武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
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产品名字索引 E
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产品名字索引 E
E2012
(Catalog# : 1810231, Cas# :
870843-42-8
)
E2012是γ-secretase分泌酶调制器(GSM)。
EBI-2511
(Catalog# : 1810165, Cas# :
2098546-05-3
)
EBI-2511是非霍奇金淋巴瘤有效的口服活性EZH2抑制剂。
Entasobulin
(Catalog# : 186293, Cas# :
501921-61-5
)
Entasobulin是一种β-tubulin聚合抑制剂,具有潜在的抗癌活性。
环氧丙烷D
(Catalog# : 186292, Cas# :
189453-10-9
)
环氧丙烷D是从纤维素粘液杆菌中分离出来的一种天然聚酮化合物
EZM2302
(Catalog# : 186272, Cas# :
1628830-21-6
)
EZM2302是一种有效的,选择性的,可口服的精氨酸甲基转移酶CARM1抑
依沙替康甲磺酸盐
(Catalog# : 186271, Cas# :
169869-90-3
)
依沙替康也叫DX 8951,是一种半合成的水溶性喜树碱衍生物,具有
艾菲康唑
(Catalog# : 186213, Cas# :
164650-44-6
)
艾菲康唑是一种三唑类抗真菌药。它被批准用于加拿大和美国作为
Erteberel
(Catalog# : 186157, Cas# :
533884-09-2
)
Erteberel,也称为LY500307,选择性雌激素受体β受体激动剂(ERβ)是治疗良
Edonerpic maleate
(Catalog# : 18671, Cas# :
519187-97-4
)
Edonerpic,也被称为T-817,是一种神经保护剂。
内昔芬 E-异构体盐酸盐
(Catalog# : 184124, Cas# :
1197194-61-8
)
内昔芬 E-异构体是一种他莫昔芬的代谢物和有效的选择性雌激素反
Ensartinib ( X396 )
(Catalog# : 184321, Cas# :
1370651-20-9
)
Ensartinib is an orally available small molecule inhibitor of the receptor tyrosine k
eCF506 ( 别名:NXP 900 )
(Catalog# : 18382, Cas# :
1914078-41-3
)
eCF506靶向一种叫做Src酪氨酸激酶的分子,这是乳腺癌细胞生长和传
Esaxerenone
(Catalog# : 1710121, Cas# :
1632006-28-0
)
Esaxerenone(cs-3150,xl-550)是一种非甾体类抗盐皮质激素Exelixis发现
EBE-A22
(Catalog# : 179831, Cas# :
229476-53-3
)
EBE-A22是PD 153035衍生物。EBE-A22,在EGF-R TK上无影响但保持高细胞毒
EPZ015666
(Catalog# : 011309, Cas# :
1616391-65-1
)
EPZ-015666 是一种强效、选择性的口服生物药,PRMT5抑制剂与Ki为5 nm
EED226
(Catalog# : 178311, Cas# :
2083627-02-3
)
EED226是一种强效、选择性抑制剂,口服生物EED抑制剂。在EZH2MUT临
厄达替尼(JNJ-42756493)
(Catalog# : 651701, Cas# :
1346242-81-6
)
Erdafitinib(JNJ-42756493) is a potent and selective panfibroblast growth factor recep
Ethyl 2-cyclohexyl-2-oxoacetate
(Catalog# : 178157, Cas# :
13275-31-5
)
Ethyl 2-cyclohexyl-2-oxoacetate
E7449
(Catalog# : 178903, Cas# :
1140964-99-3
)
E7449是一种可口服的小分子抑制剂,核酶聚(ADP-核糖)聚合酶(PARP)1和
Elenbecestat ( E2609 )
(Catalog# : 2017878, Cas# :
1388651-30-6
)
Elenbecestat是一种β-Site淀粉样前体蛋白裂解酶BACE)抑制剂,主要用
依托泊苷磷酸酯
(Catalog# : 20178213, Cas# :
117091-64-2
)
依托泊苷磷酸盐是一种半合成足叶草毒素的磷酸盐。
Elamipretide
(Catalog# : 20178210, Cas# :
736992-21-5
)
Elamipretide, 也称为MTP-131或D-Arg-Dmt-Lys-Phe-NH2,是一种心肌过氧化酶抑
[(1S)-2-(3,5-二氟苯基)-1-[(2S)-环氧乙烷基]乙基]氨基甲酸叔丁酯
(Catalog# : 20177314, Cas# :
388071-27-0
)
[(1S)-2-(3,5-二氟苯基)-1-[(2S)-环氧乙烷基]乙基]氨基甲酸叔丁酯
Etrasimod
(Catalog# : 17031018, Cas# :
1206123-37-6
)
Etrasimod,也被称为APD334,是一种多功能S1P1受体的功能拮抗剂,用
eFT-508
(Catalog# : 17031010, Cas# :
1849590-01-7
)
eFT-508 (eFT508)是一种有效且选择性的MNK1 / 2抑制剂,可能导致肿瘤细
盐酸Epetraborole
(Catalog# : 17022806, Cas# :
1234563-16-6
)
盐酸Epetraborole是一种新型的leucyl - trna合成酶(LeuRS)抑制剂。
依利格鲁司特
(Catalog# : 17022718, Cas# :
491833-29-5
)
依利格鲁司特, 也叫Genz-112638, 是一种有效的选择性的葡萄糖酰胺合
EX-527 S-enantiomer
(Catalog# : 17011802, Cas# :
848193-68-0
)
EX-527 S-enantiomer是一种有效的选择性SIRT1抑制剂,IC50为123 nM;没有对
EX-527 R-enantiomer
(Catalog# : 17011801, Cas# :
848193-69-1
)
EX-527 R-enantiomer是对活性形式EX-527 S-enantiomer(推测为参考)的负控制
4E1RCat
(Catalog# : 17011301, Cas# :
328998-25-0
)
4E1RCat是eIF4F翻译起始复合物的一种抑制剂,它阻止eIF4E:eIF4G和eIF4E
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AD-8007
(Catalog# : 26A018, Cas# :
1497439-74-3
)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
ZY-444
(Catalog# : 26A020, Cas# :
1802650-31-2
)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
AD-5584
(Catalog# : 26A019, Cas# :
2306525-79-9
)
AD-5584是一种新型脑渗透性ACSS2抑制剂。
IDB-003
(Catalog# : 26A017, Cas# :
3079716-11-0
)
IDB-003在体内抑制MDA-MB-231肿瘤生长。
Vafidemstat
(Catalog# : 18891, Cas# :
1357362-02-7
)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
LLL12
(Catalog# : 25075, Cas# :
1260247-42-4
)
LLL12是一种强效的STAT3抑制剂。LLL12在小鼠异种移植物模型中显示出
ECC-5004
(Catalog# : 26A015, Cas# :
2758659-09-3
)
ECC5004是一款每日一次、低剂量、小分子GLP-1受体激动剂。
SILA-123
(Catalog# : 26A014, Cas# :
2911585-37-8
)
SILA-123是一种II型FLT3抑制剂,对FLT3-WT(IC50=2.1 nM)和FLT3-ITD(IC50=1
Encaleret sulfate
(Catalog# : 26A013, Cas# :
1214922-52-7
)
Encaleret是一种正在研究的钙敏感受体的小分子拮抗剂,用于钙稳态
Iadademstat ( ORY-1001 ) hydrochloride
(Catalog# : 26A011, Cas# :
1431303-72-8
)
Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