武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
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产品名字索引 E
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产品名字索引 E
环氧丙烷D
(Catalog# : 186292, Cas# :
189453-10-9
)
环氧丙烷D是从纤维素粘液杆菌中分离出来的一种天然聚酮化合物
EZM2302
(Catalog# : 186272, Cas# :
1628830-21-6
)
EZM2302是一种有效的,选择性的,可口服的精氨酸甲基转移酶CARM1抑
依沙替康甲磺酸盐
(Catalog# : 186271, Cas# :
169869-90-3
)
依沙替康也叫DX 8951,是一种半合成的水溶性喜树碱衍生物,具有
艾菲康唑
(Catalog# : 186213, Cas# :
164650-44-6
)
艾菲康唑是一种三唑类抗真菌药。它被批准用于加拿大和美国作为
Erteberel
(Catalog# : 186157, Cas# :
533884-09-2
)
Erteberel,也称为LY500307,选择性雌激素受体β受体激动剂(ERβ)是治疗良
Edonerpic maleate
(Catalog# : 18671, Cas# :
519187-97-4
)
Edonerpic,也被称为T-817,是一种神经保护剂。
内昔芬 E-异构体盐酸盐
(Catalog# : 184124, Cas# :
1197194-61-8
)
内昔芬 E-异构体是一种他莫昔芬的代谢物和有效的选择性雌激素反
Ensartinib ( X396 )
(Catalog# : 184321, Cas# :
1370651-20-9
)
Ensartinib is an orally available small molecule inhibitor of the receptor tyrosine k
eCF506 ( 别名:NXP 900 )
(Catalog# : 18382, Cas# :
1914078-41-3
)
eCF506靶向一种叫做Src酪氨酸激酶的分子,这是乳腺癌细胞生长和传
Esaxerenone
(Catalog# : 1710121, Cas# :
1632006-28-0
)
Esaxerenone(cs-3150,xl-550)是一种非甾体类抗盐皮质激素Exelixis发现
EBE-A22
(Catalog# : 179831, Cas# :
229476-53-3
)
EBE-A22是PD 153035衍生物。EBE-A22,在EGF-R TK上无影响但保持高细胞毒
EPZ015666
(Catalog# : 011309, Cas# :
1616391-65-1
)
EPZ-015666 是一种强效、选择性的口服生物药,PRMT5抑制剂与Ki为5 nm
EED226
(Catalog# : 178311, Cas# :
2083627-02-3
)
EED226是一种强效、选择性抑制剂,口服生物EED抑制剂。在EZH2MUT临
厄达替尼(JNJ-42756493)
(Catalog# : 651701, Cas# :
1346242-81-6
)
Erdafitinib(JNJ-42756493) is a potent and selective panfibroblast growth factor recep
Ethyl 2-cyclohexyl-2-oxoacetate
(Catalog# : 178157, Cas# :
13275-31-5
)
Ethyl 2-cyclohexyl-2-oxoacetate
E7449
(Catalog# : 178903, Cas# :
1140964-99-3
)
E7449是一种可口服的小分子抑制剂,核酶聚(ADP-核糖)聚合酶(PARP)1和
Elenbecestat ( E2609 )
(Catalog# : 2017878, Cas# :
1388651-30-6
)
Elenbecestat是一种β-Site淀粉样前体蛋白裂解酶BACE)抑制剂,主要用
依托泊苷磷酸酯
(Catalog# : 20178213, Cas# :
117091-64-2
)
依托泊苷磷酸盐是一种半合成足叶草毒素的磷酸盐。
Elamipretide
(Catalog# : 20178210, Cas# :
736992-21-5
)
Elamipretide, 也称为MTP-131或D-Arg-Dmt-Lys-Phe-NH2,是一种心肌过氧化酶抑
[(1S)-2-(3,5-二氟苯基)-1-[(2S)-环氧乙烷基]乙基]氨基甲酸叔丁酯
(Catalog# : 20177314, Cas# :
388071-27-0
)
