武汉永璨生物科技有限公司
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抑制剂/受体激动剂
Angiogenesis
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Bromides
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Deuterated
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
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产品名字索引 H
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产品名字索引 H
20-HETE
(Catalog# : 185283, Cas# :
79551-86-3
)
20-HETE是一种细胞色素P450 (CYP450)代谢产物,在脑血管和肾血管中扮
HMN-154
(Catalog# : 184122, Cas# :
173528-92-2
)
HMN-154是一种苯磺胺的抗癌剂。HMN-154通过剂量依赖性的方式抑制NF
HJC0152
(Catalog# : 1710133, Cas# :
1420290-99-8
)
HJC0152是对人的头部和颈部鳞状细胞癌(鳞癌)的信号转导与转录
9-Hydroxyellipticin(free base)
(Catalog# : 1791313, Cas# :
51131-85-2
)
9-hydroxyellipticine,又名 IGIG 929和LS133324,是一种强效的细胞毒和抗
H3B-6527
(Catalog# : 179822, Cas# :
1702259-66-2
)
H3B-6527是一个强有力的口服活性分子抑制剂,具有潜在的抗肿瘤活
1H-吡唑并[3,4-C]吡啶
(Catalog# : 1781503, Cas# :
271-47-6
)
1H-吡唑并[3,4-C]吡啶,1H-pyrazolo[3,4-c]pyridine
H-89盐酸盐
(Catalog# : 178815, Cas# :
130964-39-5
)
H-89是一种特殊的腺苷酸环酶抑制剂(DDA),是一种循环的氨依赖性蛋
HDM201
(Catalog# : 2017872, Cas# :
1448867-41-1
)
HDM201是一种口服生物利用率在人的同源基因(HDM2)抑制剂。具有潜在
HM-61713 (BI-1482694)
(Catalog# : 17022709, Cas# :
1802181-20-9
)
BI-1482694是布鲁顿酪氨酸激酶(BTK)的一种有效的小分子抑制剂。
5-羟基吡嗪-2-羧酸
(Catalog# : 17021403, Cas# :
34604-60-9
)
5-羟基吡嗪-2-羧酸, 一种抗结核药物吡嗪酰胺(PZA)的代谢物。
Hesperadin
(Catalog# : 17011902, Cas# :
422513-13-1
)
Hesperadin是人类Aurora B的一种抑制剂,它可以阻止IC(50)为40 nM的基质
HLCL-61 HCl
(Catalog# : 16122819, Cas# :
1158279-20-9
)
HLCL-61 is a potent and selective PRMT5 inhibitor for treatment of acute myeloid leuk
Hexaminolevulinate HCl
(Catalog# : 16122818, Cas# :
140898-91-5
)
Hexaminolevulinate hydrochloride, also known as hexyl 5-aminolevulinate HCl, is the h
HA15
(Catalog# : 16122816, Cas# :
1609402-14-3
)
HA15 displayed anti-cancerous activity on all melanoma cells tested, including cells
Honokiol
(Catalog# : 161009024, Cas# :
35354-74-6
)
Houpu has traditionally been used in Eastern medicine as analgesic and to treat anxie
HS-173
(Catalog# : 161009001, Cas# :
1276110-06-5
)
HS-173 inhibited the PI3K signaling pathway, and showed anti-proliferative effects on
HUHS015
(Catalog# : 16062902, Cas# :
1453097-13-6
)
HUHS015 is a potent PCA-1/ALKBH3 inhibitor both in vitro and in vivo. The bioavailabi
HLCL-61
(Catalog# : 16062204, Cas# :
586395-74-6
)
HLCL-61 is a potent and selective PRMT5 inhibitor for treatment of acute myeloid leuk
1H-Pyrrolo[2,3-B]Pyridine-3-Carboxylic Acid
(Catalog# : 032511, Cas# :
156270-06-3
)
Coming soon!
1H-Indazole-5-boronic acid
(Catalog# : 032503, Cas# :
338454-14-1
)
Coming soon!
HTH-01-015
(Catalog# : 011306, Cas# :
1613724-42-7
)
HTH-01-015 is a potent and selective inhibitor of NUAK1 with IC50 of 100 nM, does not
hydrocortisone
(Catalog# : 010402, Cas# :
50-23-7
)
Hydrocortisone is the main glucocorticoid secreted by the ADRENAL CORTEX. Its synthet
HQL-79
(Catalog# : 121507, Cas# :
162641-16-9
)
Coming soon!
HBED-CC-PSMA ( PSMA-11 )
(Catalog# : 103003, Cas# :
1366302-52-4
)
PSMA-11, also known as HBED-CC-PSMA or Psma-hbed-CC, has potential use as a tracer fo
HBED-CC
(Catalog# : 103002, Cas# :
143557-99-7
)
Coming soon!
6-hydroxy-N-Methylbenzofuran-3-carboxaMide
(Catalog# : 92218)
Coming soon!
7-hydroxy-1H-quinolin-2-one
(Catalog# : 91706, Cas# :
70500-72-0
)
Coming soon!
3-(4-Hydroxyphenyl)propionic acid
(Catalog# : 90608, Cas# :
501-97-3
)
Coming soon!
6-Hydroxy-1-indanone
(Catalog# : 81930, Cas# :
62803-47-8
)
Coming soon!
2H-Isoindole-1-carboxylic acid methyl ester
(Catalog# : 81003, Cas# :
56365-71-0
)
Coming soon!
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AZD0095
(Catalog# : 237072, Cas# :
2750001-23-9
)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2-MNG
(Catalog# : 24129, Cas# :
2101538-28-5
)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
MAT2A-IN-9
(Catalog# : 25147, Cas# :
2439277-80-0
)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
Acoramidis hydrochloride
(Catalog# : 24068, Cas# :
2242751-53-5
)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
Crelosidenib
(Catalog# : 24101, Cas# :
2230263-60-0
)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
LOXO-435
(Catalog# : 25080, Cas# :
2833703-74-3
)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
Gridegalutamide
(Catalog# : 25138, Cas# :
2446928-30-7
)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
Chiauranib
(Catalog# : 25146, Cas# :
1256349-48-0
)
Chiauranib also known as orally available, small molecule inhibitor of select serine-