武汉永璨生物科技有限公司
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抑制剂/受体激动剂
Angiogenesis
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
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Amino Acids
Anilines
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Bromides
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Deuterated
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Indoles and Oxindoles
Iodos
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Oxazoles
Peg Linkers
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Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
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Other Azoles
Other Heterocycles
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On Sale
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定制合成
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产品名字索引 H
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产品名字索引 H
H 151
(Catalog# : 1811022, Cas# :
941987-60-6
)
H 151是一种诱捕拮抗剂,共价结合在Cys91上,阻断棕榈酰化和防止
HC-056456
(Catalog# : 1810171, Cas# :
7733-96-2
)
HC-056456是CatSper的通道调制器。
20-HETE
(Catalog# : 185283, Cas# :
79551-86-3
)
20-HETE是一种细胞色素P450 (CYP450)代谢产物,在脑血管和肾血管中扮
HMN-154
(Catalog# : 184122, Cas# :
173528-92-2
)
HMN-154是一种苯磺胺的抗癌剂。HMN-154通过剂量依赖性的方式抑制NF
HJC0152
(Catalog# : 1710133, Cas# :
1420290-99-8
)
HJC0152是对人的头部和颈部鳞状细胞癌(鳞癌)的信号转导与转录
9-Hydroxyellipticin(free base)
(Catalog# : 1791313, Cas# :
51131-85-2
)
9-hydroxyellipticine,又名 IGIG 929和LS133324,是一种强效的细胞毒和抗
H3B-6527
(Catalog# : 179822, Cas# :
1702259-66-2
)
H3B-6527是一个强有力的口服活性分子抑制剂,具有潜在的抗肿瘤活
1H-吡唑并[3,4-C]吡啶
(Catalog# : 1781503, Cas# :
271-47-6
)
1H-吡唑并[3,4-C]吡啶,1H-pyrazolo[3,4-c]pyridine
H-89盐酸盐
(Catalog# : 178815, Cas# :
130964-39-5
)
H-89是一种特殊的腺苷酸环酶抑制剂(DDA),是一种循环的氨依赖性蛋
HDM201
(Catalog# : 2017872, Cas# :
1448867-41-1
)
HDM201是一种口服生物利用率在人的同源基因(HDM2)抑制剂。具有潜在
HM-61713 (BI-1482694)
(Catalog# : 17022709, Cas# :
1802181-20-9
)
BI-1482694是布鲁顿酪氨酸激酶(BTK)的一种有效的小分子抑制剂。
5-羟基吡嗪-2-羧酸
(Catalog# : 17021403, Cas# :
34604-60-9
)
5-羟基吡嗪-2-羧酸, 一种抗结核药物吡嗪酰胺(PZA)的代谢物。
Hesperadin
(Catalog# : 17011902, Cas# :
422513-13-1
)
Hesperadin是人类Aurora B的一种抑制剂,它可以阻止IC(50)为40 nM的基质
HLCL-61 HCl
(Catalog# : 16122819, Cas# :
1158279-20-9
)
HLCL-61 is a potent and selective PRMT5 inhibitor for treatment of acute myeloid leuk
Hexaminolevulinate HCl
(Catalog# : 16122818, Cas# :
140898-91-5
)
Hexaminolevulinate hydrochloride, also known as hexyl 5-aminolevulinate HCl, is the h
HA15
(Catalog# : 16122816, Cas# :
1609402-14-3
)
HA15 displayed anti-cancerous activity on all melanoma cells tested, including cells
Honokiol
(Catalog# : 161009024, Cas# :
35354-74-6
)
Houpu has traditionally been used in Eastern medicine as analgesic and to treat anxie
HS-173
(Catalog# : 161009001, Cas# :
1276110-06-5
)
HS-173 inhibited the PI3K signaling pathway, and showed anti-proliferative effects on
HUHS015
(Catalog# : 16062902, Cas# :
1453097-13-6
)
HUHS015 is a potent PCA-1/ALKBH3 inhibitor both in vitro and in vivo. The bioavailabi
HLCL-61
(Catalog# : 16062204, Cas# :
586395-74-6
)
HLCL-61 is a potent and selective PRMT5 inhibitor for treatment of acute myeloid leuk
1H-Pyrrolo[2,3-B]Pyridine-3-Carboxylic Acid
(Catalog# : 032511, Cas# :
156270-06-3
)
Coming soon!
1H-Indazole-5-boronic acid
(Catalog# : 032503, Cas# :
338454-14-1
)
Coming soon!
HTH-01-015
(Catalog# : 011306, Cas# :
1613724-42-7
)
HTH-01-015 is a potent and selective inhibitor of NUAK1 with IC50 of 100 nM, does not
hydrocortisone
(Catalog# : 010402, Cas# :
50-23-7
)
Hydrocortisone is the main glucocorticoid secreted by the ADRENAL CORTEX. Its synthet
HQL-79
(Catalog# : 121507, Cas# :
162641-16-9
)
Coming soon!
HBED-CC-PSMA ( PSMA-11 )
(Catalog# : 103003, Cas# :
1366302-52-4
)
PSMA-11, also known as HBED-CC-PSMA or Psma-hbed-CC, has potential use as a tracer fo
HBED-CC
(Catalog# : 103002, Cas# :
143557-99-7
)
Coming soon!
6-hydroxy-N-Methylbenzofuran-3-carboxaMide
(Catalog# : 92218)
Coming soon!
7-hydroxy-1H-quinolin-2-one
(Catalog# : 91706, Cas# :
70500-72-0
)
Coming soon!
3-(4-Hydroxyphenyl)propionic acid
(Catalog# : 90608, Cas# :
501-97-3
)
Coming soon!
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
ECI830
(Catalog# : 26A031, Cas# :
3054692-62-2
)
ECI830是一种实验性的CDK2抑制剂。
GNE-317
(Catalog# : 52282, Cas# :
1394076-92-6
)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
DPTX-3186
(Catalog# : 26A010, Cas# :
3118994-80-9
)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108, Cas# :
435327-40-5
)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
Iclepertin (BI-425809)
(Catalog# : 24084, Cas# :
1421936-85-7
)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
Kartogenin ( KGN )
(Catalog# : 52215, Cas# :
4727-31-5
)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602, Cas# :
218791-21-0
)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
Apecotrep (BI 764198)
(Catalog# : 26A048, Cas# :
2311863-36-0
)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
BH-30643
(Catalog# : 26A047, Cas# :
3062177-59-4
)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制