[(1S)-2-(3,5-二氟苯基)-1-[(2S)-环氧乙烷基]乙基]氨基甲酸叔丁酯
Etrasimod
(Catalog# : 17031018, Cas# :
1206123-37-6
)
Etrasimod,也被称为APD334,是一种多功能S1P1受体的功能拮抗剂,用
eFT-508
(Catalog# : 17031010, Cas# :
1849590-01-7
)
eFT-508 (eFT508)是一种有效且选择性的MNK1 / 2抑制剂,可能导致肿瘤细
盐酸Epetraborole
(Catalog# : 17022806, Cas# :
1234563-16-6
)
盐酸Epetraborole是一种新型的leucyl - trna合成酶(LeuRS)抑制剂。
依利格鲁司特
(Catalog# : 17022718, Cas# :
491833-29-5
)
依利格鲁司特, 也叫Genz-112638, 是一种有效的选择性的葡萄糖酰胺合
EX-527 S-enantiomer
(Catalog# : 17011802, Cas# :
848193-68-0
)
EX-527 S-enantiomer是一种有效的选择性SIRT1抑制剂,IC50为123 nM;没有对
EX-527 R-enantiomer
(Catalog# : 17011801, Cas# :
848193-69-1
)
EX-527 R-enantiomer是对活性形式EX-527 S-enantiomer(推测为参考)的负控制
4E1RCat
(Catalog# : 17011301, Cas# :
328998-25-0
)
4E1RCat是eIF4F翻译起始复合物的一种抑制剂,它阻止eIF4E:eIF4G和eIF4E
Etomoxir钠盐
(Catalog# : 17011103, Cas# :
828934-41-4
)
Etomoxir是一种在线粒体内膜的外表面的一种不可逆转的CPT-1抑制剂
Eganelisib ( IPI-549 )
(Catalog# : 711401, Cas# :
1693758-51-8
)
Eganelisib (IPI-549) 是一种首创、口服、高选择性 PI3Kγ 抑制剂,单独
Ezutromid
(Catalog# : 16122944, Cas# :
945531-77-1
)
Ezutromid, also known as BMN-195 and SMTC-1100, is a first orally bioavailable utroph
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Dencatistat (STP938)
(Catalog# : 25177, Cas# :
2377000-84-3
)
Dencatistat 是一种口服生物可利用的小分子胞苷三磷酸合酶 1 (CTPS1)
DS-1001b
(Catalog# : 25178, Cas# :
1898207-64-1
)
DS-1001 是一种口服的脑渗透性突变 IDH1 选择性抑制剂。
Z57346765
(Catalog# : 25191, Cas# :
1016340-64-9
)
Z57346765 是一种 PGK1 特异性抑制剂,可降低 PGK1 糖酵解中代谢酶的
CBR-470-1
(Catalog# : 25192, Cas# :
2416095-06-0
)
CBR-470-1 是诱导 Nrf2 活性的糖酵解酶 PGK1 的抑制剂。
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
HC-7366
(Catalog# : 25076, Cas# :
2803470-63-3
)
HC-7366 is a potent and selective activator of the general control nonderepressible 2
Flavopiridol ( 夫拉平度 )
(Catalog# : 237071, Cas# :
146426-40-6
)
Alvocidib is a synthetic dihydroxyflavone that is 5,7-dihydroxyflavone which is subst
AG-270
(Catalog# : 25176, Cas# :
2201056-66-6
)
MAT2A 抑制剂 AG-270 是一种口服的蛋氨酸腺苷转移酶 II α (MAT2A) 小分
AZD-5904
(Catalog# : 181121, Cas# :
618913-30-7
)
AZD5904是一个有效的口服生物利用率MPO抑制剂。在临床前研究中,AZ
ALT-007
(Catalog# : 25157, Cas# :
2035010-37-6
)
ALT-007 是一种口服生物可利用的 SPT 抑制剂,比多球菌素更有效,