/CCR5拮抗剂,具有潜在的免疫调节
198480-56-7 | 盐酸巴多昔芬
(Catalog# : 18496)
Bazedoxifene,又名WAY-140424,是第三代选择性雌激素受体调节剂(SERM)
1513879-21-4 | BQR695
(Catalog# : 184218)
BQR695, also known as NVP-BQR695, is a potent and selective PI4K inhibitor.
1414943-88-6 | BAY1143572
(Catalog# : 181242)
Atuveciclib, also known as BAY1143572, is a highly selective, potent and orally avail
1803274-65-8 | BAY-1436032
(Catalog# : 181181)
BAY-1436032是一个强有力的,有选择性的,有效的突变异柠檬酸脱氢酶
1446090-77-2;1446090-79-4 | BGB-283
(Catalog# : 17101620)
BGB-283,也称为Beigene-283或Lifirafenib,是一种新的有效的和选择性的
1357920-84-3 | Belizatinib
(Catalog# : 17101619)
Belizatinib,也称为TSR-011,具有受体酪氨酸激酶间变性淋巴瘤激酶(
1420071-30-2 | Bioymifi
(Catalog# : 1710165)
Bioymifi是DR5的活性剂(Kd = 1.2 µM; IC50 = 2 µM). Bioymifi诱导凋亡的肿瘤
1707289-21-1 | BLU-554
(Catalog# : 1710162)
BLU-554是针对肝癌治疗的成纤维细胞生长因子受体4(FGFR4)抑制剂
1632118-69-4 | BAR-501
(Catalog# : 179821)
BAR-501是一种选择性GPBAR1激动剂,没有任何的FXR激动剂活性。BAR-50
1207293-36-4 | BI-847325
(Catalog# : 83101)
BI-847325是一种口服、具有选择性的日常生物MEK/Aurora激酶抑制剂,
1906919-67-2 | BAY-598
(Catalog# : 17982)
BAY-598是一种强效的针对SMYD2中肽-竞争的化学探测器。BAY-598拥有一
1906920-28-2 | BAY-598 R-异构体
(Catalog# : 17981)
BAY-598 R-异构体是BAY589 R-异构体。bay-598 R-异构体可以作为一个参照
171655-91-7 | 布索芬新
(Catalog# : 17916)
布索芬新是一种充分的单胺再摄取阻滞剂,已被开发用于治疗帕金
1290541-46-6 | B02
(Catalog# : 1783013)
B02,也叫RAD51 - in - 02,是一种RAD51抑制剂。B02能增强MM细胞的DOX敏
1703793-34-3 | BLU-285
(Catalog# : 1781003)
BLU-285是一种有效、具有选择性的抑制剂。
1876467-74-1 | BAY-1895344
(Catalog# : 1781002)
BAY-1895344是一种有效的、具有选择性的ATM抑制剂。
1263871-36-8 | BMS-932481
(Catalog# : 2017877)
BMS-932481调节Aβ肽在血浆和脑脊液的健康志愿者。
1334493-07-0 | BP-1-102
(Catalog# : 17030606)
BP-1-102是一种有效的口服生物和选择性抑制剂。
1799753-84-6 | BAY-876
(Catalog# : 17030604)
BAY-876是一种有效的、选择性的谷氨酸抑制剂。BAY- 876在体外具有良
1137359-47-7 | BRD-7552
(Catalog# : 17030312)
BRD-7552是一种PDX1转录诱导因子。它主要在人类胰岛和导管细胞中调
1821496-27-8 | BDA-366
(Catalog# : 17030305)
BDA - 366是BCL - BH4拮抗剂。BDA - 366抑制人骨髓瘤的生长。BDA - 366诱导
1225037-39-7 | Bimiralisib
(Catalog# : 17030116)
Bimiralisib,也被称为PQR309,是一种口服生物可用的磷脂- 3 -激酶抑
1197953-54-0 | Brigatinib (AP-26113)
(Catalog# : 16122905)
Brigatinib, also known as AP-26113, is an orally active, potent and selective Dual AL
189232-42-6 | Bohemine
(Catalog# : 16122903)
Bohemine is a potent and selective, cell-permeable, cyclin-dependent kinase (CDK) inh
1000998-59-3 | BMS-687453
(Catalog# : 16122902)
BMS-687453 is a potent and selective peroxisome proliferator activated receptor (PPAR
130370-60-4 | Batimastat
(Catalog# : 16122804)
Batimastat (also known as BB-94) is a synthetic matrix metalloproteinase inhibitor th
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产品分类
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-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
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----
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----
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----
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----
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----
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----
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----
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----
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----
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----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
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Sphingosine 1 Phosphate Receptor
----
PKA
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Adenosine Receptor
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GnRH
----
LPL Receptor
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Ras
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Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
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ChoKα
----
Newest added products
抑制剂/受体激动剂
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分子砌块
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新产品
天然化合物
最新产品
2750001-23-9 | AZD0095
(Catalog# : 237072)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2101538-28-5 | 2-MNG
(Catalog# : 24129)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
2439277-80-0 | MAT2A-IN-9
(Catalog# : 25147)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
1898206-17-1 | Safusidenib
(Catalog# : 25149)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
2669009-92-9 | Atebimetinib
(Catalog# : 25148)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
2242751-53-5 | Acoramidis hydrochloride
(Catalog# : 24068)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
2230263-60-0 | Crelosidenib
(Catalog# : 24101)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
2833703-74-3 | LOXO-435
(Catalog# : 25080)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
2446928-30-7 | Gridegalutamide
(Catalog# : 25138)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
1256349-48-0 | Chiauranib
(Catalog# : 25146)
Chiauranib also known as orally available, small molecule inhibitor of select serine-