武汉永璨生物科技有限公司
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抑制剂/受体激动剂
Angiogenesis
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Apoptosis
Autophagy
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MAPK
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Metabolism
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分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
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Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
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产品名字索引 O
ONC212
(Catalog# : 185286, Cas# :
1807861-48-8
)
ONC212是一种氟化的ONC201类似物,在黑色素瘤和肝细胞癌模型中显示
Olcegepant
(Catalog# : 185285, Cas# :
204697-65-4
)
Olcegepant,又称BIBN-4096或BIBN-4096BS,是降钙素基因相关肽1 (CGRP1)受体
OPC-21268
(Catalog# : 185163, Cas# :
131631-89-5
)
OPC-21268是一种血管加压素1受体拮抗剂,可用于治疗心力衰竭和高
OSI-930
(Catalog# : 185162, Cas# :
728033-96-3
)
OSI-930是一种选择性的噻吩衍生物酪氨酸激酶抑制剂,具有潜在的
OTSSP167游离
(Catalog# : 185161, Cas# :
1431697-89-0
)
OTSSP167,也被称为OTS167,是一种口服有效的抑制母胚胎亮氨酸拉链
Olodanrigan游离酸
(Catalog# : 1842810, Cas# :
1316755-16-4
)
Olodanrigan,又称EMA-401和PD-126055,是一种血管紧张素AT2拮抗剂,可用
OSS-128167
(Catalog# : 184214, Cas# :
887686-02-4
)
OSS-128167, also known as SIRT6-IN-1, is a potent and selective SIRT 6 inhibitor.
Osimertinib mesylate
(Catalog# : 1712154, Cas# :
1421373-66-1
)
Osimertinib, also known as mereletinib and AZD-9291, is a third-generation EGFR inhib
醋酸催产素
(Catalog# : 1791513, Cas# :
6233-83-6
)
催产素是一种药物和激素。作为一种药物,它被用来引起子宫收缩
ON1231320
(Catalog# : 1791319, Cas# :
131247-39-8
)
ON1231320,也称为GBO-006,是Plk2抑制剂。
盐酸奥达特罗
(Catalog# : 179824, Cas# :
869477-96-3
)
盐酸奥达特罗,也称为BI 1744,是一种长效β受体激动剂用于患者吸
奥扎莫德
(Catalog# : 110902, Cas# :
1306760-87-1
)
奥扎莫德是一种选择性的鞘氨醇1磷酸受体调节剂和方法,可能在
奥莫替尼
(Catalog# : 011103, Cas# :
1353550-13-6
)
奥莫替尼是一种有效的布鲁顿酪氨酸激酶(BTK)小分子抑制剂。
OXi-4503钠
(Catalog# : 178308, Cas# :
288847-34-7
)
OXi-4503是一种二磷酸酯类药物,开始是从植物纤维中分离出来的,
6-氧杂螺[4.5]癸烷-9-醇
(Catalog# : 20177315, Cas# :
855398-58-2
)
6-氧杂螺[4.5]癸烷-9-醇|6-Oxaspiro[4.5]decan-9-ol|15080-A1
Olumacostat Glasaretil
(Catalog# : 732801, Cas# :
1261491-89-7
)
Olumacostat glasaretil是一种新型的用于痤疮治疗的局部皮脂抑制剂。
OTS514
(Catalog# : 17031015, Cas# :
1338540-63-8
)
OTS514是一种高效的TOPK(T-LAK胞起源蛋白激酶)抑制剂,IC50值为2.6 nM。
奥马曲拉
(Catalog# : 17030903, Cas# :
167305-00-2
)
奥马曲拉是一种新型的抗高血压药,可抑制中性内肽酶(NEP)和血管
ON-013100
(Catalog# : 17030902, Cas# :
865783-95-5
)
ON-013100是一种细胞周期抑制剂,对治疗地幔细胞淋巴瘤有潜在的作
ONT-093
(Catalog# : 17030901, Cas# :
216227-54-2
)
ONT-093, 也称为OC-144-093,是一种口服的P-糖蛋白泵抑制剂,用于治疗
催产素
(Catalog# : 17030805, Cas# :
50-56-6
)
催产素是一种药物和荷尔蒙。作为一种药物,它被用来引起子宫收
Orteronel (外消旋)
(Catalog# : 17030610, Cas# :
426219-18-3
)
Orteronel(外消旋)是s - Orteronel和r - Orteronel异构体的混合物。Orteronel
奥巴克拉
(Catalog# : 17022707, Cas# :
803712-79-0
)
奥巴克拉对Bcl-xL细胞系中的缺乏表现出较低敏感。在 Mcl-1, Bcl-2,和
Org-26576
(Catalog# : 17021328, Cas# :
1026791-61-6;100044-96-0
)
Org-26576是一种AMPA谷氨酸受体调制器,可能用于治疗抑郁症和注意
氧化白藜芦醇
(Catalog# : 17021324, Cas# :
29700-22-9
)
氧化白藜芦醇,一种天然存在的化合物,尤其在Morus alba L中发现。
ONO-7300243
(Catalog# : 16122724, Cas# :
638132-34-0
)
ONO-7300243 is a novel, potent LPA1(Lysophosphatidic Acid Receptor) antagonist with a
Oxolinic acid
(Catalog# : 16122720, Cas# :
14698-29-4
)
Oxolinic acid is a quinolone antibiotic, inhibiting the enzyme DNA gyrase and DNA syn
ON123300
(Catalog# : 16122712, Cas# :
1357470-29-1
)
ON123300 is a potent and multi-targeted kinase inhibitor with IC50 of 3.9 nM, 5 nM, 2
Oclacitinib
(Catalog# : 16122705, Cas# :
1640292-55-2
)
Oclacitinib is a novel inhibitor of JAK family members with IC50 ranging from 10 to 9
Opicapone
(Catalog# : 6111514, Cas# :
923287-50-7
)
Opicapone(BIA 9-1067) is a long-acting, peripherally selective inhibitor of catechol-
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AZD0095
(Catalog# : 237072, Cas# :
2750001-23-9
)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2-MNG
(Catalog# : 24129, Cas# :
2101538-28-5
)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
MAT2A-IN-9
(Catalog# : 25147, Cas# :
2439277-80-0
)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
Acoramidis hydrochloride
(Catalog# : 24068, Cas# :
2242751-53-5
)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
Crelosidenib
(Catalog# : 24101, Cas# :
2230263-60-0
)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
LOXO-435
(Catalog# : 25080, Cas# :
2833703-74-3
)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
Gridegalutamide
(Catalog# : 25138, Cas# :
2446928-30-7
)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
Chiauranib
(Catalog# : 25146, Cas# :
1256349-48-0
)
Chiauranib also known as orally available, small molecule inhibitor of select serine-